WO1997008178B1 - Nouveaux bisphosphonates, procede pour leur preparation et compositions pharmaceutiques les contenant - Google Patents
Nouveaux bisphosphonates, procede pour leur preparation et compositions pharmaceutiques les contenantInfo
- Publication number
- WO1997008178B1 WO1997008178B1 PCT/IL1996/000087 IL9600087W WO9708178B1 WO 1997008178 B1 WO1997008178 B1 WO 1997008178B1 IL 9600087 W IL9600087 W IL 9600087W WO 9708178 B1 WO9708178 B1 WO 9708178B1
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- designates
- preparation
- pharmaceutical compositions
- compounds
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Abstract
L'invention concerne des composés bisphosphonates, leur préparation et des compositions pharmaceutiques contenant de tels composés en tant qu'ingrédients actifs. Ces compositions s'administrent généralement par voie orale et elles permettent de traiter efficacement les anomalies du métabolisme du calcium. Les composés préférés comportent un cycle du type 2-aminopyrimidine. Il a été trouvé que des composés hétérocycliques similaires, substitués ou non, ont une activité similaire.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU68357/96A AU6835796A (en) | 1995-08-23 | 1996-08-22 | Novel bisphosphonates, process for their preparation and pharmaceutical compositions containing them |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IL11504195A IL115041A0 (en) | 1995-08-23 | 1995-08-23 | Novel bisphosphonates process for their preparation and pharmaceutical compositions containing them |
| IL115041 | 1995-08-23 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO1997008178A1 WO1997008178A1 (fr) | 1997-03-06 |
| WO1997008178B1 true WO1997008178B1 (fr) | 1997-05-01 |
Family
ID=11067907
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/IL1996/000087 Ceased WO1997008178A1 (fr) | 1995-08-23 | 1996-08-22 | Nouveaux bisphosphonates, procede pour leur preparation et compositions pharmaceutiques les contenant |
Country Status (3)
| Country | Link |
|---|---|
| AU (1) | AU6835796A (fr) |
| IL (1) | IL115041A0 (fr) |
| WO (1) | WO1997008178A1 (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1802641B8 (fr) | 2004-10-08 | 2012-03-07 | The Board Of Trustees Of The University Of Illinois | Composes de bisphosphonate et methodes de traitement de maladies de resorption osseuse, de cancers, de douleurs osseuses, de troubles immunitaires et de maladies infectieuses |
| US8012949B2 (en) | 2004-10-08 | 2011-09-06 | The Board Of Trustees Of The University Of Illinois | Bisphosphonate compounds and methods with enhanced potency for multiple targets including FPPS, GGPPS, and DPPS |
| AU2007226964B2 (en) | 2006-03-17 | 2012-03-22 | The Board Of Trustees Of The University Of Illinois | Bisphosphonate compounds and methods |
| CN102453050B (zh) * | 2010-11-03 | 2015-01-07 | 成都云克药业有限责任公司 | 一种二膦酸化合物及其制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3776880D1 (de) * | 1986-11-21 | 1992-04-02 | Ciba Geigy Ag | Neue substituierte alkandiphosphonsaeuren. |
| CA2136819A1 (fr) * | 1992-05-29 | 1993-12-09 | Frank H. Ebetino | Composes phosphonate a azote quaternaire pour traiter le metabolisme anormal du calcium et du phosphate |
| TW401276B (en) * | 1993-10-07 | 2000-08-11 | Zeneca Ltd | Novel compounds and a method of controlling growth of plants |
-
1995
- 1995-08-23 IL IL11504195A patent/IL115041A0/xx unknown
-
1996
- 1996-08-22 WO PCT/IL1996/000087 patent/WO1997008178A1/fr not_active Ceased
- 1996-08-22 AU AU68357/96A patent/AU6835796A/en not_active Abandoned
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