UY27206A1 - METHOD OF TREATMENT OF CONDITIONS OR DEMELINIZING DISEASES - Google Patents
METHOD OF TREATMENT OF CONDITIONS OR DEMELINIZING DISEASESInfo
- Publication number
- UY27206A1 UY27206A1 UY27206A UY27206A UY27206A1 UY 27206 A1 UY27206 A1 UY 27206A1 UY 27206 A UY27206 A UY 27206A UY 27206 A UY27206 A UY 27206A UY 27206 A1 UY27206 A1 UY 27206A1
- Authority
- UY
- Uruguay
- Prior art keywords
- treatment
- diseases
- conditions
- demelinizing
- vasculocerebral
- Prior art date
Links
- 201000010099 disease Diseases 0.000 title abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 206010069632 Bladder dysfunction Diseases 0.000 abstract 1
- 206010005052 Bladder irritation Diseases 0.000 abstract 1
- 108090000746 Chymosin Proteins 0.000 abstract 1
- 208000002193 Pain Diseases 0.000 abstract 1
- ZLMJMSJWJFRBEC-UHFFFAOYSA-N Potassium Chemical compound [K] ZLMJMSJWJFRBEC-UHFFFAOYSA-N 0.000 abstract 1
- 102000004257 Potassium Channel Human genes 0.000 abstract 1
- 108010052164 Sodium Channels Proteins 0.000 abstract 1
- 102000018674 Sodium Channels Human genes 0.000 abstract 1
- 208000030886 Traumatic Brain injury Diseases 0.000 abstract 1
- 230000000903 blocking effect Effects 0.000 abstract 1
- 229940080701 chymosin Drugs 0.000 abstract 1
- 230000003210 demyelinating effect Effects 0.000 abstract 1
- 230000007794 irritation Effects 0.000 abstract 1
- 201000006417 multiple sclerosis Diseases 0.000 abstract 1
- GNOLWGAJQVLBSM-UHFFFAOYSA-N n,n,5,7-tetramethyl-1,2,3,4-tetrahydronaphthalen-1-amine Chemical compound C1=C(C)C=C2C(N(C)C)CCCC2=C1C GNOLWGAJQVLBSM-UHFFFAOYSA-N 0.000 abstract 1
- JULKLMOOTJHVHH-UHFFFAOYSA-N n-pyridin-2-ylindol-1-amine Chemical class C1=CC2=CC=CC=C2N1NC1=CC=CC=N1 JULKLMOOTJHVHH-UHFFFAOYSA-N 0.000 abstract 1
- 208000004296 neuralgia Diseases 0.000 abstract 1
- 208000021722 neuropathic pain Diseases 0.000 abstract 1
- 229910052700 potassium Inorganic materials 0.000 abstract 1
- 239000011591 potassium Substances 0.000 abstract 1
- 108020001213 potassium channel Proteins 0.000 abstract 1
- 208000020431 spinal cord injury Diseases 0.000 abstract 1
- 230000009529 traumatic brain injury Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
N-(Piridinil)-1H-indól-1-aminas de fórmula (I) proveen una singular combinación de propiedades de bloqueo tanto de los canales de potasio como los de sodio. Estos compuestos son útiles para el tratamiento de condiciones y enfermedades desmielinizantes tales como esclerosis múltiple, lesiones de la médula espinal, lesiones traumáticas del cerebro y accidentes vásculocerebrales. Los compuestos son útiles para la rehabilitación de los accidentes vásculocerebrales, para el tratamiento de disfunción e irritación de la vejiga, y para el tratamiento de dolores neuropáticos y dolores inducidos por quimosina.N- (Pyridinyl) -1H-indole-1-amines of formula (I) provide a unique combination of blocking properties of both potassium and sodium channels. These compounds are useful for the treatment of demyelinating conditions and diseases such as multiple sclerosis, spinal cord injuries, traumatic brain injuries and vasculocerebral accidents. The compounds are useful for the rehabilitation of vasculocerebral accidents, for the treatment of bladder dysfunction and irritation, and for the treatment of neuropathic pain and chymosin-induced pain.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UY27206A UY27206A1 (en) | 2002-03-13 | 2002-03-13 | METHOD OF TREATMENT OF CONDITIONS OR DEMELINIZING DISEASES |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UY27206A UY27206A1 (en) | 2002-03-13 | 2002-03-13 | METHOD OF TREATMENT OF CONDITIONS OR DEMELINIZING DISEASES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY27206A1 true UY27206A1 (en) | 2002-07-31 |
Family
ID=38812602
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY27206A UY27206A1 (en) | 2002-03-13 | 2002-03-13 | METHOD OF TREATMENT OF CONDITIONS OR DEMELINIZING DISEASES |
Country Status (1)
| Country | Link |
|---|---|
| UY (1) | UY27206A1 (en) |
-
2002
- 2002-03-13 UY UY27206A patent/UY27206A1/en unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| DESI | Application deemed to be withdrawn |
Effective date: 20111121 |