UY26900A1 - BICYCLIC HETEROCICLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION - Google Patents
BICYCLIC HETEROCICLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATIONInfo
- Publication number
- UY26900A1 UY26900A1 UY26900A UY26900A UY26900A1 UY 26900 A1 UY26900 A1 UY 26900A1 UY 26900 A UY26900 A UY 26900A UY 26900 A UY26900 A UY 26900A UY 26900 A1 UY26900 A1 UY 26900A1
- Authority
- UY
- Uruguay
- Prior art keywords
- preparation
- bicyclic
- heterocicles
- employment
- procedures
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000004022 Protein-Tyrosine Kinases Human genes 0.000 abstract 1
- 108090000412 Protein-Tyrosine Kinases Proteins 0.000 abstract 1
- 125000002618 bicyclic heterocycle group Chemical group 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 210000004072 lung Anatomy 0.000 abstract 1
- 150000007522 mineralic acids Chemical class 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
- 235000005985 organic acids Nutrition 0.000 abstract 1
- 230000000144 pharmacologic effect Effects 0.000 abstract 1
- 210000002345 respiratory system Anatomy 0.000 abstract 1
- 230000019491 signal transduction Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención se refiere a heterociclos bicíclicos de la fórmula general (I) en la que Ra a Rc´ A a E y X están definidos como en la reivindicación 1, a sus tautómeros, sus estereoisómeros y sus sales, en particular sus sales fisiológicamente compatibles con ácidos o bases inorgánicos u orgánicos, que presentan valiosas propiedades farmacológicas, en particular un efecto inhibidor sobre la transducción de senales inducida por tirosino-quinasas, a su empleo para el tratamiento de enfermedades, en particular de enfermedades tumorales, de enfermedades de los pulmones y de las vías respiratorias, y a su preparación.The present invention relates to bicyclic heterocycles of the general formula (I) in which Ra to Rc 'A to E and X are defined as in claim 1, their tautomers, their stereoisomers and their salts, in particular their physiologically salts compatible with inorganic or organic acids or bases, which have valuable pharmacological properties, in particular an inhibitory effect on tyrosine kinase-induced signal transduction, for use in the treatment of diseases, in particular of tumor diseases, of diseases of the lungs and respiratory tract, and its preparation.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UY26900A UY26900A1 (en) | 2001-08-23 | 2001-08-23 | BICYCLIC HETEROCICLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UY26900A UY26900A1 (en) | 2001-08-23 | 2001-08-23 | BICYCLIC HETEROCICLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY26900A1 true UY26900A1 (en) | 2002-03-22 |
Family
ID=38812492
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY26900A UY26900A1 (en) | 2001-08-23 | 2001-08-23 | BICYCLIC HETEROCICLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION |
Country Status (1)
| Country | Link |
|---|---|
| UY (1) | UY26900A1 (en) |
-
2001
- 2001-08-23 UY UY26900A patent/UY26900A1/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20140908 |