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UY26648A1 - Inhibidores de vasopeptidasa para tratar hipertensión sistólica aislada - Google Patents

Inhibidores de vasopeptidasa para tratar hipertensión sistólica aislada

Info

Publication number
UY26648A1
UY26648A1 UY26648A UY26648A UY26648A1 UY 26648 A1 UY26648 A1 UY 26648A1 UY 26648 A UY26648 A UY 26648A UY 26648 A UY26648 A UY 26648A UY 26648 A1 UY26648 A1 UY 26648A1
Authority
UY
Uruguay
Prior art keywords
systolic hypertension
isolated systolic
vasopeptidase inhibitors
treat isolated
vasopeptidase
Prior art date
Application number
UY26648A
Other languages
English (en)
Inventor
Richard A Reeves
Robert A Wolf
Paul I Chang
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of UY26648A1 publication Critical patent/UY26648A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Se describen los inhibidores de vasopeptidasa especialmente el omapatrilat, que son útiles en el tratamiento de la hipertensión sistólica aislada. El inhibidor de la vasopeptidasa puede ser utilizado en combinación con otros agentes farmacéuticamente activos.
UY26648A 2000-04-03 2001-04-02 Inhibidores de vasopeptidasa para tratar hipertensión sistólica aislada UY26648A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19449900P 2000-04-03 2000-04-03

Publications (1)

Publication Number Publication Date
UY26648A1 true UY26648A1 (es) 2001-11-30

Family

ID=22717832

Family Applications (1)

Application Number Title Priority Date Filing Date
UY26648A UY26648A1 (es) 2000-04-03 2001-04-02 Inhibidores de vasopeptidasa para tratar hipertensión sistólica aislada

Country Status (8)

Country Link
US (1) US20020004500A1 (es)
EP (1) EP1267855A2 (es)
JP (1) JP2003533440A (es)
AU (1) AU2001287289A1 (es)
CA (1) CA2405496A1 (es)
PE (1) PE20011316A1 (es)
UY (1) UY26648A1 (es)
WO (1) WO2001074348A2 (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1303501B1 (en) * 2000-07-13 2005-09-21 Alteon, Inc. Cyanomethyl substituted thiazoliums and imidazoliums and treatments of disorders associated with protein aging
US6777443B2 (en) 2001-05-15 2004-08-17 Novartis Ag Dipeptide derivatives
JP2005516940A (ja) * 2001-12-20 2005-06-09 ブリストル−マイヤーズ スクイブ カンパニー 高血圧患者に対する血管ペプチダーゼ阻害剤投与による脈圧と血管硬化度の低下
US7468390B2 (en) 2002-01-17 2008-12-23 Novartis Ag Methods of treatment and pharmaceutical composition
IL162661A0 (en) * 2002-01-17 2005-11-20 Novartis Ag Pharmaceutical compositions comprising valsartan and nep inhibitors
EP1750862B1 (en) * 2004-06-04 2011-01-05 Teva Pharmaceutical Industries Ltd. Pharmaceutical composition containing irbesartan
WO2007045663A2 (en) * 2005-10-19 2007-04-26 Novartis Ag Combination of an ati receptor antagonist and a np inhibitor fro treating ia hypertension and heartfailure
AR057882A1 (es) 2005-11-09 2007-12-26 Novartis Ag Compuestos de accion doble de bloqueadores del receptor de angiotensina e inhibidores de endopeptidasa neutra
JP7180673B2 (ja) 2017-11-28 2022-11-30 アナベックス ライフ サイエンス コーポレイション シグマ-1受容体アゴニスト収縮期血圧療法

Also Published As

Publication number Publication date
AU2001287289A1 (en) 2001-10-15
CA2405496A1 (en) 2001-10-11
US20020004500A1 (en) 2002-01-10
WO2001074348A2 (en) 2001-10-11
WO2001074348A8 (en) 2002-05-23
JP2003533440A (ja) 2003-11-11
PE20011316A1 (es) 2002-01-13
EP1267855A2 (en) 2003-01-02

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20130218