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US20170266205A1 - Inducing lactation in nursing females - Google Patents

Inducing lactation in nursing females Download PDF

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Publication number
US20170266205A1
US20170266205A1 US15/479,009 US201715479009A US2017266205A1 US 20170266205 A1 US20170266205 A1 US 20170266205A1 US 201715479009 A US201715479009 A US 201715479009A US 2017266205 A1 US2017266205 A1 US 2017266205A1
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US
United States
Prior art keywords
cream
canceled
androgen
stanozolol
improvement
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
US15/479,009
Inventor
Edward M. Lichten
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Priority to US15/479,009 priority Critical patent/US20170266205A1/en
Publication of US20170266205A1 publication Critical patent/US20170266205A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels

Definitions

  • the cream for the treatment of HSDD in women.
  • the cream thereof is directed to causing a local physiological effect that stimulates the vagal nerves to mediate the neuropeptides that are linked to the brain for controlling oxytocin release.
  • a topical cream which when applied to the nipple(s) of a nursing female, induces increased lactation.
  • the cream generally, comprises: (a) a base cream having from about 0.5% to about 10%, by volume, of a steroid, based upon the total volume of the cream; and (b) preferably, at least about 1% to about 10% by volume, of the steroid, based on the total volume of the cream.
  • the steroid used herein is preferably an androgen and, most preferably, stanozolol.
  • the cream hereof generally, comprises: (a) a base cream having from about 0.5% to about 10%, by volume, of a steroid, based upon the total volume of the cream; and (b) preferably, from at least about 1% to about 10% by volume, of a steroid, based on the total volume of the cream.
  • the steroid used herein is, preferably, an androgen and, is selected from the group consisting of, stanozolol, danazol and furazobol.
  • a commercially available base cream is used.
  • Commercially available base creams include emollients, water, alcohols, such as isopropyl alcohol and benzyl alcohol, glycerol, fragrances, moisturizers and the like as well as mixtures thereof.
  • a particularly preferred base cream is that sold under the mark Lipoderm.
  • Lipoderm is reported as having two forms, Lipoderm Ultra and Lipoderm Y, each, comprising a proprietary blend of yohimbine HCl, caffeine, synephrine, acetyl L-carntine, lechithin, sesamin, octopamine HCl and ascorbyl palmitate.
  • base cream may be used alone or in admixture with other creams such as commercially available face creams, body moisturizing creams and the like, as well as mixtures thereof.
  • base cream and other additional cream may be used in any amount up to about a 50:50 volumetric mixture thereof of base cream to additional cream.
  • the androgen which is, preferably, stanozolol, is present in an amount ranging from about 0.5% to about 10%, by volume, based on the total volume of the topical cream. It should be noted that other steroids, such as danazol, furazobol, and the like may be used in lieu of the stanozolol, while effective, they are to a lesser degree.
  • the stanozolol is used alone, although it may be used in conjunction with the danazol and/or the furazobol.
  • the danazol or furazobol may be substituted for the stanozolol in the same amounts as the stanozolol.
  • the stanozolol cream hereof is prepared by admixing, at room temperature, the base cream and the stanozolol. Any other ingredients or adjuvants, where used, are added thereto and stirred to form a homogenous composition.
  • stanozolol releases testosterone which triggers a spinothalmic tract which, in turn, activates oxytocin related axons from the brain and, thus, serves as a neuropeptide mediator.
  • the stanozolol minimizes the effect of the sex hormone binding globulin in the cell wall.
  • the cream is applied to a nipple prior to breast feeding.
  • the cream is left on the nipple for about five to about twenty minutes and, usually, for about five to about fifteen minutes.
  • a nursing mother having a six-month old child with the ability to achieve adequate lactation has applied a 2 ml quantity of a Lubriderm Ultra cream having two percent, by volume, stanozolol added thereto.
  • the so-applied cream is left on for about two minutes. It is then washed off.

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

A topical cream applied to a nipple of a lactating female induces lactation. The cream comprises a base cream having from about 0.5% to about 10%, by volume, of a steroid, based upon the total volume of the cream. The preferred steroid is stanozolol. Preferably, the cream comprises at least about 1% to about 10%, by volume, of stanozolol, based on the total volume of the cream.

Description

    CROSS REFERENCE TO RELATED APPLICATION
  • This application is a completion application and claims the benefit of co-pending U.S. Provisional Patent Application Ser. No. 61/935,598, filed Feb. 4, 2014 for “Induction of Lactation in Nursing Females” and is related to the subject matter of co-pending U.S. patent application Ser. No. 13/745,934, filed Jan. 21, 2013, the disclosures of both are hereby incorporated by reference in their entireties.
  • BACKGROUND OF THE INVENTION
  • In the above-referenced related application there is disclosed the use of a topical cream for the treatment of HSDD in women. As disclosed, the cream thereof is directed to causing a local physiological effect that stimulates the vagal nerves to mediate the neuropeptides that are linked to the brain for controlling oxytocin release.
  • It has now been found that the cream thereof generates an increase in the release of oxytocin in nursing females. The oxytocin release causes an induction of lactation.
  • SUMMARY OF THE INVENTION
  • In accordance herewith there is provided a topical cream, which when applied to the nipple(s) of a nursing female, induces increased lactation.
  • The cream, generally, comprises: (a) a base cream having from about 0.5% to about 10%, by volume, of a steroid, based upon the total volume of the cream; and (b) preferably, at least about 1% to about 10% by volume, of the steroid, based on the total volume of the cream.
  • The steroid used herein is preferably an androgen and, most preferably, stanozolol.
  • For a more complete understanding of the present invention, reference is made to the following detailed description and the accompanying example.
  • DESCRIPTION OF THE INVENTION
  • As noted above, the cream hereof, generally, comprises: (a) a base cream having from about 0.5% to about 10%, by volume, of a steroid, based upon the total volume of the cream; and (b) preferably, from at least about 1% to about 10% by volume, of a steroid, based on the total volume of the cream.
  • The steroid used herein is, preferably, an androgen and, is selected from the group consisting of, stanozolol, danazol and furazobol.
  • More particularly, in preparing the topical cream hereof, a commercially available base cream is used. Commercially available base creams, as is known to the skilled artisan, include emollients, water, alcohols, such as isopropyl alcohol and benzyl alcohol, glycerol, fragrances, moisturizers and the like as well as mixtures thereof.
  • A particularly preferred base cream is that sold under the mark Lipoderm. Lipoderm is reported as having two forms, Lipoderm Ultra and Lipoderm Y, each, comprising a proprietary blend of yohimbine HCl, caffeine, synephrine, acetyl L-carntine, lechithin, sesamin, octopamine HCl and ascorbyl palmitate.
  • It should be noted that the base cream may be used alone or in admixture with other creams such as commercially available face creams, body moisturizing creams and the like, as well as mixtures thereof.
  • Where used the base cream and other additional cream may be used in any amount up to about a 50:50 volumetric mixture thereof of base cream to additional cream.
  • The androgen, which is, preferably, stanozolol, is present in an amount ranging from about 0.5% to about 10%, by volume, based on the total volume of the topical cream. It should be noted that other steroids, such as danazol, furazobol, and the like may be used in lieu of the stanozolol, while effective, they are to a lesser degree.
  • Preferably, the stanozolol is used alone, although it may be used in conjunction with the danazol and/or the furazobol.
  • Also, as noted above, the danazol or furazobol may be substituted for the stanozolol in the same amounts as the stanozolol.
  • The stanozolol cream hereof is prepared by admixing, at room temperature, the base cream and the stanozolol. Any other ingredients or adjuvants, where used, are added thereto and stirred to form a homogenous composition.
  • It is hypothesized that there is a local physiological effect whereby stanozolol releases testosterone which triggers a spinothalmic tract which, in turn, activates oxytocin related axons from the brain and, thus, serves as a neuropeptide mediator. Concomitantly the stanozolol minimizes the effect of the sex hormone binding globulin in the cell wall. These effects induce lactation when the cream is applied to a women's nipple prior to nursing.
  • In use, the cream is applied to a nipple prior to breast feeding. Generally, the cream is left on the nipple for about five to about twenty minutes and, usually, for about five to about fifteen minutes.
  • It is then removed by washing. Then the mother is then ready to being nursing.
  • The utilization of the cream is continued, as needed, until adequate lactation is achieved.
  • For a more complete understanding of the present invention reference is made to the following illustrative Example. In the Example all parts are by volume, absent indications to the contrary.
  • EXAMPLE
  • A nursing mother having a six-month old child with the ability to achieve adequate lactation has applied a 2 ml quantity of a Lubriderm Ultra cream having two percent, by volume, stanozolol added thereto. The so-applied cream is left on for about two minutes. It is then washed off.
  • Thereafter, the mother reported an increase in milk production.
  • From the above, it is to be appreciated that there is described herein a topical cream which has a positive effect on women having a need to stimulate adequate lactation.

Claims (15)

Having, thus, described the invention what is claimed is:
1. (canceled)
2. (Canceled)
3. (Canceled)
4. (Canceled)
5. (Canceled)
6. (Canceled)
7. (Canceled)
8. (Canceled)
9. (Canceled)
10. (Canceled)
11. In a topical cream for inducing lactation in a female of the type which is applied to at least one nipple, the improvement which comprises:
an effective amount of an androgen consisting essentially of an androgen-containing topical cream, the cream comprising: (a) an androgen and a blend of yohimbine HCL, caffeine, synephrine, acetyl L-carnitine, lecithin, sesamin, octopamine HO2 and ascorbyl palmitate.
12. The improvement of claim 11 wherein the androgen is present in an amount ranging from about 1% to about 10%, by volume, based on the total volume of the cream.
13. The improvement of claim 12 which further includes an additional cream selected from the group consisting of face creams and body moisturizing creams.
14. The improvement of claim 13 wherein the androgen is selected from the group consisting of stanozolol, danazol and furazabol.
15. The improvement of claim 14 wherein the androgen is stanozolol.
US15/479,009 2014-02-04 2017-04-04 Inducing lactation in nursing females Abandoned US20170266205A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
US15/479,009 US20170266205A1 (en) 2014-02-04 2017-04-04 Inducing lactation in nursing females

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461935598P 2014-02-04 2014-02-04
US14/613,741 US9610296B2 (en) 2013-01-21 2015-02-04 Inducing lactation in nursing females
US15/479,009 US20170266205A1 (en) 2014-02-04 2017-04-04 Inducing lactation in nursing females

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
US14/613,741 Division US9610296B2 (en) 2012-01-19 2015-02-04 Inducing lactation in nursing females

Publications (1)

Publication Number Publication Date
US20170266205A1 true US20170266205A1 (en) 2017-09-21

Family

ID=53753910

Family Applications (2)

Application Number Title Priority Date Filing Date
US14/613,741 Expired - Fee Related US9610296B2 (en) 2012-01-19 2015-02-04 Inducing lactation in nursing females
US15/479,009 Abandoned US20170266205A1 (en) 2014-02-04 2017-04-04 Inducing lactation in nursing females

Family Applications Before (1)

Application Number Title Priority Date Filing Date
US14/613,741 Expired - Fee Related US9610296B2 (en) 2012-01-19 2015-02-04 Inducing lactation in nursing females

Country Status (1)

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US (2) US9610296B2 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016201286A1 (en) * 2015-06-11 2016-12-15 Applied Biology, Inc. Treatment of sexual dysfunction
CN112999156B (en) * 2021-03-03 2023-09-08 宁波御坊堂生物科技有限公司 Erection-assisting time-delay essential oil spray with synergistic yohimbine hydrochloride and preparation method thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2589898A (en) * 1948-04-03 1952-03-18 American Dairies Inc Method of stimulating the growth of mammary glands and lobulealveolar system of mammals
WO1998008547A1 (en) * 1996-08-29 1998-03-05 Sekisui Kagaku Kogyo Kabushiki Kaisha Stanozolol-containing percutaneously absorbable preparation
US20070207197A1 (en) * 2006-02-13 2007-09-06 Villarreal J A Composition and method for reducing symptoms of breast engorgement
US20090202645A1 (en) * 2008-02-08 2009-08-13 Acme Drugs S.R.L. Intrasynovial formulations of stanozolol

Also Published As

Publication number Publication date
US9610296B2 (en) 2017-04-04
US20150216880A1 (en) 2015-08-06

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