[go: up one dir, main page]

UA99521C2 - Quinuclidine derivatives as m3 muscarinic receptor antagonists - Google Patents

Quinuclidine derivatives as m3 muscarinic receptor antagonists

Info

Publication number
UA99521C2
UA99521C2 UAA201013072A UAA201013072A UA99521C2 UA 99521 C2 UA99521 C2 UA 99521C2 UA A201013072 A UAA201013072 A UA A201013072A UA A201013072 A UAA201013072 A UA A201013072A UA 99521 C2 UA99521 C2 UA 99521C2
Authority
UA
Ukraine
Prior art keywords
receptor antagonists
muscarinic receptor
quinuclidine derivatives
pharmaceutical compositions
quinuclidine
Prior art date
Application number
UAA201013072A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Ронан Ли Форд
Эндрю Найджел Метер
Антонио Мете
Ричард Джеймс Булл
Элизабет Анн Скидмор
Original Assignee
Астразенека Аб
Пульмаген Терапеутикс (Синерджи) Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Астразенека Аб, Пульмаген Терапеутикс (Синерджи) Лимитед filed Critical Астразенека Аб
Priority to UAA201013072A priority Critical patent/UA99521C2/en
Publication of UA99521C2 publication Critical patent/UA99521C2/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

The invention provides named compounds of formula (I), wherein R4 is a N-substituted quinuclidine (1) pharmaceutical compositions containing them and a process for preparing the pharmaceutical compositions. Their use in therapy for the treatment of conditions mediated by M3 muscarinic receptors, such as clironic obstructive pulmonary disease is also disclosed.(I)
UAA201013072A 2008-05-13 2008-05-13 Quinuclidine derivatives as m3 muscarinic receptor antagonists UA99521C2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UAA201013072A UA99521C2 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as m3 muscarinic receptor antagonists

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
UAA201013072A UA99521C2 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as m3 muscarinic receptor antagonists

Publications (1)

Publication Number Publication Date
UA99521C2 true UA99521C2 (en) 2012-08-27

Family

ID=50849609

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201013072A UA99521C2 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as m3 muscarinic receptor antagonists

Country Status (1)

Country Link
UA (1) UA99521C2 (en)

Similar Documents

Publication Publication Date Title
TNSN07164A1 (en) Quinuclidine derivatives and their use as muscarinic m3 receptor antagonists
MX2010012189A (en) Quinuclidine derivatives as muscarinic m3 receptor antagonists.
IN2012DN02968A (en)
IL204064A (en) 4-formylpiperazine-1-carboxamidine compounds useful as muscarinic receptor antagonists
MX2009004780A (en) Quiniclidine derivatives of (hetero) arylcycloheptanecarboxylic acid as muscarinic receptor antagonists.
GEP20135744B (en) Quinuclidine carbonate derivatives and medicinal compositions containing the same
MX2009006018A (en) Quinuclidinol derivatives as muscarinic receptor antagonists.
NO20076060L (en) Piperidin-4-yl amide derivatives and their use as SST receptor subtype 5 antagonists
MXPA05011739A (en) Quinuclidine derivatives binding to mucarinic m3 receptors.
SI2875011T1 (en) 5-ht3 receptor antagonists
MX353209B (en) D2 ANTAGONISTS, METHODS OF SYNTHESIS and METHODS OF USE.
MX2009008527A (en) Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists.
MX2009008323A (en) Heterocyclic derivatives as m3 muscarinic receptors.
IL202236A0 (en) Prolinamide derivatives as nk3 antagonists
UA98772C2 (en) Cyclopropyl amine derivatives as histamin h3 receptor modulators
IL195747A0 (en) Pyrimidine and quinazoline derivatives as modulators of somatostatine receptor activity
MX2009012518A (en) 4,4-disubstituted piperidine derivatives.
EA200501594A1 (en) SUBSTITUTED DERIVATIVES OF AZABICOLOGEXANE AS ANTAGONISTS OF MUSCARINE RECEPTOR
MX2012007005A (en) Bicyclic thiazoles as allosteric modulators of mglur5 receptors.
MX2007007720A (en) Pyrrolinidium derivatives as m3 muscarinic receptors.
MX2009006757A (en) 4-(heterocyclyl)alkyl-n-(arylsulfonyl) indole compounds and their use as 5-ht6 ligands.
MX2009005242A (en) 5, 6, or 7-substituted-3-(hetero)arylisoquinolinamine derivatives and therapeutic use thereof.
MX2013001988A (en) Heterocyclyl compounds as histamine h3 receptor ligands
UA88910C2 (en) Heterocyclic compounds for treatment or reduction of diseases associated with the cannabinoid receptor and processes for the preparation thereof
NZ600536A (en) Bicyclic compounds as alpha4 beta2 nicotinic acetylcholine receptor ligands