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UA94031C2 - Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищей - Google Patents

Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищей

Info

Publication number
UA94031C2
UA94031C2 UAA200703512A UAA200703512A UA94031C2 UA 94031 C2 UA94031 C2 UA 94031C2 UA A200703512 A UAA200703512 A UA A200703512A UA A200703512 A UAA200703512 A UA A200703512A UA 94031 C2 UA94031 C2 UA 94031C2
Authority
UA
Ukraine
Prior art keywords
meal
sustained
achieve
release effect
dosage forms
Prior art date
Application number
UAA200703512A
Other languages
English (en)
Ukrainian (uk)
Inventor
Хенинг Блуме
Эрнст Мутчлер
Вернер Вайтчис
Original Assignee
Аристокон Фервальтунгс-Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Аристокон Фервальтунгс-Гмбх filed Critical Аристокон Фервальтунгс-Гмбх
Publication of UA94031C2 publication Critical patent/UA94031C2/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/485Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Изобретение касается препарата с непрерывным (постоянным) высвобождением для перорального применения вместе с пищей, который содержит, по крайней мере, один фармацевтически активный ингредиент (АРЕ), и, по необходимости, один или более фармацевтически применимых наполнителей, и дополнительно содержит, по крайней мере, один карбонат как газообразующий агент и, по крайней мере, одну кислоту, при этом карбонат и кислота обеспечивают гомогенное смешивание активного фармацевтического ингредиента с содержимым желудка.
UAA200703512A 2004-08-31 2005-08-30 Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищей UA94031C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004042139A DE102004042139B4 (de) 2004-08-31 2004-08-31 Perorale Darreichungsformen zur Erzielung eines Retardierungseffektes nach der Arzneimitteleinnahme mit einer Mahlzeit

Publications (1)

Publication Number Publication Date
UA94031C2 true UA94031C2 (ru) 2011-04-11

Family

ID=35745691

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200703512A UA94031C2 (ru) 2004-08-31 2005-08-30 Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищей

Country Status (7)

Country Link
US (1) US20090010906A1 (ru)
EP (1) EP1814512A2 (ru)
JP (1) JP2008511585A (ru)
DE (1) DE102004042139B4 (ru)
EA (1) EA013429B1 (ru)
UA (1) UA94031C2 (ru)
WO (1) WO2006024638A2 (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007041588A1 (de) * 2007-09-01 2009-03-05 Lts Lohmann Therapie-Systeme Ag Arzneimittel mit Hefe
CN103142552A (zh) * 2013-02-22 2013-06-12 广州科的信医药技术有限公司 一种洛伐他汀肠溶缓释微丸胶囊及其制备方法

Family Cites Families (31)

* Cited by examiner, † Cited by third party
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GB1139991A (en) * 1965-07-19 1969-01-15 Armour Pharma Stabilized enzyme composition
GB1573487A (en) * 1977-05-23 1980-08-28 Bristol Myers Co Bile acid binding composition
CA1182049A (en) * 1981-07-13 1985-02-05 Francis J. Sterbenz Apap antacid composition
EP0205336B1 (en) * 1985-06-11 1991-09-11 Teijin Limited Oral sustained release pharmaceutical preparation
JPS61286322A (ja) * 1985-06-12 1986-12-16 Teijin Ltd 経口徐放性製剤
DE3543999A1 (de) * 1985-12-13 1987-06-19 Bayer Ag Hochreine acarbose
JPS62195323A (ja) * 1986-02-24 1987-08-28 Eisai Co Ltd 胃内滞留型粒子
JPS62207209A (ja) * 1986-03-07 1987-09-11 Teijin Ltd 経口徐放性製剤
US4929605A (en) * 1987-10-07 1990-05-29 Merrell Dow Pharmaceuticals Inc. Pharmaceutical composition for piperidinoalkanol derivatives
US5096714A (en) * 1988-06-28 1992-03-17 Hauser-Kuhrts, Inc. Prolonged release drug tablet formulations
US5004651A (en) * 1989-01-24 1991-04-02 Abbott Laboratories Stabilizing system for solid dosage forms
US4975281A (en) * 1989-01-30 1990-12-04 E. R. Squibb & Sons, Inc. Anti-ulcer composition
CA2030449A1 (en) * 1989-11-22 1991-05-23 Eric H. Kuhrts Prolonged release drug tablet formulations
GB9025372D0 (en) * 1990-11-22 1991-01-09 Nat Res Dev Pharmaceutical dosage forms
US5683719A (en) * 1990-11-22 1997-11-04 British Technology Group Limited Controlled release compositions
IE77165B1 (en) * 1991-01-30 1997-12-03 Wellcome Found Water-dispersible tablet containing acyclovir
YU48263B (sh) * 1991-06-17 1997-09-30 Byk Gulden Lomberg Chemische Fabrik Gmbh. Postupak za dobijanje farmaceutskog preparata na bazi pantoprazola
HU9203780D0 (en) * 1991-12-12 1993-03-29 Sandoz Ag Stabilized pharmaceutical products of hmg-coa reductase inhibitor and method for producing them
GB9224021D0 (en) * 1992-11-16 1993-01-06 Boots Co Plc Effervescent compositions
US6645988B2 (en) * 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US6071539A (en) * 1996-09-20 2000-06-06 Ethypharm, Sa Effervescent granules and methods for their preparation
US6649186B1 (en) * 1996-09-20 2003-11-18 Ethypharm Effervescent granules and methods for their preparation
GB9704524D0 (en) * 1997-03-05 1997-04-23 Smithkline Beecham Plc Composition
US20010046473A1 (en) * 1997-04-18 2001-11-29 Jerome Besse Gastric-retained pharmaceutical composition and method for its use
US6235311B1 (en) * 1998-03-18 2001-05-22 Bristol-Myers Squibb Company Pharmaceutical composition containing a combination of a statin and aspirin and method
SI0976395T1 (sl) * 1998-07-30 2006-04-30 Merck Sante Sas Tableta s podaljsanim sproscanjem zdravilne ucinkovine v zelodcu
MXPA01002634A (es) * 1998-09-14 2002-06-04 Ranbaxy Lab Ltd Sistema de entrega que controla a una droga oralmente administrada proporcionando control en tiempo y espacial.
WO2001010405A1 (en) * 1999-08-04 2001-02-15 Ranbaxy Laboratories Limited Hydrodynamically balanced oral drug delivery system
GB0114069D0 (en) * 2001-06-08 2001-08-01 Smithkline Beecham Plc Composition
WO2003011255A1 (en) * 2001-07-04 2003-02-13 Sun Pharmaceutical Industries Limited Gastric retention controlled drug delivery system
AU2002302890A1 (en) * 2002-02-04 2003-12-02 Ranbaxy Laboratories Limited Hydrodynamically balancing oral drug delivery system with biphasic release

Also Published As

Publication number Publication date
EA013429B1 (ru) 2010-04-30
DE102004042139A1 (de) 2006-03-02
EA200700524A1 (ru) 2007-08-31
EP1814512A2 (de) 2007-08-08
DE102004042139B4 (de) 2009-06-10
JP2008511585A (ja) 2008-04-17
US20090010906A1 (en) 2009-01-08
WO2006024638A2 (de) 2006-03-09
WO2006024638A3 (de) 2007-04-05

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