UA94031C2 - Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищей - Google Patents
Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищейInfo
- Publication number
- UA94031C2 UA94031C2 UAA200703512A UAA200703512A UA94031C2 UA 94031 C2 UA94031 C2 UA 94031C2 UA A200703512 A UAA200703512 A UA A200703512A UA A200703512 A UAA200703512 A UA A200703512A UA 94031 C2 UA94031 C2 UA 94031C2
- Authority
- UA
- Ukraine
- Prior art keywords
- meal
- sustained
- achieve
- release effect
- dosage forms
- Prior art date
Links
- 235000012054 meals Nutrition 0.000 title abstract 2
- 238000013268 sustained release Methods 0.000 title abstract 2
- 239000012730 sustained-release form Substances 0.000 title abstract 2
- 239000002552 dosage form Substances 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 230000000694 effects Effects 0.000 title 1
- 239000013543 active substance Substances 0.000 abstract 3
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 210000003736 gastrointestinal content Anatomy 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/485—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Изобретение касается препарата с непрерывным (постоянным) высвобождением для перорального применения вместе с пищей, который содержит, по крайней мере, один фармацевтически активный ингредиент (АРЕ), и, по необходимости, один или более фармацевтически применимых наполнителей, и дополнительно содержит, по крайней мере, один карбонат как газообразующий агент и, по крайней мере, одну кислоту, при этом карбонат и кислота обеспечивают гомогенное смешивание активного фармацевтического ингредиента с содержимым желудка.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004042139A DE102004042139B4 (de) | 2004-08-31 | 2004-08-31 | Perorale Darreichungsformen zur Erzielung eines Retardierungseffektes nach der Arzneimitteleinnahme mit einer Mahlzeit |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA94031C2 true UA94031C2 (ru) | 2011-04-11 |
Family
ID=35745691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200703512A UA94031C2 (ru) | 2004-08-31 | 2005-08-30 | Препарат для перорального применения с непрерывным (постоянным) высвобождением при приеме фармацевтически активного ингредиента вместе с пищей |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20090010906A1 (ru) |
| EP (1) | EP1814512A2 (ru) |
| JP (1) | JP2008511585A (ru) |
| DE (1) | DE102004042139B4 (ru) |
| EA (1) | EA013429B1 (ru) |
| UA (1) | UA94031C2 (ru) |
| WO (1) | WO2006024638A2 (ru) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102007041588A1 (de) * | 2007-09-01 | 2009-03-05 | Lts Lohmann Therapie-Systeme Ag | Arzneimittel mit Hefe |
| CN103142552A (zh) * | 2013-02-22 | 2013-06-12 | 广州科的信医药技术有限公司 | 一种洛伐他汀肠溶缓释微丸胶囊及其制备方法 |
Family Cites Families (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1139991A (en) * | 1965-07-19 | 1969-01-15 | Armour Pharma | Stabilized enzyme composition |
| GB1573487A (en) * | 1977-05-23 | 1980-08-28 | Bristol Myers Co | Bile acid binding composition |
| CA1182049A (en) * | 1981-07-13 | 1985-02-05 | Francis J. Sterbenz | Apap antacid composition |
| EP0205336B1 (en) * | 1985-06-11 | 1991-09-11 | Teijin Limited | Oral sustained release pharmaceutical preparation |
| JPS61286322A (ja) * | 1985-06-12 | 1986-12-16 | Teijin Ltd | 経口徐放性製剤 |
| DE3543999A1 (de) * | 1985-12-13 | 1987-06-19 | Bayer Ag | Hochreine acarbose |
| JPS62195323A (ja) * | 1986-02-24 | 1987-08-28 | Eisai Co Ltd | 胃内滞留型粒子 |
| JPS62207209A (ja) * | 1986-03-07 | 1987-09-11 | Teijin Ltd | 経口徐放性製剤 |
| US4929605A (en) * | 1987-10-07 | 1990-05-29 | Merrell Dow Pharmaceuticals Inc. | Pharmaceutical composition for piperidinoalkanol derivatives |
| US5096714A (en) * | 1988-06-28 | 1992-03-17 | Hauser-Kuhrts, Inc. | Prolonged release drug tablet formulations |
| US5004651A (en) * | 1989-01-24 | 1991-04-02 | Abbott Laboratories | Stabilizing system for solid dosage forms |
| US4975281A (en) * | 1989-01-30 | 1990-12-04 | E. R. Squibb & Sons, Inc. | Anti-ulcer composition |
| CA2030449A1 (en) * | 1989-11-22 | 1991-05-23 | Eric H. Kuhrts | Prolonged release drug tablet formulations |
| GB9025372D0 (en) * | 1990-11-22 | 1991-01-09 | Nat Res Dev | Pharmaceutical dosage forms |
| US5683719A (en) * | 1990-11-22 | 1997-11-04 | British Technology Group Limited | Controlled release compositions |
| IE77165B1 (en) * | 1991-01-30 | 1997-12-03 | Wellcome Found | Water-dispersible tablet containing acyclovir |
| YU48263B (sh) * | 1991-06-17 | 1997-09-30 | Byk Gulden Lomberg Chemische Fabrik Gmbh. | Postupak za dobijanje farmaceutskog preparata na bazi pantoprazola |
| HU9203780D0 (en) * | 1991-12-12 | 1993-03-29 | Sandoz Ag | Stabilized pharmaceutical products of hmg-coa reductase inhibitor and method for producing them |
| GB9224021D0 (en) * | 1992-11-16 | 1993-01-06 | Boots Co Plc | Effervescent compositions |
| US6645988B2 (en) * | 1996-01-04 | 2003-11-11 | Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
| US6071539A (en) * | 1996-09-20 | 2000-06-06 | Ethypharm, Sa | Effervescent granules and methods for their preparation |
| US6649186B1 (en) * | 1996-09-20 | 2003-11-18 | Ethypharm | Effervescent granules and methods for their preparation |
| GB9704524D0 (en) * | 1997-03-05 | 1997-04-23 | Smithkline Beecham Plc | Composition |
| US20010046473A1 (en) * | 1997-04-18 | 2001-11-29 | Jerome Besse | Gastric-retained pharmaceutical composition and method for its use |
| US6235311B1 (en) * | 1998-03-18 | 2001-05-22 | Bristol-Myers Squibb Company | Pharmaceutical composition containing a combination of a statin and aspirin and method |
| SI0976395T1 (sl) * | 1998-07-30 | 2006-04-30 | Merck Sante Sas | Tableta s podaljsanim sproscanjem zdravilne ucinkovine v zelodcu |
| MXPA01002634A (es) * | 1998-09-14 | 2002-06-04 | Ranbaxy Lab Ltd | Sistema de entrega que controla a una droga oralmente administrada proporcionando control en tiempo y espacial. |
| WO2001010405A1 (en) * | 1999-08-04 | 2001-02-15 | Ranbaxy Laboratories Limited | Hydrodynamically balanced oral drug delivery system |
| GB0114069D0 (en) * | 2001-06-08 | 2001-08-01 | Smithkline Beecham Plc | Composition |
| WO2003011255A1 (en) * | 2001-07-04 | 2003-02-13 | Sun Pharmaceutical Industries Limited | Gastric retention controlled drug delivery system |
| AU2002302890A1 (en) * | 2002-02-04 | 2003-12-02 | Ranbaxy Laboratories Limited | Hydrodynamically balancing oral drug delivery system with biphasic release |
-
2004
- 2004-08-31 DE DE102004042139A patent/DE102004042139B4/de not_active Expired - Fee Related
-
2005
- 2005-08-30 WO PCT/EP2005/054260 patent/WO2006024638A2/de not_active Ceased
- 2005-08-30 EA EA200700524A patent/EA013429B1/ru not_active IP Right Cessation
- 2005-08-30 EP EP05775898A patent/EP1814512A2/de not_active Withdrawn
- 2005-08-30 US US11/574,317 patent/US20090010906A1/en not_active Abandoned
- 2005-08-30 JP JP2007528874A patent/JP2008511585A/ja active Pending
- 2005-08-30 UA UAA200703512A patent/UA94031C2/ru unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EA013429B1 (ru) | 2010-04-30 |
| DE102004042139A1 (de) | 2006-03-02 |
| EA200700524A1 (ru) | 2007-08-31 |
| EP1814512A2 (de) | 2007-08-08 |
| DE102004042139B4 (de) | 2009-06-10 |
| JP2008511585A (ja) | 2008-04-17 |
| US20090010906A1 (en) | 2009-01-08 |
| WO2006024638A2 (de) | 2006-03-09 |
| WO2006024638A3 (de) | 2007-04-05 |
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