UA90912C2 - Cgrp antagonists, method for the production thereof and their use as medicaments - Google Patents
Cgrp antagonists, method for the production thereof and their use as medicamentsInfo
- Publication number
- UA90912C2 UA90912C2 UAA200803272A UAA200803272A UA90912C2 UA 90912 C2 UA90912 C2 UA 90912C2 UA A200803272 A UAA200803272 A UA A200803272A UA A200803272 A UAA200803272 A UA A200803272A UA 90912 C2 UA90912 C2 UA 90912C2
- Authority
- UA
- Ukraine
- Prior art keywords
- production
- salts
- medicaments
- cgrp antagonists
- hydrates
- Prior art date
Links
- 229940127597 CGRP antagonist Drugs 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000004677 hydrates Chemical class 0.000 abstract 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- YZCKVEUIGOORGS-OUBTZVSYSA-N Deuterium Chemical compound [2H] YZCKVEUIGOORGS-OUBTZVSYSA-N 0.000 abstract 1
- 229910052805 deuterium Inorganic materials 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 150000007522 mineralic acids Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
- 235000005985 organic acids Nutrition 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The invention relates to the CGRP antagonists of general formula (I) in which R, R, Rand Rare defined as in claim 1, to their tautomers, isomers, diastereoisomers and enantiomers, hydrates, mixtures and their salts as well as the hydrates of the salts, particularly their physiologically compatible salts with inorganic or organic acids or bases, as well as to the compounds of general formula (I) in which one or more hydrogen atoms are exchanged for deuterium, to medicaments containing these compounds, the use thereof and to methods for the production thereof.(I),
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005038831A DE102005038831A1 (en) | 2005-08-17 | 2005-08-17 | New N-acylalkoxycarbonyl-piperidine derivatives, useful as CGRP antagonists, for treating e.g. headaches, cardiovascular disease, skin disorders, morphine tolerance, and inflammatory diseases such as osteoarthritis and allergic rhinitis |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA90912C2 true UA90912C2 (en) | 2010-06-10 |
Family
ID=40391426
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200803272A UA90912C2 (en) | 2005-08-17 | 2006-08-15 | Cgrp antagonists, method for the production thereof and their use as medicaments |
Country Status (3)
| Country | Link |
|---|---|
| CN (1) | CN101365693A (en) |
| UA (1) | UA90912C2 (en) |
| ZA (1) | ZA200711114B (en) |
-
2006
- 2006-08-15 CN CNA2006800317640A patent/CN101365693A/en active Pending
- 2006-08-15 UA UAA200803272A patent/UA90912C2/en unknown
-
2007
- 2007-12-20 ZA ZA200711114A patent/ZA200711114B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200711114B (en) | 2009-07-29 |
| CN101365693A (en) | 2009-02-11 |
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