UA86083C2 - Pyrazole-substituted aminoheteroaryl compounds as protein kinase inhibitors - Google Patents
Pyrazole-substituted aminoheteroaryl compounds as protein kinase inhibitorsInfo
- Publication number
- UA86083C2 UA86083C2 UAA200701932A UAA200701932A UA86083C2 UA 86083 C2 UA86083 C2 UA 86083C2 UA A200701932 A UAA200701932 A UA A200701932A UA A200701932 A UAA200701932 A UA A200701932A UA 86083 C2 UA86083 C2 UA 86083C2
- Authority
- UA
- Ukraine
- Prior art keywords
- protein kinase
- pyrazole
- kinase inhibitors
- aminoheteroaryl compounds
- compounds
- Prior art date
Links
- 125000005214 aminoheteroaryl group Chemical class 0.000 title 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 title 1
- 239000003909 protein kinase inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000008022 Proto-Oncogene Proteins c-met Human genes 0.000 abstract 1
- 108010089836 Proto-Oncogene Proteins c-met Proteins 0.000 abstract 1
- 230000002159 abnormal effect Effects 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 230000010261 cell growth Effects 0.000 abstract 1
- 208000037824 growth disorder Diseases 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Изобретение касается соединений формулы 1, 1а также способов их синтеза и применения. Преобладающие соединения представляют собой эффективные ингибиторы c-Met протеинкиназы и используются при лечении заболеваний патологического клеточного роста, таких как раковые опухоли.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US60524404P | 2004-08-26 | 2004-08-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA86083C2 true UA86083C2 (en) | 2009-03-25 |
Family
ID=50557632
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200701932A UA86083C2 (en) | 2004-08-26 | 2005-08-15 | Pyrazole-substituted aminoheteroaryl compounds as protein kinase inhibitors |
Country Status (1)
| Country | Link |
|---|---|
| UA (1) | UA86083C2 (ru) |
-
2005
- 2005-08-15 UA UAA200701932A patent/UA86083C2/ru unknown
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