UA84594C2 - 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists - Google Patents
1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonistsInfo
- Publication number
- UA84594C2 UA84594C2 UAA200609435A UAA200609435A UA84594C2 UA 84594 C2 UA84594 C2 UA 84594C2 UA A200609435 A UAA200609435 A UA A200609435A UA A200609435 A UAA200609435 A UA A200609435A UA 84594 C2 UA84594 C2 UA 84594C2
- Authority
- UA
- Ukraine
- Prior art keywords
- pyrazole derivatives
- trisubstituted
- dihydro
- antagonists
- compounds
- Prior art date
Links
- -1 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole Chemical class 0.000 title abstract 2
- 229940124802 CB1 antagonist Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000009286 beneficial effect Effects 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 150000003217 pyrazoles Chemical class 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Изобретение относится к 1,3,5-тризамещенным производным 4,5-дигидро-1Н-пиразола как антагонистам СВ, способам получения этих соединений и новым промежуточным соединениям, пригодным для синтеза указанных производных пиразола. Изобретение также относится к применению указанных соединений для получения лекарственного средства, которое дает терапевтический эффект. Соединения имеют общую формулу (І)где значения соответствующих заместителей указаны в описании.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UAA200609435A UA84594C2 (en) | 2005-01-27 | 2005-01-27 | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UAA200609435A UA84594C2 (en) | 2005-01-27 | 2005-01-27 | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA84594C2 true UA84594C2 (en) | 2008-11-10 |
Family
ID=50180792
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200609435A UA84594C2 (en) | 2005-01-27 | 2005-01-27 | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |
Country Status (1)
| Country | Link |
|---|---|
| UA (1) | UA84594C2 (ru) |
-
2005
- 2005-01-27 UA UAA200609435A patent/UA84594C2/ru unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL176547A0 (en) | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity | |
| MX2009013592A (es) | Proceso para la preparacion de pirazoles. | |
| TNSN06409A1 (en) | Novel fluoroglycoside derivatives of pyrazoles, medicaments containing these compounds, and the use thereof | |
| WO2009016460A3 (en) | Pyrazole compounds and their use as raf inhibitors | |
| UA94833C2 (en) | Substituted bicyclolactams | |
| MX2007007845A (es) | Sulfonilpirrolidinas, metodo para producir las mismas y su uso como medicamento. | |
| MX2009007713A (es) | Derivados de piridazina, procedimientos para su preparacion y su uso como fungicidas. | |
| WO2005087771A3 (de) | 5,6-dialkyl-7-amino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel | |
| WO2009121033A3 (en) | Substituted nitrogen heterocycles and synthesis and uses thereof | |
| WO2010056644A8 (en) | 1-(arylsulfonyl)-4-(piperazin-1-yl)-1h-benzimidazoles as 5-hydroxytryptamine-6 ligands | |
| WO2009116074A3 (en) | Substituted benzimidazoles as cannabinoid modulator | |
| TNSN07006A1 (en) | Novel heterocyclic compounds | |
| MY147502A (en) | Substituted pyrazoles, compositions containing these, method of production and use | |
| ATE411296T1 (de) | Imidazolinderivate mit cb1-antagonistischer wirkung | |
| UA100862C2 (ru) | Шестичленные ароматические соединения, их получение и применение (варианты) | |
| TW200714598A (en) | Urea derivatives, methods for their manufacture, and uses therefor | |
| TW200745039A (en) | Isotopically substituted pantoprazole | |
| GB0513886D0 (en) | Novel compounds | |
| TW200716564A (en) | Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents | |
| TW200640911A (en) | Novel, long acting betamimetics for the treatment of respiratory diseases | |
| WO2008059513A3 (en) | Compounds suitable as modulators of hdl | |
| PL1745010T3 (pl) | Podstawione pochodne cykloheksylo-1,4-diaminy | |
| TW200621703A (en) | Alkylidene-tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents | |
| TW200619201A (en) | Process for the preparation of pyrazoles | |
| UA84594C2 (en) | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |