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UA83311C2 - 3-aminocyclopentanecarboxamides as modulators of chemokine receptors - Google Patents

3-aminocyclopentanecarboxamides as modulators of chemokine receptors

Info

Publication number
UA83311C2
UA83311C2 UAA200613944A UAA200613944A UA83311C2 UA 83311 C2 UA83311 C2 UA 83311C2 UA A200613944 A UAA200613944 A UA A200613944A UA A200613944 A UAA200613944 A UA A200613944A UA 83311 C2 UA83311 C2 UA 83311C2
Authority
UA
Ukraine
Prior art keywords
modulators
aminocyclopentanecarboxamides
chemokine receptors
compounds
chemokine
Prior art date
Application number
UAA200613944A
Other languages
English (en)
Ukrainian (uk)
Inventor
Чу-Бяо Сюе
Чаншен Чжен
Хао Фен
Майкл Ксиа
Джозеф Гленн
Ганьфен Цао
Original Assignee
Инсайт Корпорейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Инсайт Корпорейшн filed Critical Инсайт Корпорейшн
Publication of UA83311C2 publication Critical patent/UA83311C2/ru

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    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/14—Nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Diabetes (AREA)
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  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
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  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
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  • Tropical Medicine & Parasitology (AREA)
  • Child & Adolescent Psychology (AREA)
  • AIDS & HIV (AREA)
  • Transplantation (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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Abstract

Данное изобретение касается соединений формулы І, которые являются модуляторами хемокиновых рецепторов. Соединение по данному изобретению и его композиция полезны при лечении заболеваний, связанных с экспрессией и/или активностью хемокинового рецептора.I
UAA200613944A 2004-06-28 2005-06-27 3-aminocyclopentanecarboxamides as modulators of chemokine receptors UA83311C2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US58348204P 2004-06-28 2004-06-28
US62448104P 2004-11-01 2004-11-01
PCT/US2005/022909 WO2006004741A2 (en) 2004-06-28 2005-06-27 3-aminocyclopentanecarboxamides as modulators of chemokine receptors

Publications (1)

Publication Number Publication Date
UA83311C2 true UA83311C2 (en) 2008-06-25

Family

ID=35783315

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200613944A UA83311C2 (en) 2004-06-28 2005-06-27 3-aminocyclopentanecarboxamides as modulators of chemokine receptors

Country Status (22)

Country Link
US (2) US7618970B2 (ru)
EP (1) EP1763347A4 (ru)
JP (2) JP4116671B2 (ru)
KR (1) KR100856155B1 (ru)
CN (1) CN102382088A (ru)
AP (1) AP2006003848A0 (ru)
AR (1) AR052215A1 (ru)
AU (1) AU2005259983B2 (ru)
BR (1) BRPI0512634A (ru)
CA (1) CA2571397C (ru)
CR (1) CR8759A (ru)
EA (1) EA012649B1 (ru)
EC (1) ECSP067121A (ru)
GE (1) GEP20094844B (ru)
IL (1) IL179735A0 (ru)
MA (1) MA28681B1 (ru)
MX (1) MXPA06014673A (ru)
NO (1) NO20070489L (ru)
NZ (1) NZ551673A (ru)
TW (1) TWI366458B (ru)
UA (1) UA83311C2 (ru)
WO (1) WO2006004741A2 (ru)

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Also Published As

Publication number Publication date
TWI366458B (en) 2012-06-21
WO2006004741A3 (en) 2006-05-04
AR052215A1 (es) 2007-03-07
AU2005259983B2 (en) 2011-07-28
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