TW349100B - Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines - Google Patents

Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines

Info

Publication number: TW349100B
Authority: TW; Taiwan
Prior art keywords: hydrogen; represent; alkyl; thiazolylimidazo; thienodiazepines
Prior art date: 1994-11-11

Application number

TW084110653A

Other languages

English (en)

Inventor

Bernd Buttelmann

Thierry Godel

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-11-11

Filing date

1995-10-11

Publication date

1999-01-01

1995-10-11 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1999-01-01 Application granted granted Critical

1999-01-01 Publication of TW349100B publication Critical patent/TW349100B/zh

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

TW084110653A 1994-11-11 1995-10-11 Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines TW349100B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH338694		1994-11-11
CH226195		1995-08-04

Publications (1)

Publication Number	Publication Date
TW349100B true TW349100B (en)	1999-01-01

Family

ID=25689945

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TW084110653A TW349100B (en)	1994-11-11	1995-10-11	Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines

Country Status (12)

Country	Link
US (2)	US5885986A (zh)
EP (1)	EP0790999A1 (zh)
JP (1)	JP2989013B2 (zh)
CN (1)	CN1046519C (zh)
AU (1)	AU3982695A (zh)
BR (1)	BR9509711A (zh)
FI (1)	FI971990A0 (zh)
IL (1)	IL115882A (zh)
MA (1)	MA23716A1 (zh)
MX (1)	MX9703288A (zh)
TW (1)	TW349100B (zh)
WO (1)	WO1996015129A1 (zh)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1648512A4 (en) *	2003-07-31	2009-01-21	Immunomedics Inc	ANTI-CD19 ANTIBODIES
WO2009024325A2 (en)	2007-08-20	2009-02-26	Evotec Neurosciences Gmbh	Treatment of sleep disorders
US20090054412A1 (en) *	2007-08-20	2009-02-26	John Alan Kemp	Treatment of Sleep Disorders
AU2017313753B2 (en)	2016-08-16	2022-01-27	The Trustees Of Columbia University In The City Of New York	GABA(A) receptor modulators and methods to control airway hyperresponsiveness and inflammation in asthma
CN111285878B (zh) *	2020-04-03	2022-05-13	杭州新博思生物医药有限公司	二氮杂卓类化合物及制法与其药用盐、前药和用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1143728A (en) *	1979-10-04	1983-03-29	Max Gerecke	Imidazodiazepine derivatives
DE3587913D1 (de) *	1984-01-19	1994-10-06	Hoffmann La Roche	Imidazodiazepin-Derivate.
AU587802B2 (en) *	1985-03-08	1989-08-31	Ferrosan A/S	Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
US4771051A (en) *	1985-05-17	1988-09-13	A/S Ferrosan	3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
TW201311B (zh) *	1991-06-17	1993-03-01	Hoffmann La Roche
CA2143246C (en) *	1994-03-16	2000-08-22	Thierry Godel	Imidazodiazepines

1995
- 1995-10-11 TW TW084110653A patent/TW349100B/zh active
- 1995-11-06 IL IL11588295A patent/IL115882A/en not_active IP Right Cessation
- 1995-11-08 US US08/817,665 patent/US5885986A/en not_active Expired - Fee Related
- 1995-11-08 EP EP95938437A patent/EP0790999A1/en not_active Withdrawn
- 1995-11-08 JP JP8515709A patent/JP2989013B2/ja not_active Expired - Lifetime
- 1995-11-08 MX MX9703288A patent/MX9703288A/es not_active Application Discontinuation
- 1995-11-08 AU AU39826/95A patent/AU3982695A/en not_active Abandoned
- 1995-11-08 BR BR9509711A patent/BR9509711A/pt not_active Application Discontinuation
- 1995-11-08 WO PCT/EP1995/004393 patent/WO1996015129A1/en not_active Ceased
- 1995-11-08 FI FI971990A patent/FI971990A0/fi unknown
- 1995-11-08 CN CN95196171A patent/CN1046519C/zh not_active Expired - Fee Related
- 1995-11-08 MA MA24061A patent/MA23716A1/fr unknown
1997
- 1997-11-25 US US08/978,351 patent/US5962450A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US5885986A (en)	1999-03-23
MA23716A1 (fr)	1996-07-01
IL115882A0 (en)	1996-01-31
EP0790999A1 (en)	1997-08-27
JPH10505098A (ja)	1998-05-19
CN1046519C (zh)	1999-11-17
FI971990A7 (fi)	1997-05-09
JP2989013B2 (ja)	1999-12-13
IL115882A (en)	1998-10-30
AU3982695A (en)	1996-06-06
CN1167487A (zh)	1997-12-10
US5962450A (en)	1999-10-05
WO1996015129A1 (en)	1996-05-23
BR9509711A (pt)	1997-09-30
MX9703288A (es)	1997-08-30
FI971990L (fi)	1997-05-09
FI971990A0 (fi)	1997-05-09

Publication	Publication Date	Title
TW347387B (en)	1998-12-11	Piperidine derivatives
AU4950993A (en)	1994-03-29	Combination of germicidal agents
CA2086404A1 (en)	1993-07-01	Triazolopyrimidine derivatives
IL108731A (en)	1997-03-18	6, N-DISUBSTITUTED-£1, 2, 4\| TRIAZOLO-£1, 5-a\| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
CA2339272A1 (en)	2000-03-02	Nitrogen-containing heterocyclic carboxamide derivatives or salts thereof and antiviral agents comprising the same
GB2208294B (en)	1991-04-24	Cyclosporins
AU8794291A (en)	1992-05-21	New oxazolopyridine derivatives, processes for preparing these and pharmaceutical compositions containing them
MX9606331A (es)	1997-03-29	Nuevos compuestos, procesos para la preparacion de los mismos y agentes antitumor.
EP0482410A3 (en)	1992-09-09	Anti-microbial compounds, including substituted 2-cyclohexyl-amine derivatives and their preparation
GR3030490T3 (en)	1999-10-29	Substituted biphenyl derivatives as phosphodiesterase inhibitors
MY104626A (en)	1994-04-30	A 1-phenylimidazole derivative and its production and use.
HUP9600071A2 (hu)	1998-09-28	Indolil-piperidin-származékok, e vegyületeket tartalmazó gyógyászati készítmények, eljárás előállításukra és alkalmazásuk
MY108541A (en)	1996-10-31	Purine derivatives and use thereof in therapy.
MX9700928A (es)	1997-04-30	Derivado de triazian y medicina que lo contiene.
MY131641A (en)	2007-08-30	Indoline derivatives, process of preparation and use
HUP9902256A1 (hu)	1999-10-28	Proteázgátló amidinoszármazékok, valamint e vegyületeket tartalmazó gyógyászati készítmények
TW349100B (en)	1999-01-01	Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines
MY117092A (en)	2004-05-31	Chemotherapeutic pyrrolocarbazole derivatives
GB2207433B (en)	1990-10-10	Acyclic cyclosporins
NZ240575A (en)	1993-07-27	N-benzoylproline derivatives and pharmaceutical compositions
GR3007118T3 (zh)	1993-07-30
TW328957B (en)	1998-04-01	Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation
TW333532B (en)	1998-06-11	Benzopyrans
MXPA02007973A (es)	2005-10-05	Compuestos de aminoacidos y su uso como inhibidores de nep, ace y ece.
TW327598B (en)	1998-03-01	N-acetonylbenzamide fungicides