TW200938233A - Oral dispersable tablet - Google Patents
Oral dispersable tablet Download PDFInfo
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- TW200938233A TW200938233A TW97146532A TW97146532A TW200938233A TW 200938233 A TW200938233 A TW 200938233A TW 97146532 A TW97146532 A TW 97146532A TW 97146532 A TW97146532 A TW 97146532A TW 200938233 A TW200938233 A TW 200938233A
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- Prior art keywords
- tablet
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- active agent
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- 239000013543 active substance Substances 0.000 claims abstract description 33
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims abstract description 10
- 239000004094 surface-active agent Substances 0.000 claims abstract description 9
- 239000003826 tablet Substances 0.000 claims description 40
- 239000003795 chemical substances by application Substances 0.000 claims description 24
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- 239000007937 lozenge Substances 0.000 claims description 13
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- 239000000203 mixture Substances 0.000 claims description 10
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- 230000000694 effects Effects 0.000 claims description 6
- 238000004519 manufacturing process Methods 0.000 claims description 6
- 150000003839 salts Chemical class 0.000 claims description 6
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
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- A—HUMAN NECESSITIES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
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- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07023802 | 2007-12-08 |
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| TW200938233A true TW200938233A (en) | 2009-09-16 |
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| TW97146532A TW200938233A (en) | 2007-12-08 | 2008-12-01 | Oral dispersable tablet |
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| EP (1) | EP2231126A2 (ru) |
| JP (2) | JP2011506279A (ru) |
| KR (1) | KR20100096140A (ru) |
| CN (1) | CN101888834A (ru) |
| BR (1) | BRPI0820861A2 (ru) |
| MX (1) | MX2010005175A (ru) |
| RU (1) | RU2010128019A (ru) |
| TW (1) | TW200938233A (ru) |
| WO (1) | WO2009071219A2 (ru) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| KR101560438B1 (ko) * | 2009-09-08 | 2015-10-14 | 교와 가가꾸고교 가부시키가이샤 | 제산ㆍ완하용 정제 |
| CN101797236B (zh) * | 2010-03-23 | 2012-05-23 | 西南大学 | 重酒石酸卡巴拉汀口腔崩解片及其制备方法 |
| EP2563329B1 (en) * | 2010-04-27 | 2017-04-12 | Bayer Intellectual Property GmbH | Orally disintegrating tablet containing acarbose |
| US20110300216A1 (en) * | 2010-06-03 | 2011-12-08 | First Eric R | Chewable, swallowable and effervescent solid dosage form for oral delivery of pharmaceutical actives |
| JP5750856B2 (ja) * | 2010-10-04 | 2015-07-22 | ライオン株式会社 | 固形医薬組成物及び医薬製剤 |
| KR101237646B1 (ko) * | 2010-12-09 | 2013-03-04 | 주식회사 드림파마 | 생체이용률이 개선된 셀레콕시브 함유 고체 분산체, 이를 포함하는 약학 조성물 및 이의 제조방법 |
| FR2968995B1 (fr) * | 2010-12-16 | 2013-03-22 | Sanofi Aventis | Composition pharmaceutioue pour une administration par voie orale destinee a eviter le mesusage |
| FR2968992B1 (fr) * | 2010-12-16 | 2013-02-08 | Sanofi Aventis | Comprime pharmaceutique orodispersible a base de zolpidem |
| TR201100150A2 (tr) * | 2011-01-06 | 2012-07-23 | Bi̇lgi̇ç Mahmut | Suda çözünür dozaj formları |
| WO2013115741A1 (en) * | 2012-01-31 | 2013-08-08 | Mahmut Bilgic | Pharmaceutical compositions comprising alpha-glucosidase inhibitor |
| CN102600149B (zh) * | 2012-02-02 | 2013-12-04 | 西藏易明西雅生物医药科技有限公司 | 一种治疗糖尿病的药物组合物 |
| HK1221915A1 (zh) * | 2013-07-19 | 2017-06-16 | Bayer Pharma Aktiengesellschaft | Api米格列醇的超快速崩解片剂配方 |
| EP3023109A4 (en) | 2013-07-19 | 2017-01-04 | Sanwa Kagaku Kenkyusho Co., Ltd | Orally disintegrating tablet |
| CN103877041B (zh) * | 2014-03-14 | 2016-07-06 | 崔书豪 | 一种吡罗昔康分散片及其制备方法 |
| JP6467071B2 (ja) | 2016-01-29 | 2019-02-06 | 小林 光 | 固形製剤、固形製剤の製造方法及び水素発生方法 |
| CN105640954B (zh) * | 2016-02-04 | 2019-03-05 | 青岛市海慈医疗集团 | 一种治疗消化不良的西沙必利片剂 |
| US10076494B2 (en) | 2016-06-16 | 2018-09-18 | Dexcel Pharma Technologies Ltd. | Stable orally disintegrating pharmaceutical compositions |
| CN107595788B (zh) * | 2016-07-11 | 2020-08-21 | 武汉朗来科技发展有限公司 | 一种用于口服固体制剂的复合崩解剂体系及含有该复合崩解剂体系的口服固体制剂 |
| CN110191860A (zh) | 2016-08-23 | 2019-08-30 | 小林光 | 调配物与其制造方法、及氢供给方法 |
| EP3505151A4 (en) | 2016-08-23 | 2020-03-11 | Hikaru Kobayashi | HYDROGEN SUPPLY MATERIAL AND MANUFACTURING METHOD THEREFOR, AND HYDROGEN SUPPLY PROCESS |
| CN107334742B (zh) * | 2017-08-18 | 2020-01-31 | 山东力诺制药有限公司 | 一种盐酸氟西汀分散片及其制备方法 |
| BR112020003077A2 (pt) * | 2017-09-28 | 2020-08-25 | Hanmi Pharm. Co., Ltd. | composição farmacêutica e método para preparar a composição farmacêutica |
| CN110840850B (zh) * | 2018-07-24 | 2023-03-17 | 烟台药物研究所 | 一种高生物利用度的塞来昔布冻干口崩片及其制备方法 |
| CN109864971B (zh) * | 2019-04-08 | 2021-12-17 | 西安远大德天药业股份有限公司 | 一种拉莫三嗪固体分散体的颗粒剂及其制备方法 |
| CN114224855B (zh) * | 2021-12-01 | 2023-11-28 | 北京悦康科创医药科技股份有限公司 | 一种甲磺酸多沙唑嗪口含片及其制备方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19802700A1 (de) * | 1998-01-24 | 1999-07-29 | Bayer Ag | Verfahren zur Herstellung einer im Mund schnell zerfallenden Arzneiform, die als Wirkstoff Acarbose enthält |
| PL373914A1 (en) * | 2002-02-01 | 2005-09-19 | Pfizer Products Inc. | Immediate release dosage forms containing solid drug dispersions |
| US20040265375A1 (en) * | 2003-04-16 | 2004-12-30 | Platteeuw Johannes J. | Orally disintegrating tablets |
| US7749533B2 (en) * | 2003-05-07 | 2010-07-06 | Akina, Inc. | Highly plastic granules for making fast melting tablets |
| US7230016B2 (en) * | 2003-05-13 | 2007-06-12 | Synthon Ip Inc. | Pioglitazone salts, such as pioglitazone sulfate, and pharmaceutical compositions and processes using the same |
| US20070196477A1 (en) * | 2004-04-30 | 2007-08-23 | Withiam Michael C | Rapidly dissolving tablets comprising low surface area calcium phosphates |
| US20070196474A1 (en) * | 2004-04-30 | 2007-08-23 | Withiam Michael C | Rapidly disintegrating low friability tablets comprising calcium carbonate |
| GB0423103D0 (en) * | 2004-10-19 | 2004-11-17 | Boots Healthcare Int Ltd | Therapeutic agents |
-
2008
- 2008-11-25 RU RU2010128019/15A patent/RU2010128019A/ru not_active Application Discontinuation
- 2008-11-25 JP JP2010536354A patent/JP2011506279A/ja active Pending
- 2008-11-25 EP EP08856436A patent/EP2231126A2/en not_active Withdrawn
- 2008-11-25 WO PCT/EP2008/009968 patent/WO2009071219A2/en not_active Ceased
- 2008-11-25 KR KR1020107012467A patent/KR20100096140A/ko not_active Withdrawn
- 2008-11-25 BR BRPI0820861-1A patent/BRPI0820861A2/pt not_active IP Right Cessation
- 2008-11-25 CN CN2008801194609A patent/CN101888834A/zh active Pending
- 2008-11-25 MX MX2010005175A patent/MX2010005175A/es not_active Application Discontinuation
- 2008-12-01 TW TW97146532A patent/TW200938233A/zh unknown
-
2014
- 2014-10-09 JP JP2014208122A patent/JP2015038123A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP2015038123A (ja) | 2015-02-26 |
| WO2009071219A3 (en) | 2009-09-11 |
| BRPI0820861A2 (pt) | 2015-06-16 |
| WO2009071219A2 (en) | 2009-06-11 |
| EP2231126A2 (en) | 2010-09-29 |
| MX2010005175A (es) | 2010-08-02 |
| RU2010128019A (ru) | 2012-01-20 |
| CN101888834A (zh) | 2010-11-17 |
| KR20100096140A (ko) | 2010-09-01 |
| JP2011506279A (ja) | 2011-03-03 |
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