TW200732337A - Organic compounds - Google Patents
Organic compoundsInfo
- Publication number
- TW200732337A TW200732337A TW095146173A TW95146173A TW200732337A TW 200732337 A TW200732337 A TW 200732337A TW 095146173 A TW095146173 A TW 095146173A TW 95146173 A TW95146173 A TW 95146173A TW 200732337 A TW200732337 A TW 200732337A
- Authority
- TW
- Taiwan
- Prior art keywords
- organic compounds
- pharmaceuticals
- preparing
- formula
- free
- Prior art date
Links
- 150000002894 organic compounds Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Pulmonology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0525144.2A GB0525144D0 (en) | 2005-12-09 | 2005-12-09 | Organic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW200732337A true TW200732337A (en) | 2007-09-01 |
Family
ID=35735863
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW095146173A TW200732337A (en) | 2005-12-09 | 2006-12-08 | Organic compounds |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US20080312229A1 (zh) |
| EP (1) | EP1960398B1 (zh) |
| JP (1) | JP2009518343A (zh) |
| KR (1) | KR20080065699A (zh) |
| CN (1) | CN101326185A (zh) |
| AR (1) | AR056887A1 (zh) |
| AT (1) | ATE482957T1 (zh) |
| AU (1) | AU2006322206B2 (zh) |
| BR (1) | BRPI0619529A2 (zh) |
| CA (1) | CA2630611A1 (zh) |
| DE (1) | DE602006017256D1 (zh) |
| GB (1) | GB0525144D0 (zh) |
| PE (1) | PE20071035A1 (zh) |
| PT (1) | PT1960398E (zh) |
| RU (1) | RU2008127439A (zh) |
| TW (1) | TW200732337A (zh) |
| WO (1) | WO2007065683A1 (zh) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY144903A (en) * | 2004-06-17 | 2011-11-30 | Novartis Ag | Pyrrolopyridine derivatives and their use as crth2 antagonists |
| GB0525143D0 (en) * | 2005-12-09 | 2006-01-18 | Novartis Ag | Organic compounds |
| SI2051962T1 (sl) | 2006-08-07 | 2012-02-29 | Actelion Pharmaceuticals Ltd | Derivati (3-amino-1,2,3,4-tetrahidro-9h-karbazol-9-il)-ocetne kisline |
| US8563573B2 (en) | 2007-11-02 | 2013-10-22 | Vertex Pharmaceuticals Incorporated | Azaindole derivatives as CFTR modulators |
| WO2009093029A1 (en) * | 2008-01-22 | 2009-07-30 | Oxagen Limited | Compounds having crth2 antagonist activity |
| CN108383789A (zh) * | 2010-01-27 | 2018-08-10 | 艾克提麦斯医药品有限公司 | 作为crth2拮抗剂的吡唑化合物 |
| DK2558447T3 (da) | 2010-03-22 | 2014-11-10 | Actelion Pharmaceuticals Ltd | 3-(heteroaryl-amino)-1,2,3,4-tetrahydro-9h-carbazolderivater og deres anvendelse som prostaglandin d2-receptormodulatorer |
| US8802868B2 (en) | 2010-03-25 | 2014-08-12 | Vertex Pharmaceuticals Incorporated | Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide |
| MX2012012204A (es) | 2010-04-22 | 2012-12-05 | Vertex Pharma | Proceso para producir compuestos de cicloalquilcarboxamido-indol. |
| EP2457900A1 (en) | 2010-11-25 | 2012-05-30 | Almirall, S.A. | New pyrazole derivatives having CRTh2 antagonistic behaviour |
| MY165623A (en) | 2011-04-14 | 2018-04-18 | Idorsia Pharmaceuticals Ltd | 7-(heteroaryl-amino)-6,7,8,9-tetrahydropyrido[1,2-a]indol acetic acid derivatives and their use as prostaglandin d2 receptor modulators |
| MX350516B (es) * | 2011-11-17 | 2017-09-08 | Kbp Biosciences Co Ltd | Compuestos de anillo fusionado que contienen nitrogeno como antagonistas crth2. |
| LT3119779T (lt) | 2014-03-17 | 2018-09-10 | Idorsia Pharmaceuticals Ltd | Azaindolo acto rūgšties dariniai ir jų panaudojimas kaip prostaglandino d2 receptoriaus moduliatorių |
| MX2016011900A (es) | 2014-03-18 | 2016-12-05 | Actelion Pharmaceuticals Ltd | Derivados de acido azaindol-acetico y su uso como moduladores del receptor de prostaglandina d2. |
| DK3925607T3 (da) | 2014-04-15 | 2023-08-21 | Vertex Pharma | Farmaceutiske sammensætninger til behandlingen af cystisk fibrosetransmembrankonduktansregulator-medierede sygdomme |
| CA2993893A1 (en) | 2015-09-15 | 2017-03-23 | Idorsia Pharmaceuticals Ltd | Crystalline forms |
| KR20200104291A (ko) | 2017-11-06 | 2020-09-03 | 랩트 테라퓨틱스, 인크. | 항암제 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3320268A (en) * | 1964-08-14 | 1967-05-16 | Merck & Co Inc | 1-aroyl or heteroaroyl-7-azaindole-3-carboxylates and derivatives |
| HUE026285T2 (en) * | 2003-02-06 | 2016-05-30 | Dompe Farm Spa | 2-arylacetic acid compounds and their derivatives and pharmaceutical compositions containing them |
| MY144903A (en) * | 2004-06-17 | 2011-11-30 | Novartis Ag | Pyrrolopyridine derivatives and their use as crth2 antagonists |
-
2005
- 2005-12-09 GB GBGB0525144.2A patent/GB0525144D0/en not_active Ceased
-
2006
- 2006-12-06 PE PE2006001570A patent/PE20071035A1/es not_active Application Discontinuation
- 2006-12-07 RU RU2008127439/04A patent/RU2008127439A/ru unknown
- 2006-12-07 AU AU2006322206A patent/AU2006322206B2/en not_active Ceased
- 2006-12-07 CN CNA2006800462767A patent/CN101326185A/zh active Pending
- 2006-12-07 US US12/096,453 patent/US20080312229A1/en not_active Abandoned
- 2006-12-07 PT PT06819000T patent/PT1960398E/pt unknown
- 2006-12-07 KR KR1020087013721A patent/KR20080065699A/ko not_active Abandoned
- 2006-12-07 CA CA002630611A patent/CA2630611A1/en not_active Abandoned
- 2006-12-07 BR BRPI0619529-6A patent/BRPI0619529A2/pt not_active IP Right Cessation
- 2006-12-07 DE DE602006017256T patent/DE602006017256D1/de active Active
- 2006-12-07 AT AT06819000T patent/ATE482957T1/de not_active IP Right Cessation
- 2006-12-07 AR ARP060105412A patent/AR056887A1/es unknown
- 2006-12-07 JP JP2008543732A patent/JP2009518343A/ja active Pending
- 2006-12-07 WO PCT/EP2006/011770 patent/WO2007065683A1/en not_active Ceased
- 2006-12-07 EP EP06819000A patent/EP1960398B1/en not_active Not-in-force
- 2006-12-08 TW TW095146173A patent/TW200732337A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ATE482957T1 (de) | 2010-10-15 |
| CN101326185A (zh) | 2008-12-17 |
| RU2008127439A (ru) | 2010-01-20 |
| CA2630611A1 (en) | 2007-06-14 |
| WO2007065683A1 (en) | 2007-06-14 |
| EP1960398A1 (en) | 2008-08-27 |
| AU2006322206A1 (en) | 2007-06-14 |
| US20080312229A1 (en) | 2008-12-18 |
| AU2006322206B2 (en) | 2010-08-19 |
| PE20071035A1 (es) | 2007-10-30 |
| KR20080065699A (ko) | 2008-07-14 |
| BRPI0619529A2 (pt) | 2011-10-04 |
| JP2009518343A (ja) | 2009-05-07 |
| PT1960398E (pt) | 2010-11-26 |
| EP1960398B1 (en) | 2010-09-29 |
| AR056887A1 (es) | 2007-10-31 |
| GB0525144D0 (en) | 2006-01-18 |
| DE602006017256D1 (de) | 2010-11-11 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| TW200732335A (en) | Organic compounds | |
| TW200617009A (en) | Organic compounds | |
| TW200635921A (en) | Organic compounds | |
| SG169989A1 (en) | Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof | |
| TW200800999A (en) | Novel compounds | |
| TW200732337A (en) | Organic compounds | |
| TW200745084A (en) | Novel compounds | |
| MX2009007713A (es) | Derivados de piridazina, procedimientos para su preparacion y su uso como fungicidas. | |
| TW200505920A (en) | Organic compounds | |
| TW200800967A (en) | Benzimidazole thiophene compounds | |
| DE602004024213D1 (en) | Aminopropanolderivate | |
| SE0401762D0 (sv) | Novel compounds | |
| TW200637837A (en) | Fungicides | |
| GB0412769D0 (en) | Organic compounds | |
| GB0508318D0 (en) | Organic compounds | |
| TW200508197A (en) | Indolone-acetamide derivatives, processes for preparing them and their uses | |
| ES2368594T3 (es) | Derivados sustituidos de ciclohexilmetilo. | |
| JO2734B1 (en) | Organic compounds | |
| TW200638930A (en) | Acetylene derivatives | |
| MXPA05013823A (es) | Derivados de pirrolidinio y piperidino como ligandos para el receptor m3 muscarinico. | |
| MY140739A (en) | 2, 6-quinolinyl derivatives, processes for preparing them and their uses | |
| GB0411929D0 (en) | Organic compounds | |
| BRPI0519292A2 (pt) | compostos orgÂnicos | |
| GB0508314D0 (en) | Organic compounds | |
| WO2007065684A3 (en) | Bicyclic heteroyclic compounds as antiinflammatory or antiallergic agents |