TR201000948A1 - Aripiprazol formülasyonları. - Google Patents
Aripiprazol formülasyonları.Info
- Publication number
- TR201000948A1 TR201000948A1 TR2010/00948A TR201000948A TR201000948A1 TR 201000948 A1 TR201000948 A1 TR 201000948A1 TR 2010/00948 A TR2010/00948 A TR 2010/00948A TR 201000948 A TR201000948 A TR 201000948A TR 201000948 A1 TR201000948 A1 TR 201000948A1
- Authority
- TR
- Turkey
- Prior art keywords
- aripiprazole formulations
- aripiprazole
- aripiprazole monohydrate
- formulations
- formulation
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 3
- 238000009472 formulation Methods 0.000 title abstract 2
- CEUORZQYGODEFX-UHFFFAOYSA-N Aripirazole Chemical compound ClC1=CC=CC(N2CCN(CCCCOC=3C=C4NC(=O)CCC4=CC=3)CC2)=C1Cl CEUORZQYGODEFX-UHFFFAOYSA-N 0.000 title 1
- 229960004372 aripiprazole Drugs 0.000 title 1
- UXQBDXJXIVDBTF-UHFFFAOYSA-N 7-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]-3,4-dihydro-1h-quinolin-2-one;hydrate Chemical compound O.ClC1=CC=CC(N2CCN(CCCCOC=3C=C4NC(=O)CCC4=CC=3)CC2)=C1Cl UXQBDXJXIVDBTF-UHFFFAOYSA-N 0.000 abstract 2
- 239000002270 dispersing agent Substances 0.000 abstract 1
- 238000004090 dissolution Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Buluş farmasötik bir formülasyon olup özelliği, aripiprazol monohidrat ile süper dağıtıcı ve dağıtıcı karışımı içermesi ile karakterize edilmektedir. Daha da özel olarak buluş aripiprazol monohidratın yüksek çözünürlüğe ve çözünme hızına, dolayısı ile yüksek biyoyararlanıma sahip formülasyonu ile ilgilidir.
Priority Applications (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2010/00948A TR201000948A1 (tr) | 2010-02-09 | 2010-02-09 | Aripiprazol formülasyonları. |
| PL11153639T PL2359816T3 (pl) | 2010-02-09 | 2011-02-08 | Formulacje aripiprazolu |
| EP11153639.7A EP2359816B1 (en) | 2010-02-09 | 2011-02-08 | Aripiprazole formulations |
| ES11153639.7T ES2607440T3 (es) | 2010-02-09 | 2011-02-08 | Formulaciones de aripiprazol |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2010/00948A TR201000948A1 (tr) | 2010-02-09 | 2010-02-09 | Aripiprazol formülasyonları. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201000948A1 true TR201000948A1 (tr) | 2011-08-22 |
Family
ID=42551366
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2010/00948A TR201000948A1 (tr) | 2010-02-09 | 2010-02-09 | Aripiprazol formülasyonları. |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP2359816B1 (tr) |
| ES (1) | ES2607440T3 (tr) |
| PL (1) | PL2359816T3 (tr) |
| TR (1) | TR201000948A1 (tr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JO3753B1 (ar) | 2011-10-14 | 2021-01-31 | Otsuka Pharma Co Ltd | قرص يتألف من 7-[4-(4-بينزو[بي]ثيوفين-4-ايل-ببرازين-1-1ايل)بوتكسيل]-1اتش-كوينولين-2-وان أو ملح منه |
| WO2013100878A1 (en) * | 2011-12-27 | 2013-07-04 | Mahmut Bilgic | Pharmaceutical formulations comprising aripiprazole |
| WO2014104989A1 (en) * | 2011-12-27 | 2014-07-03 | Mahmut Bilgic | Pharmaceutical compositions comprising aripiprazole |
| WO2013175508A2 (en) | 2012-05-24 | 2013-11-28 | Medreich Limited | Stable pharmaceutical composition of aripiprazole |
| WO2015067313A1 (en) * | 2013-11-07 | 2015-05-14 | Synthon B.V. | Orodispersible pharmaceutical compositions comprising aripiprazole |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003030868A1 (en) * | 2001-10-09 | 2003-04-17 | Bristol-Myers Squibb Company | Flashmelt oral dosage formulation |
| WO2006097344A1 (en) * | 2005-03-17 | 2006-09-21 | Synthon B.V. | Pharmaceutical tablets of crystalline type ii aripiprazole |
| WO2006105798A2 (en) * | 2005-07-11 | 2006-10-12 | Nycomed Danmark Aps | Benzimidazole formulation |
| US20070148100A1 (en) * | 2005-09-15 | 2007-06-28 | Elan Pharma International, Limited | Nanoparticulate aripiprazole formulations |
| EP1808165A1 (en) * | 2006-01-05 | 2007-07-18 | Teva Pharmaceutical Industries Ltd | Dry formulations of aripiprazole |
| WO2008020820A2 (en) * | 2006-08-15 | 2008-02-21 | Nobel Ilac Sanayii Ve Ticaret A.S. | Pharmaceutical compositions comprising aripiprazole |
| EP2082735A1 (en) * | 2008-01-23 | 2009-07-29 | Helm AG | Amorphous Aripiprazole and Process for the Preparation thereof |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5006528A (en) | 1988-10-31 | 1991-04-09 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
| MY129350A (en) | 2001-04-25 | 2007-03-30 | Bristol Myers Squibb Co | Aripiprazole oral solution |
| JP4310605B2 (ja) | 2001-05-25 | 2009-08-12 | 大塚製薬株式会社 | 医薬用組成物 |
| US20090198059A1 (en) | 2004-09-13 | 2009-08-06 | Chava Satyanarayana | Process for the preparation of polymorphs, solvates of aripiprazole using aripirazole acid salts |
| WO2006053781A1 (en) | 2004-11-18 | 2006-05-26 | Synthon B.V. | Process of making crystalline aripiprazole |
| WO2007113846A1 (en) | 2006-04-03 | 2007-10-11 | Alembic Limited | A process for the preparation of aripiprazole |
| EP1880714A1 (en) | 2006-07-20 | 2008-01-23 | Helm AG | Amorphous Aripiprazole and Process for the Preparation thereof |
| WO2010079506A2 (en) * | 2008-06-23 | 2010-07-15 | Torrent Pharmaceuticals Ltd. | Pharmaceutical composition of aripiprazole |
-
2010
- 2010-02-09 TR TR2010/00948A patent/TR201000948A1/tr unknown
-
2011
- 2011-02-08 PL PL11153639T patent/PL2359816T3/pl unknown
- 2011-02-08 EP EP11153639.7A patent/EP2359816B1/en active Active
- 2011-02-08 ES ES11153639.7T patent/ES2607440T3/es active Active
Patent Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003030868A1 (en) * | 2001-10-09 | 2003-04-17 | Bristol-Myers Squibb Company | Flashmelt oral dosage formulation |
| WO2006097344A1 (en) * | 2005-03-17 | 2006-09-21 | Synthon B.V. | Pharmaceutical tablets of crystalline type ii aripiprazole |
| WO2006105798A2 (en) * | 2005-07-11 | 2006-10-12 | Nycomed Danmark Aps | Benzimidazole formulation |
| US20070148100A1 (en) * | 2005-09-15 | 2007-06-28 | Elan Pharma International, Limited | Nanoparticulate aripiprazole formulations |
| EP1808165A1 (en) * | 2006-01-05 | 2007-07-18 | Teva Pharmaceutical Industries Ltd | Dry formulations of aripiprazole |
| WO2008020820A2 (en) * | 2006-08-15 | 2008-02-21 | Nobel Ilac Sanayii Ve Ticaret A.S. | Pharmaceutical compositions comprising aripiprazole |
| EP2082735A1 (en) * | 2008-01-23 | 2009-07-29 | Helm AG | Amorphous Aripiprazole and Process for the Preparation thereof |
Also Published As
| Publication number | Publication date |
|---|---|
| ES2607440T3 (es) | 2017-03-31 |
| EP2359816A1 (en) | 2011-08-24 |
| PL2359816T3 (pl) | 2017-04-28 |
| EP2359816B1 (en) | 2016-09-21 |
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