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TR200202129T2 - Yeni ikameli propenon türevlerinin hazırlanması için prosesler. - Google Patents

Yeni ikameli propenon türevlerinin hazırlanması için prosesler.

Info

Publication number
TR200202129T2
TR200202129T2 TR2002/02129T TR200202129T TR200202129T2 TR 200202129 T2 TR200202129 T2 TR 200202129T2 TR 2002/02129 T TR2002/02129 T TR 2002/02129T TR 200202129 T TR200202129 T TR 200202129T TR 200202129 T2 TR200202129 T2 TR 200202129T2
Authority
TR
Turkey
Prior art keywords
preparation
processes
derivatives
new substituted
substituted propane
Prior art date
Application number
TR2002/02129T
Other languages
English (en)
Inventor
Uenaka Masaaki
Kawata Kyozo
Nagai Masahiko
Endoh Takeshi
Original Assignee
Shionogi & Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co., Ltd. filed Critical Shionogi & Co., Ltd.
Publication of TR200202129T2 publication Critical patent/TR200202129T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/40—Radicals substituted by oxygen atoms
    • C07D307/46—Doubly bound oxygen atoms, or two oxygen atoms singly bound to the same carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Bu bulus, anti-HIV faaliyeti olan 2-asil-5-benzilfuran türevleri, 1, 2, 4-triazol-3-karbosiklik asit ester türevleri ve propenon türevlerinin ve bunlarin faydali kristallerinin hazirlanmasi sinai ve piyasaya yönelik prosesler sunmaktadir. R1, R2 ve R4'ün her birinin bagimsiz olarak hidrojen vb, A'nin CR6 veya N, R6'nin hidrojen vb, Q'nun bir koruma grubu ve L'nin bir ayrilan grup oldugu formül.
TR2002/02129T 1999-06-02 2000-05-29 Yeni ikameli propenon türevlerinin hazırlanması için prosesler. TR200202129T2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP15550399 1999-06-02
JP23030599 1999-08-17

Publications (1)

Publication Number Publication Date
TR200202129T2 true TR200202129T2 (tr) 2003-03-21

Family

ID=26483489

Family Applications (2)

Application Number Title Priority Date Filing Date
TR2002/02129T TR200202129T2 (tr) 1999-06-02 2000-05-29 Yeni ikameli propenon türevlerinin hazırlanması için prosesler.
TR2001/03801T TR200103801T2 (tr) 1999-06-02 2000-05-29 Yeni ikameli propenon türevlerinin hazırlanması için prosesler

Family Applications After (1)

Application Number Title Priority Date Filing Date
TR2001/03801T TR200103801T2 (tr) 1999-06-02 2000-05-29 Yeni ikameli propenon türevlerinin hazırlanması için prosesler

Country Status (10)

Country Link
US (1) US6831177B1 (tr)
EP (1) EP1186599A4 (tr)
KR (1) KR100423781B1 (tr)
CN (1) CN1367784A (tr)
AU (1) AU763231B2 (tr)
BR (1) BR0011246A (tr)
CA (1) CA2376043A1 (tr)
MX (1) MXPA01012299A (tr)
TR (2) TR200202129T2 (tr)
WO (1) WO2000075122A1 (tr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2370500A1 (en) * 1999-06-25 2001-01-04 Lekhanh O. Tran 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
IL153363A0 (en) * 2000-06-13 2003-07-06 Shionogi & Co Pharmaceutical compositions containing propenone derivatives
US20040157804A1 (en) 2002-10-16 2004-08-12 Gilead Sciences, Inc. Pre-organized tricyclic integrase inhibitor compounds
CA2537325A1 (en) 2003-09-19 2005-03-31 Gilead Sciences, Inc. Aza-quinolinol phosphonate integrase inhibitor compounds
WO2007054105A2 (en) * 2005-11-14 2007-05-18 H. Lundbeck A/S Method for the preparation of escitalopram
NZ572367A (en) 2006-05-16 2011-09-30 Gilead Sciences Inc Fused cyclic compounds as integrase inhibitors
AU2009206673B2 (en) 2008-01-25 2015-04-23 Chimerix, Inc. Methods of treating viral infections
CA2766643C (en) 2009-07-08 2017-01-03 Dermira (Canada), Inc. Tofa analogs useful in treating dermatological disorders or conditions
HUE032860T2 (en) 2010-02-12 2017-11-28 Chimerix Inc A method for treating a virus infection
BR112013000925A2 (pt) 2010-07-15 2020-12-01 Bayer Intellectual Property Gmbh compostos heterocíclicos como pesticidas
WO2014064697A1 (en) 2012-10-25 2014-05-01 Technion Research And Development Foundation Ltd. Method of treatment of disease

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1481990A (en) 1974-12-23 1977-08-03 May & Baker Ltd Herbicidal 3-benzyl-pyridazine derivatives
JPS5268182A (en) 1975-11-29 1977-06-06 Sumitomo Chem Co Ltd Preparation of novel triazole derivatives
JPS6153275A (ja) 1984-08-23 1986-03-17 Arakawa Chem Ind Co Ltd ２−アシルフラン系化合物の製法
GB2271566A (en) * 1992-10-14 1994-04-20 Merck & Co Inc HIV integrase inhibitors
JP2530102B2 (ja) 1993-07-14 1996-09-04 株式会社東芝 半導体ディスク装置およびその制御方法
JPH0778057A (ja) 1993-06-25 1995-03-20 Casio Comput Co Ltd プリンタ制御システム
WO1996040255A2 (en) * 1995-06-07 1996-12-19 G.D. Searle & Co. Method to treat cardiofibrosis with a combination therapy of an angiotensin ii antagonist and an epoxy-steroidal aldosterone antagonist
GB2306476A (en) * 1995-10-27 1997-05-07 Merck & Co Inc Hiv integrase inhibitors
US5759842A (en) 1996-10-24 1998-06-02 Merck & Co., Inc. In vitro HIV integrase inhibitors
CA2280518A1 (en) 1997-02-06 1998-08-13 Deborah L. Zink Hiv integrase inhibitors
IL137974A0 (en) 1998-03-26 2001-10-31 Shionogi & Co Indole derivatives having antiviral activity
TR200101886T2 (tr) 1998-12-25 2001-12-21 Shionogi & Co., Ltd. HIV integrazını önleme aktivitesi olan aromatik heterosikl bileşimleri.

Also Published As

Publication number Publication date
WO2000075122A1 (en) 2000-12-14
EP1186599A1 (en) 2002-03-13
CA2376043A1 (en) 2000-12-14
MXPA01012299A (es) 2002-07-30
CN1367784A (zh) 2002-09-04
BR0011246A (pt) 2002-03-05
US6831177B1 (en) 2004-12-14
TR200103801T2 (tr) 2002-04-22
EP1186599A4 (en) 2003-02-26
AU763231B2 (en) 2003-07-17
AU4782700A (en) 2000-12-28
KR20020020718A (ko) 2002-03-15
KR100423781B1 (ko) 2004-03-22

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