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TR200000333T2 - 4-aminopyrol (3,2-d) pyrimidines as Y receptor antagonists. - Google Patents

4-aminopyrol (3,2-d) pyrimidines as Y receptor antagonists.

Info

Publication number
TR200000333T2
TR200000333T2 TR2000/00333T TR200000333T TR200000333T2 TR 200000333 T2 TR200000333 T2 TR 200000333T2 TR 2000/00333 T TR2000/00333 T TR 2000/00333T TR 200000333 T TR200000333 T TR 200000333T TR 200000333 T2 TR200000333 T2 TR 200000333T2
Authority
TR
Turkey
Prior art keywords
aminopyrol
pyrimidines
receptor antagonists
neuropeptide
excess
Prior art date
Application number
TR2000/00333T
Other languages
Turkish (tr)
Inventor
Lee Dow Robert
Hammond Marlys
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of TR200000333T2 publication Critical patent/TR200000333T2/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Nöropeptid Y'nin fazlaligiyla iliskilendirilen kosullarin tedavisi için formül (I) bilesimleriCompounds of formula (I) for the treatment of conditions associated with an excess of neuropeptide Y

TR2000/00333T 1997-08-05 1998-07-10 4-aminopyrol (3,2-d) pyrimidines as Y receptor antagonists. TR200000333T2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5473497P 1997-08-05 1997-08-05

Publications (1)

Publication Number Publication Date
TR200000333T2 true TR200000333T2 (en) 2000-05-22

Family

ID=21993163

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/00333T TR200000333T2 (en) 1997-08-05 1998-07-10 4-aminopyrol (3,2-d) pyrimidines as Y receptor antagonists.

Country Status (32)

Country Link
US (1) US6187778B1 (en)
EP (1) EP1003744B1 (en)
JP (1) JP3711238B2 (en)
KR (1) KR20010022583A (en)
CN (1) CN1264381A (en)
AP (1) AP9801312A0 (en)
AT (1) ATE296825T1 (en)
AU (1) AU7927498A (en)
BG (1) BG104107A (en)
BR (1) BR9811844A (en)
CA (1) CA2293621C (en)
CO (1) CO4960634A1 (en)
DE (1) DE69830409T2 (en)
EA (1) EA200000098A1 (en)
ES (1) ES2241146T3 (en)
GT (1) GT199800114A (en)
HR (1) HRP980434A2 (en)
HU (1) HUP0002956A3 (en)
ID (1) ID24300A (en)
IL (1) IL133430A0 (en)
IS (1) IS5294A (en)
MA (1) MA24629A1 (en)
NO (1) NO996178L (en)
OA (1) OA11277A (en)
PA (1) PA8456601A1 (en)
PE (1) PE106199A1 (en)
PL (1) PL338575A1 (en)
SA (1) SA98190435A (en)
TN (1) TNSN98148A1 (en)
TR (1) TR200000333T2 (en)
WO (1) WO1999007703A1 (en)
ZA (1) ZA986968B (en)

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US7507740B2 (en) 2004-06-02 2009-03-24 Takeda Pharmaceutical Company Limited Fused heterocyclic compound
MXPA06014798A (en) 2004-06-17 2007-06-22 Wyeth Corp Gonadotropin releasing hormone receptor antagonists.
RU2007101509A (en) 2004-06-17 2008-07-27 Уайт (Us) METHOD FOR PRODUCING HORMONE RECEPTOR ANTAGONISTS RELEASING GONADOTROPINE
MX2007001399A (en) * 2004-08-02 2007-04-18 Osi Pharm Inc Aryl-amino substituted pyrrolopyrimidine multi-kinase inhibiting compounds.
MY179032A (en) 2004-10-25 2020-10-26 Cancer Research Tech Ltd Ortho-condensed pyridine and pyrimidine derivatives (e.g.purines) as protein kinase inhibitors
KR20060087386A (en) 2005-01-28 2006-08-02 주식회사 대웅제약 Novel benzoimidazole derivatives and pharmaceutical compositions containing them
PL1861387T3 (en) * 2005-01-28 2014-08-29 Dae Woong Pharma Benzimidazole derivatives and pharmaceutical compositions thereof
US7538113B2 (en) 2005-02-18 2009-05-26 Wyeth 4-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7534796B2 (en) 2005-02-18 2009-05-19 Wyeth Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor
US7582634B2 (en) 2005-02-18 2009-09-01 Wyeth 7-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
WO2006108218A1 (en) * 2005-04-15 2006-10-19 Regenertech Pty Limited Use of neuropeptide y (npy) and agonists and antagonists thereof for tissue regeneration
US7531542B2 (en) 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
US7582636B2 (en) 2005-05-26 2009-09-01 Wyeth Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor
WO2007007910A1 (en) * 2005-07-13 2007-01-18 Banyu Pharmaceutical Co., Ltd. Heterocycle-substituted benzimidazole derivative
UY29825A1 (en) * 2005-10-03 2007-05-31 Astrazeneca Ab SUBSTITUTED DERIVATIVES OF 3H-IMIDAZOL- (4.5 B (BETA)) PIRIDINA-2-IL BENZOATES AND BENZAMIDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND APPLICATIONS
AR057525A1 (en) * 2005-10-03 2007-12-05 Astrazeneca Ab GSK3 SELECTIVE INHIBITING COMPOUNDS AND A PROCESS FOR PREPARATION
US20070129364A1 (en) * 2005-12-07 2007-06-07 Han-Qing Dong Pyrrolopyridine kinase inhibiting compounds
ES2526813T3 (en) * 2005-12-22 2015-01-15 Cancer Research Technology Limited Enzyme inhibitors
KR20080085232A (en) 2006-02-17 2008-09-23 화이자 리미티드 3-deazapurine derivatives as TLR7 modulators
JP5606734B2 (en) 2006-04-25 2014-10-15 アステックス、セラピューティックス、リミテッド Pharmaceutical compounds
EP2054405B1 (en) 2006-07-11 2013-09-18 Daewoong Pharmaceutical Co., Ltd. Novel biaryl benzoimidazole derivatives and pharmaceutical composition comprising the same
KR101134239B1 (en) 2006-07-11 2012-04-10 주식회사 대웅제약 Novel biaryl benzoimidazole derivatives and pharmaceutical composition comprising the same
CL2007002617A1 (en) 2006-09-11 2008-05-16 Sanofi Aventis COMPOUNDS DERIVED FROM PIRROLO [2,3-B] PIRAZIN-6-ILO; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT INFLAMMATION OF THE ARTICULATIONS, Rheumatoid Arthritis, TUMORS, LYMPHOMA OF THE CELLS OF THE MANTO.
WO2008121064A1 (en) * 2007-03-30 2008-10-09 Astrazeneca Ab New imidazo[4,5-b]pyridine-6-halo-7-aryl/heteroaryl compounds 705
DE102007027800A1 (en) 2007-06-16 2008-12-18 Bayer Healthcare Ag Substituted bicyclic heteroaryl compounds and their use
JP4705695B2 (en) 2007-10-11 2011-06-22 アストラゼネカ アクチボラグ Pyrrolo [2,3-D] pyrimidine derivatives as protein kinase B inhibitors
CA2711777A1 (en) 2008-01-11 2009-08-13 Natco Pharma Limited Novel pyrazolo [3,4-d] pyrimidine derivatives as anti-cancer drugs
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JP7530360B2 (en) * 2018-11-30 2024-08-07 武田薬品工業株式会社 TYK2 INHIBITORS AND USES THEREOF

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US5877178A (en) * 1991-04-08 1999-03-02 Duquesne University Of The Holy Ghost Pyrimidine derivatives and methods of making and using these derivatives
US5235053A (en) * 1992-06-22 1993-08-10 Eli Lilly And Company Process for the synthesis of 4-hydroxy-5-halopyrrold[2,3-d]pyrimidine intermediates
US5284971A (en) 1992-07-16 1994-02-08 Syntex (U.S.A.) Inc. 4-(3-cyclohexyl-4-hydroxy or-methoxy phenylsulfonyl) 3,5 dibromo phenyl acetic thyromimetic cholesterol-lowering agents
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Also Published As

Publication number Publication date
HUP0002956A3 (en) 2002-01-28
IL133430A0 (en) 2001-04-30
HRP980434A2 (en) 1999-04-30
EP1003744B1 (en) 2005-06-01
CA2293621A1 (en) 1999-02-18
AP9801312A0 (en) 2000-01-30
NO996178L (en) 2000-02-14
GT199800114A (en) 2000-01-18
DE69830409T2 (en) 2006-01-26
ID24300A (en) 2000-07-13
AU7927498A (en) 1999-03-01
US6187778B1 (en) 2001-02-13
ZA986968B (en) 2000-02-04
ATE296825T1 (en) 2005-06-15
EP1003744A1 (en) 2000-05-31
KR20010022583A (en) 2001-03-26
CO4960634A1 (en) 2000-09-25
SA98190435A (en) 2005-12-03
PE106199A1 (en) 1999-11-02
JP2001512729A (en) 2001-08-28
PL338575A1 (en) 2000-11-06
JP3711238B2 (en) 2005-11-02
BG104107A (en) 2000-08-31
TNSN98148A1 (en) 2005-03-15
OA11277A (en) 2003-07-29
ES2241146T3 (en) 2005-10-16
NO996178D0 (en) 1999-12-14
MA24629A1 (en) 1999-04-01
BR9811844A (en) 2000-08-08
CN1264381A (en) 2000-08-23
CA2293621C (en) 2003-12-30
WO1999007703A1 (en) 1999-02-18
EA200000098A1 (en) 2000-08-28
PA8456601A1 (en) 2000-05-24
HUP0002956A2 (en) 2001-08-28
DE69830409D1 (en) 2005-07-07
IS5294A (en) 1999-12-10

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