TNSN97033A1 - NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS. - Google Patents
NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS.Info
- Publication number
- TNSN97033A1 TNSN97033A1 TNTNSN97033A TNSN97033A TNSN97033A1 TN SN97033 A1 TNSN97033 A1 TN SN97033A1 TN TNSN97033 A TNTNSN97033 A TN TNSN97033A TN SN97033 A TNSN97033 A TN SN97033A TN SN97033 A1 TNSN97033 A1 TN SN97033A1
- Authority
- TN
- Tunisia
- Prior art keywords
- oxazolidinones
- preparing
- medicaments
- novel heteroaryl
- heteroaryl
- Prior art date
Links
- 239000003814 drug Substances 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 229940088710 antibiotic agent Drugs 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
L'INVENTION CONCERNE DE NOUVELLES HETEROARYL-OXAZOLIDINONES DE FORMULE GENERALE ( I) DANS LAQUELLE LES SUBSTITUANTS SONT TELS QUE DEFINIS DANS LA DESCRIPTION, DES PROCEDES POUR LES PREPARER, ET LEUR UTILISATION EN TANT QUE MEDICAMENTS, EN PARTICULIER EN TANT QUE MEDICAMENTS ANTIBACTERIENS.THE INVENTION RELATES TO NEW HETEROARYL-OXAZOLIDINONES OF GENERAL FORMULA (I) IN WHICH THE SUBSTITUTES ARE AS DEFINED IN THE DESCRIPTION, METHODS FOR PREPARING THEM, AND THEIR USE AS DRUGS, PARTICULARLY AS ANTIBACTERIALS.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19604224 | 1996-02-06 | ||
| DE19649095A DE19649095A1 (en) | 1996-02-06 | 1996-11-27 | New 5-(acyl-aminomethyl)-3-hetero-aryl-oxazolidinone compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TNSN97033A1 true TNSN97033A1 (en) | 2005-03-15 |
Family
ID=7784634
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TNTNSN97033A TNSN97033A1 (en) | 1996-02-06 | 1997-02-04 | NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS. |
Country Status (10)
| Country | Link |
|---|---|
| KR (1) | KR970061891A (en) |
| AR (1) | AR005704A1 (en) |
| CO (1) | CO4761067A1 (en) |
| DE (1) | DE19649095A1 (en) |
| PE (1) | PE36098A1 (en) |
| SV (1) | SV1997000010A (en) |
| TN (1) | TNSN97033A1 (en) |
| TW (1) | TW362974B (en) |
| YU (1) | YU4497A (en) |
| ZA (1) | ZA97928B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
| DE19802239A1 (en) * | 1998-01-22 | 1999-07-29 | Bayer Ag | New oxazolidinone derivatives useful as antimicrobial agents against Gram-positive and some Gram-negative bacteria, mycobacteria, etc. |
| US6562844B2 (en) | 1998-01-23 | 2003-05-13 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
| US7002020B1 (en) | 1998-01-23 | 2006-02-21 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
| WO1999037630A1 (en) * | 1998-01-23 | 1999-07-29 | Versicor, Inc. | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
| WO2006106426A1 (en) * | 2005-04-06 | 2006-10-12 | Pharmacia & Upjohn Company Llc | An oxindole oxazolidinone as antibacterial agent |
| AU2006231919A1 (en) | 2005-04-06 | 2006-10-12 | Pharmacia & Upjohn Company Llc | 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents |
| WO2008021337A1 (en) | 2006-08-15 | 2008-02-21 | Wyeth | Oxazinan-2-one derivatives useful as pr modulators |
| TW200815428A (en) | 2006-08-15 | 2008-04-01 | Wyeth Corp | Oxazolidone derivatives as PR modulators |
-
1996
- 1996-11-27 DE DE19649095A patent/DE19649095A1/en not_active Withdrawn
-
1997
- 1997-02-04 TN TNTNSN97033A patent/TNSN97033A1/en unknown
- 1997-02-04 AR ARP970100440A patent/AR005704A1/en unknown
- 1997-02-04 TW TW086101260A patent/TW362974B/en active
- 1997-02-05 KR KR1019970003609A patent/KR970061891A/en not_active Withdrawn
- 1997-02-05 ZA ZA9700928A patent/ZA97928B/en unknown
- 1997-02-05 YU YU4497A patent/YU4497A/en unknown
- 1997-02-05 PE PE1997000072A patent/PE36098A1/en not_active Application Discontinuation
- 1997-02-06 CO CO97006152A patent/CO4761067A1/en unknown
- 1997-02-06 SV SV1997000010A patent/SV1997000010A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CO4761067A1 (en) | 1999-04-27 |
| KR970061891A (en) | 1997-09-12 |
| PE36098A1 (en) | 1998-08-29 |
| DE19649095A1 (en) | 1997-08-07 |
| AR005704A1 (en) | 1999-07-14 |
| ZA97928B (en) | 1997-08-05 |
| YU4497A (en) | 1999-09-27 |
| TW362974B (en) | 1999-07-01 |
| SV1997000010A (en) | 1997-10-23 |
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