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TN2011000151A1 - Hiv integrase inhibitors - Google Patents

Hiv integrase inhibitors

Info

Publication number
TN2011000151A1
TN2011000151A1 TN2011000151A TN2011000151A TN2011000151A1 TN 2011000151 A1 TN2011000151 A1 TN 2011000151A1 TN 2011000151 A TN2011000151 A TN 2011000151A TN 2011000151 A TN2011000151 A TN 2011000151A TN 2011000151 A1 TN2011000151 A1 TN 2011000151A1
Authority
TN
Tunisia
Prior art keywords
compounds
hiv
hiv integrase
inhibitors
integrase inhibitors
Prior art date
Application number
TN2011000151A
Other languages
French (fr)
Inventor
Richard C A Isaacs
Wayne J Thompson
Peter D Williams
Dai-Shi Su
Shankar Venkatraman
Mark W Embrey
Thorsten E Fisher
John S Wai
David C Dubost
Richard G Ball
Eric J Choi
Tao Pei
Sarah L Trice
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2009/059306 external-priority patent/WO2010042391A2/en
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of TN2011000151A1 publication Critical patent/TN2011000151A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Compounds of Formula I are inhibitors of HIV integrase and inhibitors of HIV replication: (I), wherein X1, X2, Y, R1A, R1B, R2 and R3 are defined herein. The compounds are useful for the prophylaxis or treatment of infection by HIV and the prophylaxis, treatment, or delay in the onset or progression of AIDS. The compounds are employed against HIV infection and AIDS as compounds per se (or as hydrates or solvates thereof) or in the form of pharmaceutically acceptable salts. The compounds and their salts can be employed as ingredients in pharmaceutical compositions, optionally in combination with other antivirals, immunomodulators, antibiotics or vaccines.
TN2011000151A 2009-10-02 2011-03-30 Hiv integrase inhibitors TN2011000151A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2009/059306 WO2010042391A2 (en) 2008-10-06 2009-10-02 Hiv integrase inhibitors

Publications (1)

Publication Number Publication Date
TN2011000151A1 true TN2011000151A1 (en) 2012-09-05

Family

ID=55024437

Family Applications (1)

Application Number Title Priority Date Filing Date
TN2011000151A TN2011000151A1 (en) 2009-10-02 2011-03-30 Hiv integrase inhibitors

Country Status (1)

Country Link
TN (1) TN2011000151A1 (en)

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