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SV2009003231A - Uso de valerato de estradiol o 17b-estradiol en combinacion con dienogest en una terapia oral para mantener y/o implementar la libido femenina - Google Patents

Uso de valerato de estradiol o 17b-estradiol en combinacion con dienogest en una terapia oral para mantener y/o implementar la libido femenina

Info

Publication number
SV2009003231A
SV2009003231A SV2009003231A SV2009003231A SV2009003231A SV 2009003231 A SV2009003231 A SV 2009003231A SV 2009003231 A SV2009003231 A SV 2009003231A SV 2009003231 A SV2009003231 A SV 2009003231A SV 2009003231 A SV2009003231 A SV 2009003231A
Authority
SV
El Salvador
Prior art keywords
estradiol
combination
dienogest
maintain
implement
Prior art date
Application number
SV2009003231A
Other languages
English (en)
Inventor
Susan Zeun
Holger Zimmermann
Susanne Parke
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of SV2009003231A publication Critical patent/SV2009003231A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

LA INVENCIÓN SE RELACIONA CON EL USO DE VALERATO DE ESTRADIOL O 17BETA-ESTRADIOL (ESTRADIOL) EN COMBINACIÓN CON 17ALFA-CIANOMETIL-17-BETA-HIDROXIESTRA-4,9-DIEN-3-ONA (DIENOGEST) EN UN PRODUCTO COMBINADO DE MÚLTIPLES FASES O DE UNA SOLA FASE EN UNA TERAPIA ORAL PARA MANTENER Y/O INCREMENTAR LA LIBIDO FEMENINA, CUANDO FUERA APROPIADO TAMBIÉN JUNTO CON UNA CONTRACEPCIÓN ORAL. LAS UNIDADES DE DOSIS DIARIAS TOTALES DE LA COMBINACIÓN DE MÚLTIPLES FASES Y DEL PLACEBO FARMACÉUTICAMENTE ACEPTABLE O LAS UNIDADES DE DOSIS DIARIAS DE LA COMBINACIÓN DE UNA SOLA FASE Y SIN INGREDIENTE ACTIVO Y SIN PLACEBO CORRESPONDEN A 28 DÍAS
SV2009003231A 2006-10-20 2009-04-20 Uso de valerato de estradiol o 17b-estradiol en combinacion con dienogest en una terapia oral para mantener y/o implementar la libido femenina SV2009003231A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06022091 2006-10-20
EP07009373A EP1930010A1 (de) 2006-10-20 2007-05-10 Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido

Publications (1)

Publication Number Publication Date
SV2009003231A true SV2009003231A (es) 2009-11-09

Family

ID=38809728

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2009003231A SV2009003231A (es) 2006-10-20 2009-04-20 Uso de valerato de estradiol o 17b-estradiol en combinacion con dienogest en una terapia oral para mantener y/o implementar la libido femenina

Country Status (17)

Country Link
US (1) US8349820B2 (es)
EP (2) EP1930010A1 (es)
JP (1) JP2010506867A (es)
KR (1) KR20090080989A (es)
AU (1) AU2007312626A1 (es)
BR (1) BRPI0717462A2 (es)
CA (1) CA2666829C (es)
CO (1) CO6160297A2 (es)
CR (1) CR10732A (es)
EA (1) EA016631B1 (es)
GT (1) GT200900090A (es)
IL (1) IL198200A (es)
MX (1) MX2009004179A (es)
NO (1) NO20091954L (es)
NZ (1) NZ576336A (es)
SV (1) SV2009003231A (es)
WO (1) WO2008046559A1 (es)

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US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
EP3936133A1 (en) 2011-11-23 2022-01-12 TherapeuticsMD, Inc. Natural combination hormone replacement formulations and therapies
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10206932B2 (en) 2014-05-22 2019-02-19 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
CA3020153A1 (en) 2016-04-01 2017-10-05 Therapeuticsmd, Inc. Steroid hormone pharmaceutical composition
US10286077B2 (en) 2016-04-01 2019-05-14 Therapeuticsmd, Inc. Steroid hormone compositions in medium chain oils
US11633405B2 (en) 2020-02-07 2023-04-25 Therapeuticsmd, Inc. Steroid hormone pharmaceutical formulations

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Also Published As

Publication number Publication date
CA2666829A1 (en) 2008-04-24
EA016631B1 (ru) 2012-06-29
WO2008046559A1 (de) 2008-04-24
MX2009004179A (es) 2009-04-30
NO20091954L (no) 2009-05-19
IL198200A0 (en) 2009-12-24
JP2010506867A (ja) 2010-03-04
BRPI0717462A2 (pt) 2013-12-24
CA2666829C (en) 2012-02-07
AU2007312626A1 (en) 2008-04-24
NZ576336A (en) 2012-03-30
EP2083827A1 (de) 2009-08-05
US20080125401A1 (en) 2008-05-29
EA200900491A1 (ru) 2009-10-30
US8349820B2 (en) 2013-01-08
KR20090080989A (ko) 2009-07-27
CR10732A (es) 2009-05-25
GT200900090A (es) 2011-11-29
CO6160297A2 (es) 2010-05-20
EP1930010A1 (de) 2008-06-11
IL198200A (en) 2012-10-31

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