[go: up one dir, main page]

SV2006001970A - Hormonas de administracion transdermica que no necesitan potenciadores de penetracion ref. p-sv-77.461/cd - Google Patents

Hormonas de administracion transdermica que no necesitan potenciadores de penetracion ref. p-sv-77.461/cd

Info

Publication number
SV2006001970A
SV2006001970A SV2004001970A SV2004001970A SV2006001970A SV 2006001970 A SV2006001970 A SV 2006001970A SV 2004001970 A SV2004001970 A SV 2004001970A SV 2004001970 A SV2004001970 A SV 2004001970A SV 2006001970 A SV2006001970 A SV 2006001970A
Authority
SV
El Salvador
Prior art keywords
hormones
penetration
potentizers
ref
transdermal administration
Prior art date
Application number
SV2004001970A
Other languages
English (en)
Inventor
Thomas Langguth
Stefan Bracht
Michael Dittgen
Dirk Schenk
Petra Huber
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34924031&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2006001970(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Ag filed Critical Schering Ag
Publication of SV2006001970A publication Critical patent/SV2006001970A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061Polyacrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7076Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising ingredients of undetermined constitution or reaction products thereof, e.g. rosin or other plant resins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Botany (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

UN PARCHE QUE COMPRENDE UNA CAPA DE DROGA CON UN BAJO CONTENIDO DE HORMONAS, COMO POR EJEMPLO GESTODENO, Y OPCIONALMENTE UN ESTROGENO POR EJEMPLO ETINILESTRADIOL). AL APLICAR EL PARCHE A UNA MUJER, SE CONSIGUEN NIVELES EN PLASMA DE AL MENOS 1, ONG/ML DE GESTODENO EN CONDICIONES DE ESTADO ESTACIONARIO SIN NECESIDAD DE INCORPORAR POTENCIADORES DE PENETRACION NI MEJORADORES DE PERMEACION EN LA CAPA QUE CONTIENE DROGA, TAMBIEN SON SATISFACTORIOS LOS NIVELES EN PLASMA DE LAS HORMONAS QUE SE CONSIGUEN DURANTE TODO UN PERIODO DE AL MENOS 1 SEMANA, HACIENDO QUE EL PARCHE SE PUEDA APLICAR PARA UTILIZARLO EN ANTICONCEPCION FEMENINA CON EL CONCEPTO DE APLICAR PARA UTILIZAR EN ANTICONCEPCION FEMENIA CON EL CONCEPTO DE APLICAR EL PARCHE UNA VEZ A LA SEMANA
SV2004001970A 2003-12-12 2004-12-10 Hormonas de administracion transdermica que no necesitan potenciadores de penetracion ref. p-sv-77.461/cd SV2006001970A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP03078881 2003-12-12

Publications (1)

Publication Number Publication Date
SV2006001970A true SV2006001970A (es) 2006-02-16

Family

ID=34924031

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2004001970A SV2006001970A (es) 2003-12-12 2004-12-10 Hormonas de administracion transdermica que no necesitan potenciadores de penetracion ref. p-sv-77.461/cd

Country Status (23)

Country Link
EP (2) EP2138169B1 (es)
CN (1) CN101843603B (es)
AR (1) AR046762A1 (es)
AT (1) ATE457168T1 (es)
CR (1) CR8465A (es)
CY (2) CY1110637T1 (es)
DE (1) DE602004025444D1 (es)
DK (2) DK2138169T3 (es)
ES (2) ES2340925T3 (es)
GT (1) GT200400262A (es)
HN (1) HN2004000526A (es)
HR (2) HRP20100254T1 (es)
JO (1) JO2606B1 (es)
ME (1) ME01069B (es)
MY (2) MY144053A (es)
PE (1) PE20051035A1 (es)
PL (2) PL2138169T3 (es)
PT (2) PT2138169E (es)
RS (2) RS51260B (es)
SI (2) SI1541137T1 (es)
SV (1) SV2006001970A (es)
TW (1) TWI257299B (es)
UA (1) UA89766C2 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1594483E (pt) 2003-02-21 2006-12-29 Schering Ag Penso transdérmico estável aos uv
US8668925B2 (en) 2003-12-12 2014-03-11 Bayer Intellectual Property Gmbh Transdermal delivery of hormones without the need of penetration enhancers
US8962013B2 (en) 2005-05-02 2015-02-24 Bayer Intellectual Property Gmbh Multi-layered transdermal system with triazine UV absorber
DE102005050729A1 (de) * 2005-10-19 2007-04-26 Schering Ag Verfahren zur präventiven bedarfsweisen hormonalen Kontrazeption
WO2010042610A1 (en) 2008-10-08 2010-04-15 Agile Therapeutics, Inc. Transdermal delivery
CA2740002C (en) 2008-10-08 2016-11-01 Agile Therapeutics, Inc. Transdermal delivery
CA2740005C (en) 2008-10-08 2016-11-01 Agile Therapeutics, Inc. Transdermal delivery
EP2410859A4 (en) 2009-03-27 2013-03-13 Agile Therapeutics Inc TRANSDERMAL ADMINISTRATION
DE102010040299A1 (de) * 2010-09-06 2012-03-08 Bayer Schering Pharma Aktiengesellschaft Transdermale therapeutische Systeme mit kristallisationsinhibierender Schutzfolie (Release Liner)
AU2015203180B2 (en) * 2010-09-06 2016-06-30 Bayer Intellectual Property Gmbh Transdermal therapeutic systems with crystallization-inhibiting protective film (release liner)
HRP20170292T1 (hr) 2010-09-06 2017-04-21 Bayer Intellectual Property Gmbh Transdermalni flasteri niske doze s visokim otpuštanjem lijeka
HK1204287A1 (en) * 2012-01-27 2015-11-13 敏捷治疗公司 Transdermal hormone delivery

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4081537A (en) 1975-10-10 1978-03-28 Schering Aktiengesellschaft Δ15 -Steroids and pharmaceutical compositions thereof
JP3238389B2 (ja) * 1988-10-27 2001-12-10 シエーリング アクチエンゲゼルシヤフト ゲストデン含有の経皮適用のための薬剤
PT99338A (pt) 1990-10-29 1992-10-30 Alza Corp Processo para a preparacao de composicoes de farmacos anticoncepcionais administradas transdermicamente contendo uma mistura dum estrogeno e gestodeno e dispositivos para a sua administracao transdermica
US5512292A (en) 1990-10-29 1996-04-30 Alza Corporation Transdermal contraceptive formulations methods and devices
DE4336557C2 (de) 1993-05-06 1997-07-17 Lohmann Therapie Syst Lts Estradiolhaltiges transdermales therapeutisches System, Verfahren zu seiner Herstellung und seine Verwendung
DE4329242A1 (de) * 1993-08-26 1995-03-02 Schering Ag Mittel zur transdermalen Applikation enthaltend Gestodenester
DE4405898A1 (de) 1994-02-18 1995-08-24 Schering Ag Transdermale therapeutische Systeme enthaltend Sexualsteroide
US5762956A (en) 1996-04-24 1998-06-09 Rutgers, The State University Of New Jersey Transdermal contraceptive delivery system and process
DE19906152B4 (de) 1999-02-10 2005-02-10 Jenapharm Gmbh & Co. Kg Wirkstoffhaltige Laminate für Transdermalsysteme
EP1242012B1 (en) 1999-11-24 2009-12-30 Agile Therapeutics, Inc. Improved transdermal contraceptive delivery system and process
DE10053375C1 (de) * 2000-10-27 2002-01-24 Lohmann Therapie Syst Lts Transdermale therapeutische Systeme mit lichtempfindlichen Wirkstoffen
TWI287455B (en) 2000-12-05 2007-10-01 Noven Pharma Crystallization inhibition of drugs in transdermal drug delivery systems and methods of use

Also Published As

Publication number Publication date
CN101843603B (zh) 2012-06-27
PT1541137E (pt) 2010-05-17
ATE457168T1 (de) 2010-02-15
CN101843603A (zh) 2010-09-29
EP2138169A3 (en) 2011-04-06
EP1541137B1 (en) 2010-02-10
CR8465A (es) 2007-06-06
HK1074801A1 (en) 2005-11-25
PL1541137T3 (pl) 2010-07-30
JO2606B1 (en) 2011-11-01
ES2340925T3 (es) 2010-06-11
CY1110637T1 (el) 2015-04-29
EP1541137A3 (en) 2005-11-16
CY1115064T1 (el) 2016-12-14
PE20051035A1 (es) 2006-02-08
MY152750A (en) 2014-11-28
DK1541137T3 (da) 2010-04-26
MY144053A (en) 2011-08-15
ME01069B (me) 2012-10-20
HRP20140077T1 (hr) 2014-02-28
EP1541137A2 (en) 2005-06-15
EP2138169B1 (en) 2013-11-06
PL2138169T3 (pl) 2014-04-30
DE602004025444D1 (de) 2010-03-25
DK2138169T3 (da) 2013-11-18
AR046762A1 (es) 2005-12-21
HK1132682A1 (en) 2010-03-05
HRP20100254T1 (hr) 2010-06-30
HN2004000526A (es) 2010-02-01
ES2445690T3 (es) 2014-03-04
RS51260B (sr) 2010-12-31
TWI257299B (en) 2006-07-01
RS53182B (sr) 2014-06-30
GT200400262A (es) 2005-10-31
TW200528073A (en) 2005-09-01
SI1541137T1 (sl) 2010-06-30
EP2138169A2 (en) 2009-12-30
UA89766C2 (en) 2010-03-10
SI2138169T1 (sl) 2014-03-31
PT2138169E (pt) 2014-02-17

Similar Documents

Publication Publication Date Title
CU20100143A7 (es) Hormonas de administración transdérmica que no necesitan potenciadores de penetración
SV2006001970A (es) Hormonas de administracion transdermica que no necesitan potenciadores de penetracion ref. p-sv-77.461/cd
CY1125035T1 (el) Ουσια-φορεας φαρμακων και κιτ ουσιας-φορεα φαρμακων για αναστολη ινωσης
ATE329586T1 (de) Zusammensetzungen enthaltend carotenoide und deren verwendung zur verhinderung hormon- induzierter nebenwirkungen
MX2022008277A (es) Composiciones de gel para administracion transdermica para maximizar las concentraciones de farmaco en el estrato corneo y suero, y metodos de uso de las mismas.
ES2190472T3 (es) Parche transdermico para la administracion de 17-deacetil norgestimato, solo o en combinacion con un estrogeno.
ES2167061T3 (es) Formas de dosificacion para mejorar la disfuncion erectil en pacientes de sexo masculino.
AR048878A1 (es) Composiciones topicas de metadona y metodos para usarlas
ECSP003847A (es) Composiciones farmaceuticas que proporcionan concentraciones potenciadas de farmaco
AR033808A1 (es) Una composicion topica de anestesia local y los parches y los envases que la contienen
SV2006002165A (es) Regimenes y kits de progestina ciclica ref. am101677
AR021459A1 (es) PARCHE QUE CONTIENE ESTRADIOL PARA LA APLICACIoN PERCUTÁNEA DE HORMONAS.
EA201590907A1 (ru) Усиленные полиамином составы для ионтофореза соединения триптана
AR044350A1 (es) Manguito y parche analgesico microencapsulado de uso topico para el tratamiento del dolor
EA200702102A1 (ru) Пластинки, содержащие стероидные гормоны
CR8059A (es) Composicion farmaceutica en forma de hidrogel para administracion transdermica de sustancias activas
HN2001000038A (es) Sistema de administracion oral controlada para la ingestion diaria de ciprofloxacina
UY28668A1 (es) Hormonas de administración transdérmica que no necesitan potenciadores de penetración
CU23649B7 (es) Hormonas de administración transdérmica que no necesitan potenciadores de penetración
WO2006091719A3 (en) Compositions and methods enhancing transdermal delivery of drugs and biologics
AR044939A1 (es) Sistema de administracion para medicaciones topicas
AR029096A1 (es) Combinacion de sustancias activas que contiene montirelina y un compuesto de efecto opioide, medicamentos y formulaciones medicamentosas que contienen dicha combinacion y su uso para la preparacion de medicamentos para tratamiento del dolor
ATE269063T1 (de) Formulierungen zur transdermalen verabreichung von fenoldopam
WO2007016146A3 (en) Method for retarding systemic delivery rate for easily absorbable active agents
UY28579A1 (es) Formulaciones farmacéuticas transdermicas

Legal Events

Date Code Title Description
FD Lapse