SV2003000979A - DERIVATIVES OF PIRAZOL REF. PCS10958 - Google Patents
DERIVATIVES OF PIRAZOL REF. PCS10958Info
- Publication number
- SV2003000979A SV2003000979A SV2002000979A SV2002000979A SV2003000979A SV 2003000979 A SV2003000979 A SV 2003000979A SV 2002000979 A SV2002000979 A SV 2002000979A SV 2002000979 A SV2002000979 A SV 2002000979A SV 2003000979 A SV2003000979 A SV 2003000979A
- Authority
- SV
- El Salvador
- Prior art keywords
- derivatives
- pirazol
- invested
- transcript
- compounds
- Prior art date
Links
- 208000030507 AIDS Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 102000004190 Enzymes Human genes 0.000 abstract 1
- 108090000790 Enzymes Proteins 0.000 abstract 1
- 206010061598 Immunodeficiency Diseases 0.000 abstract 1
- 208000029462 Immunodeficiency disease Diseases 0.000 abstract 1
- 241000700605 Viruses Species 0.000 abstract 1
- 230000007813 immunodeficiency Effects 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
ESTA INVENCION SE REFIERE A DERIVADOS DE PIRAZOL DE FORMULA (I)VER FORMULA O A SALES, SOLVATOS O DERIVADOS FARMACEUTICAMENTE ACEPTABLES DE LOS MISMOS, EN LA QUE R1 A R4 SE DEFINEN EN LA DESCRIPCION, Y A PROCEDIMIENTOS PARA LA PREPARACION DE LOS MISMOS, A INTERMEDIOS USADOS EN SU PREPARACION, A COMPOSICIONES QUE LOS CONTIENEN Y A LOS USOS DE TALES DERIVADOS.LOS COMPUESTOS DE LA PRESENTE INVENCION SE UNEN A LA ENZIMA TRANSCRIPTASA INVERSA Y SON MODULADORES, ESPECIALMENTE INHIBIDORES, DE LA MISMA. COMO TALES, LOS COMPUESTOS DE LA PRESENTE INVENCION SON UTILES, EN EL TRATAMIENTO DE UNA DIVERSIDAD DE TRASTORNOS, INCLUYENDO AQUELLOS EN LOS QUE ESTA IMPLICADA LA INHIBICION DE LA TRANSCRIPTASA INVERSA. LOS TRASTORNOS DE INTERES INCLUYEN LOS CAUSADOS POR EL VIRUS DE LA INMUNODEFICIENCIA HUMANA (VIH) Y POR RRETROVIRUS RELACIONADOS GENETICAMENTE, TALES COMO EL SINDROME DE INMUNODEFICIENCIA ADQUIRIDA (SIDA)THIS INVENTION REFERS TO PIRAZOL DERIVATIVES OF FORMULA (I) SEE FORMULA OR SALTS, SOLVATES OR PHARMACEUTICALLY ACCEPTABLE DERIVATIVES OF THE SAME, IN WHICH R1 TO R4 ARE DEFINED IN THE DESCRIPTION, AND PROCEDURES FOR THE PREPARATION OF THEM, USED IN ITS PREPARATION, TO COMPOSITIONS THAT CONTAIN THEM AND TO THE USES OF SUCH DERIVATIVES. THE COMPOUNDS OF THE PRESENT INVENTION JOIN THE INVESTED TRANSCRIPT ENZYME AND ARE MODULATORS, ESPECIALLY INHIBITING, OF THE SAME. AS SUCH, THE COMPOUNDS OF THE PRESENT INVENTION ARE USEFUL, IN THE TREATMENT OF A DIVERSITY OF DISORDERS, INCLUDING THOSE IN WHICH THE INHIBITION OF THE INVESTED TRANSCRIPT IS INVOLVED. INTEREST DISORDERS INCLUDE THOSE CAUSED BY THE VIRUS OF HUMAN IMMUNODEFICIENCY (HIV) AND GENRETICALLY RELATED RRETROVIRUS, SUCH AS THE ACQUIRED IMMUNODEFICIENCY SYNDROME (AIDS)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0127426A GB0127426D0 (en) | 2001-11-15 | 2001-11-15 | Pyrazole derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2003000979A true SV2003000979A (en) | 2003-07-29 |
Family
ID=9925828
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2002000979A SV2003000979A (en) | 2001-11-15 | 2002-04-09 | DERIVATIVES OF PIRAZOL REF. PCS10958 |
Country Status (3)
| Country | Link |
|---|---|
| AP (1) | AP1846A (en) |
| GB (1) | GB0127426D0 (en) |
| SV (1) | SV2003000979A (en) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3963742A (en) * | 1974-07-12 | 1976-06-15 | American Cyanamid Company | 1,2-Dialkyl-3,4,5-trisubstituted pyrazolium salts as herbicidal agents |
-
2001
- 2001-11-15 GB GB0127426A patent/GB0127426D0/en not_active Ceased
-
2002
- 2002-04-04 AP APAP/P/2002/002469A patent/AP1846A/en active
- 2002-04-09 SV SV2002000979A patent/SV2003000979A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB0127426D0 (en) | 2002-01-09 |
| AP1846A (en) | 2008-05-09 |
| AP2002002469A0 (en) | 2002-06-30 |
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