SV2002000375A - PIPERIDINE OF BENZOAMIDE CONTAINING RELATED COMPOUNDS AND COMPOUNDS REF. PC10723 / 20161 / BB - Google Patents
PIPERIDINE OF BENZOAMIDE CONTAINING RELATED COMPOUNDS AND COMPOUNDS REF. PC10723 / 20161 / BBInfo
- Publication number
- SV2002000375A SV2002000375A SV2001000375A SV2001000375A SV2002000375A SV 2002000375 A SV2002000375 A SV 2002000375A SV 2001000375 A SV2001000375 A SV 2001000375A SV 2001000375 A SV2001000375 A SV 2001000375A SV 2002000375 A SV2002000375 A SV 2002000375A
- Authority
- SV
- El Salvador
- Prior art keywords
- compounds
- disorders
- piperidine
- benzoamide
- ref
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 title 2
- KXDAEFPNCMNJSK-UHFFFAOYSA-N Benzamide Chemical compound NC(=O)C1=CC=CC=C1 KXDAEFPNCMNJSK-UHFFFAOYSA-N 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 4
- 208000035475 disorder Diseases 0.000 abstract 4
- 239000005557 antagonist Substances 0.000 abstract 2
- GVBNSPFBYXGREE-UHFFFAOYSA-N (10-acetyloxy-8,8-dimethyl-2-oxo-9,10-dihydropyrano[2,3-f]chromen-9-yl) 2-methylbutanoate Chemical compound C1=CC(=O)OC2=C1C=CC1=C2C(OC(C)=O)C(OC(=O)C(C)CC)C(C)(C)O1 GVBNSPFBYXGREE-UHFFFAOYSA-N 0.000 abstract 1
- 241000589989 Helicobacter Species 0.000 abstract 1
- 208000019695 Migraine disease Diseases 0.000 abstract 1
- 208000002193 Pain Diseases 0.000 abstract 1
- 206010046543 Urinary incontinence Diseases 0.000 abstract 1
- 206010047700 Vomiting Diseases 0.000 abstract 1
- 230000033115 angiogenesis Effects 0.000 abstract 1
- 230000001364 causal effect Effects 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 210000000987 immune system Anatomy 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 206010027599 migraine Diseases 0.000 abstract 1
- ITNXJLXLFAFOHO-UHFFFAOYSA-N n-piperidin-1-ylbenzamide Chemical compound C=1C=CC=CC=1C(=O)NN1CCCCC1 ITNXJLXLFAFOHO-UHFFFAOYSA-N 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A CIERTOS COMPUESTOS QUE CONTIENEN BENZAMIDO-PIPERIDINA Y COMPUESTOS RELACIONADOS QUE PRESENTAN ACTIVIDAD COMO ANTAGONISTAS DEL RECEPTOR NK-1. (POR EJEMPLO, LOS ANTAGONISTAS DEL RECEPTOR DE LA SUSTANCIA P), A COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN, Y A SU USO EN EL TRATAMIENTO Y PREVENCION DE TRASTORNOS DEL SISTEMA NERVIOSO CENTRAL, TRASTORNOS INFLAMATORIOS, TRASTORNOS CARDIOVASCULARES, TRASTORNOS OFTALMICOS, TRASTORNOS GASTROINTESTINALES, TRASTORNOS CAUSADOS POR EL HELICOBACTER PYLON; TRASTORNOS DEL SISTEMA INMUNITARIO, INCONTINENCIA URINARIA, DOLOR, MIGRAÑA, EMESIS, ANGIOGÉNESIS Y OTROS TRASTORNOSTHIS INVENTION REFERS TO CERTAIN COMPOUNDS CONTAINING BENZAMIDO-PIPERIDINE AND RELATED COMPOUNDS THAT PRESENT ACTIVITY AS ANTAGONISTS OF THE NK-1 RECEIVER. (FOR EXAMPLE, THE ANTAGONISTS OF THE SUBSTANCE RECEIVER P), TO PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND TO ITS USE IN THE TREATMENT AND PREVENTION OF CENTRAL NERVOUS SYSTEMS, INFLAMMATORY DISORDERS, CAUSAL DISORDER DISORDERS, CARDIN DISORDERS FOR THE HELICOBACTER PYLON; IMMUNE SYSTEM SYSTEMS, URINARY INCONTINENCE, PAIN, MIGRAINE, EMESIS, ANGIOGENESIS AND OTHER DISORDERS
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US21292200P | 2000-06-20 | 2000-06-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2002000375A true SV2002000375A (en) | 2002-07-03 |
Family
ID=40094443
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2001000375A SV2002000375A (en) | 2000-06-20 | 2001-04-06 | PIPERIDINE OF BENZOAMIDE CONTAINING RELATED COMPOUNDS AND COMPOUNDS REF. PC10723 / 20161 / BB |
Country Status (2)
| Country | Link |
|---|---|
| SV (1) | SV2002000375A (en) |
| TN (1) | TNSN01054A1 (en) |
-
2001
- 2001-04-06 TN TNTNSN01054A patent/TNSN01054A1/en unknown
- 2001-04-06 SV SV2001000375A patent/SV2002000375A/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| TNSN01054A1 (en) | 2005-11-10 |
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