SE7408321L - - Google Patents
Info
- Publication number
- SE7408321L SE7408321L SE7408321A SE7408321A SE7408321L SE 7408321 L SE7408321 L SE 7408321L SE 7408321 A SE7408321 A SE 7408321A SE 7408321 A SE7408321 A SE 7408321A SE 7408321 L SE7408321 L SE 7408321L
- Authority
- SE
- Sweden
- Prior art keywords
- carbon atoms
- denotes
- carbalkoxy
- appropriately substituted
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
- C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
The novel anthelmintically active 2-carbalkoxy-amino-benzimidazole-5(6)-phenyl ethers and thioethers of the formula I <IMAGE> wherein R1 denotes alkyl having 1 to 4 carbon atoms, R2 and R3 independently of one another each denote hydrogen, hydroxyl, alkoxy having 1 to 4 carbon atoms, halogen, trifluoromethyl, alkyl having 1 to 4 carbon atoms or carbalkoxy having 1 to 4 carbon atoms in the alkoxy radical, R4 denotes hydrogen or chlorine and X denotes oxygen of sulphur, are prepared by reaction of appropriately substituted o-phenylenediamine derivatives with an appropriately substituted dithiomethyleneamino-formic acid ester. The compounds are valuable chemotherapeutics for the control of parasitic diseases in man and animals. They are particularly active against a large number of helminths, for example Haemonchus, Trichostrongylus, Ostertagia, Strongyloides, Cooperia, Chabertia, Oesophagostomum, Hyostrongylus, Ankylostoma, Askaris and Heterakis.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2332343A DE2332343A1 (en) | 1973-06-26 | 1973-06-26 | 2-CARBALCOXY-AMINO-BENZIMIDAZOL-5 (6) PHENYL ETHER, THEIR PRODUCTION AND USE IN AGENTS AGAINST HELMETS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SE7408321L true SE7408321L (en) | 1974-12-27 |
Family
ID=5885065
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7408321A SE7408321L (en) | 1973-06-26 | 1974-06-25 |
Country Status (12)
| Country | Link |
|---|---|
| JP (1) | JPS5758343B2 (en) |
| AT (1) | AT342041B (en) |
| CA (1) | CA1031781A (en) |
| CH (1) | CH614706A5 (en) |
| DE (1) | DE2332343A1 (en) |
| DK (1) | DK341474A (en) |
| ES (1) | ES427455A1 (en) |
| HU (1) | HU168527B (en) |
| IT (1) | IT1056735B (en) |
| NL (1) | NL7408394A (en) |
| SE (1) | SE7408321L (en) |
| YU (1) | YU37147B (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0028455A1 (en) * | 1979-10-12 | 1981-05-13 | Imperial Chemical Industries Plc | 5-Phenylselenobenzimidazole derivatives, their preparation and anthelmintic or fasciolicidal compositions containing them |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
-
1973
- 1973-06-26 DE DE2332343A patent/DE2332343A1/en active Pending
-
1974
- 1974-06-20 ES ES427455A patent/ES427455A1/en not_active Expired
- 1974-06-21 NL NL7408394A patent/NL7408394A/xx not_active Application Discontinuation
- 1974-06-24 IT IT24345/74A patent/IT1056735B/en active
- 1974-06-25 HU HUHO1682A patent/HU168527B/hu unknown
- 1974-06-25 DK DK341474A patent/DK341474A/da unknown
- 1974-06-25 CA CA203,352A patent/CA1031781A/en not_active Expired
- 1974-06-25 SE SE7408321A patent/SE7408321L/xx not_active Application Discontinuation
- 1974-06-25 YU YU1780/74A patent/YU37147B/en unknown
- 1974-06-25 CH CH871574A patent/CH614706A5/en not_active IP Right Cessation
- 1974-06-25 AT AT525274A patent/AT342041B/en not_active IP Right Cessation
- 1974-06-26 JP JP49073154A patent/JPS5758343B2/ja not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| NL7408394A (en) | 1974-12-30 |
| HU168527B (en) | 1976-05-28 |
| YU178074A (en) | 1982-06-18 |
| YU37147B (en) | 1984-08-31 |
| CH614706A5 (en) | 1979-12-14 |
| DE2332343A1 (en) | 1975-01-16 |
| ES427455A1 (en) | 1976-07-16 |
| IT1056735B (en) | 1982-02-20 |
| ATA525274A (en) | 1977-07-15 |
| JPS5758343B2 (en) | 1982-12-09 |
| DK341474A (en) | 1975-03-17 |
| AT342041B (en) | 1978-03-10 |
| JPS5040564A (en) | 1975-04-14 |
| CA1031781A (en) | 1978-05-23 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| SE7506589L (en) | PROCEDURE FOR THE PREPARATION OF ANALOGA ASSOCIATIONS FOR DAUNOMYCIN | |
| ES2043761T3 (en) | AQUEOUS SOLUTIONS OR DISPERSIONS OF POLYURETHANES, A PROCEDURE FOR ITS MANUFACTURE AND ITS USE AS COATING MEDIA OR FOR THE MANUFACTURE OF COATING MEDIA. | |
| ES8104275A1 (en) | A METHOD FOR THE PREPARATION OF PHTHALIMIDINE DERIVATIVES | |
| IE780704L (en) | Anthelmintics | |
| SE7712060L (en) | PROCEDURE FOR THE PREPARATION OF FUROCUMARINES | |
| ES393881A1 (en) | 2-amino-4,5,7,8-tetrahydro-6h-thiazolo or oxazolo(5,4-d)azepines and salts | |
| SE7408321L (en) | ||
| ES8106891A1 (en) | PROCEDURE FOR THE OBTAINING OF 2-HYDROXIALKYL-3,4,5- TRIHIDROXI-PIPERIDINES | |
| SE7408320L (en) | ||
| KR850004467A (en) | Method for preparing benzimidazole derivatives | |
| KR870007895A (en) | Process for preparing Phenylsulfonylazole | |
| GB660305A (en) | Pesticidal compositions | |
| GB1418598A (en) | 3-aminocarbazole derivatives and test devices containing them | |
| ES8703459A1 (en) | PROCEDURE FOR THE PREPARATION OF ACID DERIVATIVES 4- (ISOXAZOLIL) -TIAZOL-2-OXAMICO | |
| GB1147035A (en) | Seed-treatment nematocides, and certain novel 2,4-dihalophenylsulphonates having nematocidal properties | |
| US3335146A (en) | Pyridinol compound | |
| KR840000172A (en) | Sterilization and growth control compositions and their preparation | |
| GB1301505A (en) | ||
| GB1118131A (en) | Improvements in or relating to substituted benzimidazoles and the manufacture thereof | |
| ES8305378A1 (en) | "PROCEDURE FOR OBTAINING THYOLIC DERIVATIVES OF ERYTHROMYCIN AND THE PROPIONIC ESTER OF ERYTHROMYCIN". | |
| ES436317A1 (en) | PROCEDURE FOR THE PREPARATION OF NEW ISOQUINOLEINS. | |
| HU180660B (en) | Process for preparing substituted o-phenylene-diamine derivatives | |
| KR840006335A (en) | Process for preparing substituted benzene sulfonic acid ester | |
| GB1382658A (en) | Manufacture of tetramisole | |
| ES2034537T3 (en) | PROCEDURE FOR THE OBTAINING OF ACID DERIVATIVES 5- (N-3,4,5,6-TETRAHIDROFTALIMIDO) -CANIMICO. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NAV | Patent application has lapsed |
Ref document number: 7408321-3 Format of ref document f/p: F |