RU2012125812A - METHOD FOR PRODUCING ANTIBACTERIAL PRODUCT IN THE FORM OF POWDER FOR INJECTION SOLUTION - Google Patents
METHOD FOR PRODUCING ANTIBACTERIAL PRODUCT IN THE FORM OF POWDER FOR INJECTION SOLUTION Download PDFInfo
- Publication number
- RU2012125812A RU2012125812A RU2012125812/15A RU2012125812A RU2012125812A RU 2012125812 A RU2012125812 A RU 2012125812A RU 2012125812/15 A RU2012125812/15 A RU 2012125812/15A RU 2012125812 A RU2012125812 A RU 2012125812A RU 2012125812 A RU2012125812 A RU 2012125812A
- Authority
- RU
- Russia
- Prior art keywords
- cephalosporin
- powder
- antibacterial agent
- producing
- sulbactam
- Prior art date
Links
- 238000002347 injection Methods 0.000 title claims abstract 5
- 239000007924 injection Substances 0.000 title claims abstract 5
- 238000004519 manufacturing process Methods 0.000 title claims abstract 4
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 239000000243 solution Substances 0.000 title 1
- 229930186147 Cephalosporin Natural products 0.000 claims abstract 18
- 229940124587 cephalosporin Drugs 0.000 claims abstract 18
- 150000001780 cephalosporins Chemical class 0.000 claims abstract 18
- 239000000843 powder Substances 0.000 claims abstract 12
- 239000003242 anti bacterial agent Substances 0.000 claims abstract 10
- 238000000034 method Methods 0.000 claims abstract 9
- 229960005256 sulbactam Drugs 0.000 claims abstract 4
- 239000003781 beta lactamase inhibitor Substances 0.000 claims abstract 2
- 229940126813 beta-lactamase inhibitor Drugs 0.000 claims abstract 2
- HVFLCNVBZFFHBT-ZKDACBOMSA-N cefepime Chemical compound S([C@@H]1[C@@H](C(N1C=1C([O-])=O)=O)NC(=O)\C(=N/OC)C=2N=C(N)SC=2)CC=1C[N+]1(C)CCCC1 HVFLCNVBZFFHBT-ZKDACBOMSA-N 0.000 claims abstract 2
- 229960002100 cefepime Drugs 0.000 claims abstract 2
- GCFBRXLSHGKWDP-XCGNWRKASA-N cefoperazone Chemical compound O=C1C(=O)N(CC)CCN1C(=O)N[C@H](C=1C=CC(O)=CC=1)C(=O)N[C@@H]1C(=O)N2C(C(O)=O)=C(CSC=3N(N=NN=3)C)CS[C@@H]21 GCFBRXLSHGKWDP-XCGNWRKASA-N 0.000 claims abstract 2
- 229960004682 cefoperazone Drugs 0.000 claims abstract 2
- 229960000484 ceftazidime Drugs 0.000 claims abstract 2
- NMVPEQXCMGEDNH-TZVUEUGBSA-N ceftazidime pentahydrate Chemical compound O.O.O.O.O.S([C@@H]1[C@@H](C(N1C=1C([O-])=O)=O)NC(=O)\C(=N/OC(C)(C)C(O)=O)C=2N=C(N)SC=2)CC=1C[N+]1=CC=CC=C1 NMVPEQXCMGEDNH-TZVUEUGBSA-N 0.000 claims abstract 2
- 239000011261 inert gas Substances 0.000 claims abstract 2
- 239000003112 inhibitor Substances 0.000 claims abstract 2
- 239000002245 particle Substances 0.000 claims abstract 2
- FKENQMMABCRJMK-RITPCOANSA-N sulbactam Chemical compound O=S1(=O)C(C)(C)[C@H](C(O)=O)N2C(=O)C[C@H]21 FKENQMMABCRJMK-RITPCOANSA-N 0.000 claims abstract 2
- 229940126085 β‑Lactamase Inhibitor Drugs 0.000 claims abstract 2
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
1. Способ получения порошка антибактериального средства для раствора для инъекций на основе цефалоспорина и ингибитора β-лактамаз путем их смешивания, отличающийся тем, что как цефалоспорин используют цефалоспорин III или IV поколения, как ингибитор β-лактамаз-сульбактам, при молекулярном соотношении цефалоспорин/сульбактам (1,5-2,2):(2,1-2,2), предварительно компоненты измельчают с получением порошка с размером частиц 60 мкм и менее, а затем смешивают в указанном количестве, процесс проводят в атмосфере инертного газа.2. Способ получения порошка антибактериального средства по п.1, отличающийся тем, что как цефалоспорин используют цефтазидим.3. Способ получения порошка антибактериального средства по п.1, отличающийся тем, что как цефалоспорин используют цефоперазон.4. Способ получения порошка антибактериального средства по п.1, отличающийся тем, что как цефалоспорин используют цефепим.5. Способ получения порошка антибактериального средства по п.1, отличающийся тем, что как цефалоспорин используют цефпиром.1. A method of obtaining a powder of an antibacterial agent for injection for injection based on cephalosporin and a β-lactamase inhibitor by mixing them, characterized in that cephalosporin is used in generation III or IV cephalosporin, as a β-lactamase-sulbactam inhibitor, with a molecular ratio of cephalosporin / sulbactam (1.5-2.2) :( 2.1-2.2), the components are first crushed to obtain a powder with a particle size of 60 μm or less, and then mixed in the specified amount, the process is carried out in an inert gas atmosphere. 2. A method of obtaining a powder of an antibacterial agent according to claim 1, characterized in that ceftazidime is used as cephalosporin. A method for producing an antibacterial agent powder according to claim 1, characterized in that cefoperazone is used as cephalosporin. A method for producing an antibacterial agent powder according to claim 1, characterized in that cefepime is used as cephalosporin. A method of producing an antibacterial agent powder according to claim 1, characterized in that cephalosporin is used as cephalosporin.
Claims (5)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UAU201203787 | 2012-03-28 | ||
| UAU201203787U UA73553U (en) | 2012-03-28 | 2012-03-28 | Method for manufacturing powder of antibacterial agent for injectional solution |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RU2012125812A true RU2012125812A (en) | 2013-12-27 |
Family
ID=49785911
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2012125812/15A RU2012125812A (en) | 2012-03-28 | 2012-06-20 | METHOD FOR PRODUCING ANTIBACTERIAL PRODUCT IN THE FORM OF POWDER FOR INJECTION SOLUTION |
Country Status (2)
| Country | Link |
|---|---|
| RU (1) | RU2012125812A (en) |
| UA (1) | UA73553U (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN109864970A (en) * | 2019-04-22 | 2019-06-11 | 苏州东瑞制药有限公司 | A kind of sulbactam sodium composition aseptic powder and preparation method thereof |
-
2012
- 2012-03-28 UA UAU201203787U patent/UA73553U/en unknown
- 2012-06-20 RU RU2012125812/15A patent/RU2012125812A/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| UA73553U (en) | 2012-09-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA92 | Acknowledgement of application withdrawn (lack of supplementary materials submitted) |
Effective date: 20161025 |