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PT86695A - Process for the preparation of tetrahydropyridoý3',4':4,5¨pyrr oloý2,3-c¨quinolines and their derivatives - Google Patents

Process for the preparation of tetrahydropyridoý3',4':4,5¨pyrr oloý2,3-c¨quinolines and their derivatives

Info

Publication number
PT86695A
PT86695A PT86695A PT8669588A PT86695A PT 86695 A PT86695 A PT 86695A PT 86695 A PT86695 A PT 86695A PT 8669588 A PT8669588 A PT 8669588A PT 86695 A PT86695 A PT 86695A
Authority
PT
Portugal
Prior art keywords
oloý2
cinhinolines
pyrr
derivatives
preparation
Prior art date
Application number
PT86695A
Other languages
English (en)
Other versions
PT86695B (pt
Inventor
Karl Schoenafinger
Helen Hu Ong
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT86695A publication Critical patent/PT86695A/pt
Publication of PT86695B publication Critical patent/PT86695B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT86695A 1987-02-05 1988-02-04 Processo para a preparacao de tetra-hidro-pirido{3',4':4,5}pirrolo{2,3-c}quinolinas, dos seus intermediarios PT86695B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/012,715 US4771052A (en) 1987-02-05 1987-02-05 Tetrahydropyrido[3',4':4,5]pyrrolo[2,3-c]quinolines and their use as hypotensive agents

Publications (2)

Publication Number Publication Date
PT86695A true PT86695A (pt) 1988-03-01
PT86695B PT86695B (pt) 1992-04-30

Family

ID=21756344

Family Applications (1)

Application Number Title Priority Date Filing Date
PT86695A PT86695B (pt) 1987-02-05 1988-02-04 Processo para a preparacao de tetra-hidro-pirido{3',4':4,5}pirrolo{2,3-c}quinolinas, dos seus intermediarios

Country Status (6)

Country Link
US (1) US4771052A (pt)
EP (1) EP0277625A3 (pt)
JP (1) JPS63196584A (pt)
DK (1) DK56888A (pt)
IE (1) IE880306L (pt)
PT (1) PT86695B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5281608A (en) * 1992-08-28 1994-01-25 American Home Products Corporation Substituted tetrahydropyrido[3',4':4,5]-pyrrolo[3,2-c]quinolines
CN1477976A (zh) * 2000-11-30 2004-02-25 �Ʒ� Gaba激动剂与醛糖还原酶抑制剂的组合
GB0522715D0 (en) 2005-11-08 2005-12-14 Helperby Therapeutics Ltd New use
US11932641B1 (en) 2023-07-17 2024-03-19 King Faisal University Pyrido[4′,3′:4,5]pyrrolo[3,2-b][1,7]naphthyridine compounds as CK2 inhibitors
US11884668B1 (en) 2023-08-02 2024-01-30 King Faisal University Substituted pyrido[3′,4′:4,5]pyrrolo[2,3-c]quinolines as CK2 inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3272824A (en) * 1962-12-06 1966-09-13 Norwich Pharma Co 4-amino-6, 7-di(lower) alkoxyquinolines

Also Published As

Publication number Publication date
US4771052A (en) 1988-09-13
DK56888D0 (da) 1988-02-04
DK56888A (da) 1988-08-06
JPS63196584A (ja) 1988-08-15
IE880306L (en) 1988-08-05
EP0277625A3 (en) 1990-07-11
EP0277625A2 (en) 1988-08-10
PT86695B (pt) 1992-04-30

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Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19911016

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19930430