PL345037A1 - Cyclic somatostatin analogs - Google Patents

Cyclic somatostatin analogs

Info

Publication number: PL345037A1
Authority: PL; Poland
Prior art keywords: somatostatin analogs; cyclic somatostatin; cyclic; analogs; somatostatin
Prior art date: 1998-06-16

Application number

PL99345037A

Inventor

Thomas D Gordon

Original Assignee

Sod Conseils Rech Applic

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-06-16

Filing date

1999-06-11

Publication date

2001-11-19

1999-06-11 Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic

2001-11-19 Publication of PL345037A1 publication Critical patent/PL345037A1/en

Links

NHXLMOGPVYXJNR-ATOGVRKGSA-N somatostatin Chemical class C([C@H]1C(=O)N[C@H](C(N[C@@H](CO)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N1)[C@@H](C)O)NC(=O)CNC(=O)[C@H](C)N)C(O)=O)=O)[C@H](O)C)C1=CC=CC=C1 NHXLMOGPVYXJNR-ATOGVRKGSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Diabetes (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Hematology (AREA)
Obesity (AREA)
Emergency Medicine (AREA)
Pain & Pain Management (AREA)
Transplantation (AREA)
Ophthalmology & Optometry (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Urology & Nephrology (AREA)
Toxicology (AREA)
Zoology (AREA)
Gastroenterology & Hepatology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)

PL99345037A 1998-06-16 1999-06-11 Cyclic somatostatin analogs PL345037A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US8950398P	1998-06-16	1998-06-16
US9818198A	1998-06-16	1998-06-16
PCT/US1999/013304 WO1999065942A1 (en)	1998-06-16	1999-06-11	Cyclic somatostatin analogs

Publications (1)

Publication Number	Publication Date
PL345037A1 true PL345037A1 (en)	2001-11-19

Family

ID=26780645

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL99345037A PL345037A1 (en)	1998-06-16	1999-06-11	Cyclic somatostatin analogs

Country Status (12)

Country	Link
EP (1)	EP1086131A1 (en)
JP (1)	JP2002518409A (en)
CN (1)	CN1200000C (en)
AR (1)	AR021161A1 (en)
AU (1)	AU745493B2 (en)
CA (1)	CA2335184A1 (en)
HU (1)	HUP0102902A3 (en)
NO (1)	NO20006320L (en)
PL (1)	PL345037A1 (en)
RU (1)	RU2242481C2 (en)
TW (3)	TW527361B (en)
WO (1)	WO1999065942A1 (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP2003523921A (en)	1998-06-12	2003-08-12	ソシエテ・ドゥ・コンセイユ・ドゥ・ルシェルシュ・エ・ダプリカーション・シャンティフィック・エス・ア・エス	Imidazolyl derivatives
FR2796945B1 (en) *	1999-07-30	2002-06-28	Sod Conseils Rech Applic	NOVEL DERIVATIVES OF HYDANTOINS, THIOHYDANTOINS, PYRIMIDINEDIONES AND THIOXOPYRIMIDINONES, PROCESSES FOR THEIR PREPARATION AND THEIR APPLICATION AS MEDICAMENTS
AR035040A1 (en) *	2000-08-01	2004-04-14	Sod Conseils Rech Applic	IMIDAZOLIL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THE USE OF THEM FOR THE PREPARATION OF MEDICINES ABLE TO SELECTIVELY JOIN SUBTIPOS OF THE SOMATOSTATIN RECEIVER
US20040186151A1 (en) *	2003-02-12	2004-09-23	Mjalli Adnan M.M.	Substituted azole derivatives as therapeutic agents
WO2006063465A1 (en) *	2004-12-15	2006-06-22	Diamedica Inc.	Treatment of insulin resistance by modulating somatostatin using somatostatin receptor antagonists
ATE511502T1 (en)	2005-12-14	2011-06-15	Bristol Myers Squibb Co	ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPINAMIDE OR ARYLMETHYLUREA ANALOGUES AS FACTOR XIA INHIBITORS
CN101341129B (en) *	2005-12-14	2011-12-14	布里斯托尔-迈尔斯斯奎布公司	Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor xia inhibitors
EA201170493A1 (en)	2008-09-26	2011-10-31	Амбркс, Инк.	MICROORGANISMS AND VACCINES DEPENDING ON REPLICATION OF NON-NATURAL AMINO ACIDS
EP2168983A1 (en) *	2008-09-30	2010-03-31	Ipsen Pharma	New octapeptide compounds and their therapeutic use
WO2010050445A1 (en)	2008-10-27	2010-05-06	武田薬品工業株式会社	Bicyclic compound
IL320126A (en) *	2016-02-09	2025-06-01	Cdrd Ventures Inc	Somatostatin receptor antagonist compounds and methods of using the same

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5770687A (en) *	1995-06-07	1998-06-23	Peptor Limited	Comformationally constrained backbone cyclized somatostatin analogs
GB9513224D0 (en) *	1995-06-29	1995-09-06	Sandoz Ltd	Organic compounds
US6673927B2 (en) *	1996-02-16	2004-01-06	Societe De Conseils De Recherches Et D'applications Scientifiques, S.A.S.	Farnesyl transferase inhibitors

1999
- 1999-06-11 RU RU2001101530/04A patent/RU2242481C2/en not_active IP Right Cessation
- 1999-06-11 PL PL99345037A patent/PL345037A1/en not_active Application Discontinuation
- 1999-06-11 HU HU0102902A patent/HUP0102902A3/en unknown
- 1999-06-11 JP JP2000554767A patent/JP2002518409A/en active Pending
- 1999-06-11 AU AU48223/99A patent/AU745493B2/en not_active Ceased
- 1999-06-11 CN CNB998075027A patent/CN1200000C/en not_active Expired - Fee Related
- 1999-06-11 EP EP99931793A patent/EP1086131A1/en not_active Withdrawn
- 1999-06-11 WO PCT/US1999/013304 patent/WO1999065942A1/en not_active Ceased
- 1999-06-11 CA CA002335184A patent/CA2335184A1/en not_active Abandoned
- 1999-06-15 TW TW088110016A patent/TW527361B/en not_active IP Right Cessation
- 1999-06-15 TW TW091115003A patent/TWI242441B/en active
- 1999-06-15 AR ARP990102857A patent/AR021161A1/en unknown
- 1999-06-15 TW TW093100348A patent/TWI242442B/en active
2000
- 2000-12-12 NO NO20006320A patent/NO20006320L/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
NO20006320D0 (en)	2000-12-12
EP1086131A1 (en)	2001-03-28
WO1999065942A1 (en)	1999-12-23
AU745493B2 (en)	2002-03-21
NO20006320L (en)	2001-02-12
TW200410986A (en)	2004-07-01
WO1999065942A8 (en)	2000-02-17
AR021161A1 (en)	2002-07-03
RU2242481C2 (en)	2004-12-20
CN1305496A (en)	2001-07-25
TWI242441B (en)	2005-11-01
AU4822399A (en)	2000-01-05
TWI242442B (en)	2005-11-01
JP2002518409A (en)	2002-06-25
TW527361B (en)	2003-04-11
CN1200000C (en)	2005-05-04
HUP0102902A2 (en)	2002-01-28
CA2335184A1 (en)	1999-12-23
HUP0102902A3 (en)	2002-02-28

Publication	Publication Date	Title
SI1307486T1 (en)	2008-08-31	Somatostatin analogues
CZ20011342A3 (en)	2001-09-12	Cyclic tetrapeptides
CZ20012876A3 (en)	2002-06-12	SP-C analogs
IL139885A0 (en)	2002-02-10	Cyclic boroproline compounds
HUP0202812A3 (en)	2005-01-28	Novel bicyclonucleoside analogues
GB9926183D0 (en)	2000-01-12	LED components
ZA9830B (en)	1999-07-05	Cyclic sulfone derivatives
AU4114201A (en)	2001-11-12	Cyclic compounds
DE69941708D1 (en)	2010-01-07	PACAP PEPTIDE ANALOGS
EP0996458A4 (en)	2001-05-02	SANDRAMYCIN ANALOGS
AU4524401A (en)	2001-06-25	Receptor-selective somatostatin analogs
EG23909A (en)	2007-12-30	Vatamin d, analogs
PL348763A1 (en)	2002-06-03	Phenyl-substituted cyclic enaminones
IL141276A0 (en)	2002-03-10	Backbone cyclized radiolabelled somatostatin analogs
PL345037A1 (en)	2001-11-19	Cyclic somatostatin analogs
IL139218A0 (en)	2001-11-25	2-aroyl-4-acyl-paclitaxel (taxol) analogs
ZA985896B (en)	1999-06-14	Cyclic azapeptides
EP1233774A4 (en)	2004-06-16	Urotensin-ii analogs
GB9823835D0 (en)	1998-12-23	Component for vaccine
AU1126300A (en)	2000-06-13	Hydrophilic somatostatin analogs
GB9929433D0 (en)	2000-02-09	Cyclic compound
AU6382999A (en)	2000-03-14	Somatostatin analogs
TW329729U (en)	1998-04-11	Cyclic tool
GB9828612D0 (en)	1999-02-17	Sequence
GB9823638D0 (en)	1998-12-23	Sequence

Legal Events

Date	Code	Title	Description
2007-12-31	REFS	Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)