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PE20201494A1 - Anticuerpo anti-pacap - Google Patents

Anticuerpo anti-pacap

Info

Publication number
PE20201494A1
PE20201494A1 PE2020000375A PE2020000375A PE20201494A1 PE 20201494 A1 PE20201494 A1 PE 20201494A1 PE 2020000375 A PE2020000375 A PE 2020000375A PE 2020000375 A PE2020000375 A PE 2020000375A PE 20201494 A1 PE20201494 A1 PE 20201494A1
Authority
PE
Peru
Prior art keywords
seq
antibody
variable region
heavy chain
light chain
Prior art date
Application number
PE2020000375A
Other languages
English (en)
Inventor
Catherine Brautigam Beidler
Michael Parvin Johnson
Chetankumar Natvarlal Patel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PE20201494A1 publication Critical patent/PE20201494A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/005Enzyme inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/177Receptors; Cell surface antigens; Cell surface determinants
    • A61K38/1796Receptors; Cell surface antigens; Cell surface determinants for hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/76Antagonist effect on antigen, e.g. neutralization or inhibition of binding
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/92Affinity (KD), association rate (Ka), dissociation rate (Kd) or EC50 value
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/94Stability, e.g. half-life, pH, temperature or enzyme-resistance

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Cell Biology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Endocrinology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se refiere a un anticuerpo que se une al peptido activador de la adenilato ciclasa de la pituitaria humana (PACAP), el cual comprende una region variable de cadena pesada (HCVR) es la SEQ ID NO.9 que comprende regiones determinantes de la complementariedad HCDR1 cuya secuencia de aminoacidos es la SEQ ID NO.3, HCDR2 es la SEQ ID NO.4 y HCDR3 es la SEQ ID NO.5; y comprende una region variable de cadena ligera (LCVR) es la SEQ ID NO. 10 que comprende LCDR1 es la SEQ ID NO.6, LCDR2 es la SEQ ID NO.7 y LCDR3 es la SEQ ID NO.8; asi como una cadena pesada (HC) que comprende la SEQ ID NO.1 y una cadena ligera (LC) que comprende la SEQ ID NO.2. Dicho anticuerpo es util en el tratamiento del dolor incluyendo cefalea y/o migrana.
PE2020000375A 2017-09-29 2018-09-20 Anticuerpo anti-pacap PE20201494A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762565278P 2017-09-29 2017-09-29
PCT/US2018/051898 WO2019067293A1 (en) 2017-09-29 2018-09-20 ANTI-PACAP ANTIBODIES

Publications (1)

Publication Number Publication Date
PE20201494A1 true PE20201494A1 (es) 2020-12-29

Family

ID=63794713

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2020000375A PE20201494A1 (es) 2017-09-29 2018-09-20 Anticuerpo anti-pacap

Country Status (27)

Country Link
US (3) US10519225B2 (es)
EP (1) EP3688035A1 (es)
JP (2) JP6952888B2 (es)
KR (1) KR102453573B1 (es)
CN (1) CN111164105B (es)
AR (1) AR113022A1 (es)
AU (1) AU2018341959B2 (es)
BR (1) BR112020003628A2 (es)
CA (1) CA3077304C (es)
CL (1) CL2020000705A1 (es)
CO (1) CO2020002170A2 (es)
CR (1) CR20200127A (es)
DO (1) DOP2020000060A (es)
EA (1) EA202090563A1 (es)
EC (1) ECSP20020293A (es)
IL (1) IL273529A (es)
JO (1) JOP20200069A1 (es)
MA (1) MA50654A (es)
MX (1) MX2020003563A (es)
MY (1) MY199876A (es)
NZ (1) NZ762312A (es)
PE (1) PE20201494A1 (es)
PH (1) PH12020550340A1 (es)
SG (1) SG11202002572YA (es)
TW (1) TWI701260B (es)
WO (1) WO2019067293A1 (es)
ZA (1) ZA202001058B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2017013113A (es) 2015-04-16 2018-07-06 Alder Biopharmaceuticals Inc Anticuerpos anti-pacap y sus usos.
CA3020839A1 (en) 2016-04-15 2017-10-19 Alder Biopharmaceuticals, Inc. Anti-pacap antibodies and uses thereof
CA3154522A1 (en) 2019-10-15 2021-04-22 Christopher Carl Frye Recombinantly engineered, lipase/esterase-deficient mammalian cell lines
CA3227549A1 (en) 2021-07-29 2023-02-02 Cephalon Llc Compositions and methods for anti-pacap antibodies
WO2023051786A1 (zh) * 2021-09-30 2023-04-06 江苏恒瑞医药股份有限公司 特异性结合cgrp和pacap的抗原结合分子及其医药用途
KR102839881B1 (ko) * 2021-11-19 2025-07-31 대한민국 방송통신기자재 성능 측정 시스템 및 그 방법
WO2024218541A1 (en) * 2023-04-20 2024-10-24 Mark Hasleton Treatment of migraine

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE210680T1 (de) * 1990-03-17 2001-12-15 Takeda Chemical Industries Ltd Antikörper gegen hypophysäre adenylatzyklase aktivierende peptid-pacap, hybridome und bestimmung von pacap
US6037321A (en) 1995-05-03 2000-03-14 Biostar Inc. Fusion proteins comprising vasoactive intestinal peptide or PACAP
FR2826747B1 (fr) 2001-07-02 2005-02-25 Gemplus Card Int Procede et dispositif de traitement de donnees pour la personnalisation d'une application sur un dispositif communicant portatif, par exemple une carte a puce
US7615219B2 (en) 2003-01-16 2009-11-10 Life Sciences Research Partners Vzw Inhibition of PACAP signalling for the prevention and treatment of thrombocytopenia
WO2012106407A2 (en) 2011-02-01 2012-08-09 The University Of Vermont And State Agricultural College Diagnostic and therapeutic methods and products related to anxiety disorders
JP6064861B2 (ja) 2013-03-05 2017-01-25 株式会社デンソー 熱電変換装置の製造方法
PE20151923A1 (es) * 2013-03-15 2016-01-14 Amgen Inc Anticuerpos humanos pac1
EP3035950A4 (en) 2013-08-14 2017-05-03 The Arizona Board Of Regents On Behalf Of The University Of Arizona Glycosylated pacap/vip analogues with enhanced cns penetration for treatment of neurodegenerative diseases
MX2017013113A (es) 2015-04-16 2018-07-06 Alder Biopharmaceuticals Inc Anticuerpos anti-pacap y sus usos.
WO2017106578A1 (en) * 2015-12-15 2017-06-22 Amgen Inc. Pacap antibodies and uses thereof
WO2017142961A1 (en) 2016-02-16 2017-08-24 The Arizona Board Of Regents On Behalf Of The University Of Arizona Treatment of traumatic brain injury or stroke

Also Published As

Publication number Publication date
AU2018341959B2 (en) 2021-11-25
TW201920280A (zh) 2019-06-01
TWI701260B (zh) 2020-08-11
WO2019067293A1 (en) 2019-04-04
US20190100579A1 (en) 2019-04-04
MY199876A (en) 2023-11-27
ZA202001058B (en) 2022-06-29
CL2020000705A1 (es) 2020-09-11
DOP2020000060A (es) 2020-08-15
CA3077304C (en) 2023-08-01
AR113022A1 (es) 2020-01-15
NZ762312A (en) 2022-11-25
US10519225B2 (en) 2019-12-31
BR112020003628A2 (pt) 2020-09-01
CN111164105B (zh) 2023-07-04
AU2018341959A1 (en) 2020-03-05
KR102453573B1 (ko) 2022-10-12
MX2020003563A (es) 2020-08-03
JP7221352B2 (ja) 2023-02-13
KR20200040881A (ko) 2020-04-20
US10954292B2 (en) 2021-03-23
EP3688035A1 (en) 2020-08-05
IL273529A (en) 2020-05-31
JP2020535167A (ja) 2020-12-03
PH12020550340A1 (en) 2022-05-02
CA3077304A1 (en) 2019-04-04
JP6952888B2 (ja) 2021-10-27
SG11202002572YA (en) 2020-04-29
CN111164105A (zh) 2020-05-15
JOP20200069A1 (ar) 2020-04-28
ECSP20020293A (es) 2020-06-30
JP2022000049A (ja) 2022-01-04
US20200131256A1 (en) 2020-04-30
US20210171616A1 (en) 2021-06-10
EA202090563A1 (ru) 2020-06-24
CR20200127A (es) 2020-04-08
CO2020002170A2 (es) 2020-04-01
MA50654A (fr) 2020-08-05

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