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PE20070698A1 - Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol - Google Patents

Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol

Info

Publication number
PE20070698A1
PE20070698A1 PE2006001419A PE2006001419A PE20070698A1 PE 20070698 A1 PE20070698 A1 PE 20070698A1 PE 2006001419 A PE2006001419 A PE 2006001419A PE 2006001419 A PE2006001419 A PE 2006001419A PE 20070698 A1 PE20070698 A1 PE 20070698A1
Authority
PE
Peru
Prior art keywords
disgregation
composition
ambroxol hydrochloride
amount
tablet containing
Prior art date
Application number
PE2006001419A
Other languages
English (en)
Inventor
Tomoya Akutagawa
Masahiko Narasaki
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Publication of PE20070698A1 publication Critical patent/PE20070698A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/131Amines acyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/375Ascorbic acid, i.e. vitamin C; Salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Zoology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA SOLIDA TAL COMO UN COMPRIMIDO DE DISGREGACION RAPIDA INTRAORAL QUE COMPRENDE: A) UN GRANULO QUE TIENE UN ESPACIO VACIO DENTRO DEL MISMO QUE CONTIENE i) UN DESINTEGRANTE TAL COMO CROSPOVIDONA EN UNA CANTIDAD DE 4% A 20% EN PESO DE LA COMPOSICION; ii) HIDROCLORURO DE AMBROXOL; iii) ERITRITOL O MANITOL; B) UN DESINTEGRANTE UTILIZADO COMO RECUBRIMIENTO DEL GRANULO TAL COMO CROSPOVIDONA EN UNA CANTIDAD DE 4% A 20% EN PESO DE LA COMPOSICION; C) UN LUBRICANTE TAL COMO ACIDO SILICICO ANHIDRO LIGERO O UNA SAL DE ESTEARATO. SE REFIERE TAMBIEN A UN PROCEDIMIENTO DE PREPARACION. DICHA COMPOSICION SE DESINTEGRA RAPIDAMENTE CON UNA BUENA SENSACION EN LA CAVIDAD ORAL
PE2006001419A 2005-11-14 2006-11-13 Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol PE20070698A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005328722 2005-11-14

Publications (1)

Publication Number Publication Date
PE20070698A1 true PE20070698A1 (es) 2007-08-17

Family

ID=38023405

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2006001419A PE20070698A1 (es) 2005-11-14 2006-11-13 Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol

Country Status (12)

Country Link
US (2) US10300021B2 (es)
EP (2) EP1951203A4 (es)
JP (2) JP4934144B2 (es)
KR (1) KR101298379B1 (es)
CN (2) CN103637996A (es)
AR (1) AR057581A1 (es)
AU (1) AU2006312566B2 (es)
CA (1) CA2629487C (es)
ES (1) ES2702757T3 (es)
PE (1) PE20070698A1 (es)
TW (1) TWI478732B (es)
WO (2) WO2007055427A1 (es)

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* Cited by examiner, † Cited by third party
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PE20070698A1 (es) 2005-11-14 2007-08-17 Teijin Pharma Ltd Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol
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JP6718866B2 (ja) 2014-10-16 2020-07-08 カーギル インコーポレイテッド 直接圧縮性のエリスリトールの調製方法及びその使用
ES2982524T3 (es) * 2016-06-16 2024-10-16 Towa Pharmaceutical Co Ltd Comprimido de disgregación por vía oral
TWI767923B (zh) * 2016-07-27 2022-06-21 日商澤井製藥股份有限公司 口腔內崩解錠添加用組成物及其製造方法以及口腔內崩解錠
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KR20230087405A (ko) 2021-12-09 2023-06-16 블룸 에너지 코퍼레이션 연료 활용도가 100 퍼센트에 가까운 연료 전지 시스템 및 이의 동작 방법

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Also Published As

Publication number Publication date
EP1951203A4 (en) 2011-07-06
CA2629487C (en) 2014-11-18
AU2006312566B2 (en) 2012-04-12
EP1957051B1 (en) 2018-11-14
CA2629487A1 (en) 2007-05-18
JP2009515871A (ja) 2009-04-16
US20100009004A1 (en) 2010-01-14
AR057581A1 (es) 2007-12-05
JP2011225624A (ja) 2011-11-10
WO2007055428A1 (en) 2007-05-18
TW200738282A (en) 2007-10-16
EP1957051A1 (en) 2008-08-20
US20090117182A1 (en) 2009-05-07
KR20080073335A (ko) 2008-08-08
EP1957051A4 (en) 2011-07-06
WO2007055427A1 (en) 2007-05-18
AU2006312566A1 (en) 2007-05-18
CN101309672A (zh) 2008-11-19
US10300021B2 (en) 2019-05-28
EP1951203A1 (en) 2008-08-06
JP4934144B2 (ja) 2012-05-16
CN101309672B (zh) 2015-07-29
KR101298379B1 (ko) 2013-08-20
US9511029B2 (en) 2016-12-06
ES2702757T3 (es) 2019-03-05
CN103637996A (zh) 2014-03-19
TWI478732B (zh) 2015-04-01

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