PE20020903A1 - Metodo para prevenir la diarrea - Google Patents
Metodo para prevenir la diarreaInfo
- Publication number
- PE20020903A1 PE20020903A1 PE2001000284A PE2001000284A PE20020903A1 PE 20020903 A1 PE20020903 A1 PE 20020903A1 PE 2001000284 A PE2001000284 A PE 2001000284A PE 2001000284 A PE2001000284 A PE 2001000284A PE 20020903 A1 PE20020903 A1 PE 20020903A1
- Authority
- PE
- Peru
- Prior art keywords
- octreotide
- irinotecan
- administration
- refers
- prevent diarrhea
- Prior art date
Links
- 206010012735 Diarrhoea Diseases 0.000 title abstract 3
- DEQANNDTNATYII-OULOTJBUSA-N (4r,7s,10s,13r,16s,19r)-10-(4-aminobutyl)-19-[[(2r)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-n-[(2r,3r)-1,3-dihydroxybutan-2-yl]-7-[(1r)-1-hydroxyethyl]-13-(1h-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxa Chemical compound C([C@@H](N)C(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC=2C3=CC=CC=C3NC=2)NC(=O)[C@H](CC=2C=CC=CC=2)NC1=O)C(=O)N[C@H](CO)[C@H](O)C)C1=CC=CC=C1 DEQANNDTNATYII-OULOTJBUSA-N 0.000 abstract 2
- 108010016076 Octreotide Proteins 0.000 abstract 2
- UWKQSNNFCGGAFS-XIFFEERXSA-N irinotecan Chemical compound C1=C2C(CC)=C3CN(C(C4=C([C@@](C(=O)OC4)(O)CC)C=4)=O)C=4C3=NC2=CC=C1OC(=O)N(CC1)CCC1N1CCCCC1 UWKQSNNFCGGAFS-XIFFEERXSA-N 0.000 abstract 2
- 229960004768 irinotecan Drugs 0.000 abstract 2
- 229960002700 octreotide Drugs 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- QTBSBXVTEAMEQO-UHFFFAOYSA-M Acetate Chemical compound CC([O-])=O QTBSBXVTEAMEQO-UHFFFAOYSA-M 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- 239000002207 metabolite Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/31—Somatostatins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Zoology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
SE REFIERE A UN METODO PARA PREVENIR LA DIARREA CAUSADA POR LA ADMINISTRACION DE IRINOTECAN O UNA SAL O UN METABOLITO FARMACEUTICAMENTE ACEPTABLE QUE COMPRENDE ADMINISTRAR A UN PACIENTE UNA CANTIDAD EFECTIVA DE UN OCTREOTIDO EN FORMA DE SAL ACETATO. EL OCTREOTIDO SE FORMULA EN UNA FORMA DE DOSIFICACION DE LIBERACION CON ACCION PROLONGADA. SE REFIERE TAMBIEN A FORMULACIONES DE COMBINACION Y A KITS PARA PREVENIR LA DIARREA PROVOCADA POR EL IRINOTECAN O LA ADMINISTRACION DE UN ANALOGO DE CAMPTOTECINA
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/450,201 US6159935A (en) | 1999-11-29 | 1999-11-29 | Method for preventing diarrhea |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20020903A1 true PE20020903A1 (es) | 2002-10-23 |
Family
ID=23787180
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2001000284A PE20020903A1 (es) | 1999-11-29 | 2001-03-27 | Metodo para prevenir la diarrea |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US6159935A (es) |
| AR (1) | AR026606A1 (es) |
| AU (1) | AU3439301A (es) |
| CO (1) | CO5271647A1 (es) |
| PE (1) | PE20020903A1 (es) |
| WO (1) | WO2001037784A2 (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20060205681A1 (en) * | 2002-06-21 | 2006-09-14 | Maryam Moaddeb | Homogenous paste formulations |
| US7396855B2 (en) | 2002-07-24 | 2008-07-08 | Children's Hospital Medical Center | Compositions and products containing S-equol, and methods for their making |
| PT1787658E (pt) | 2005-11-10 | 2012-06-22 | Chemi Spa | Formulações de libertação sustentada de análogos de somatostatina inibidores da hormona do crescimento |
| AU2009294320B2 (en) | 2008-09-17 | 2015-04-16 | Amryt Endo, Inc. | Pharmaceutical compositions and related methods of delivery |
| AU2016215350B2 (en) | 2015-02-03 | 2021-11-25 | Amryt Endo, Inc. | Method of treating diseases |
| MA43800A (fr) * | 2016-01-21 | 2021-05-12 | Chiasma Inc | Octréotide par voie orale pour le traitement de maladies |
| US11141457B1 (en) | 2020-12-28 | 2021-10-12 | Amryt Endo, Inc. | Oral octreotide therapy and contraceptive methods |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19375086I2 (de) * | 1979-11-27 | 2003-01-09 | Novartis Ag | Polypeptide Verfahren zu ihrer Herstellung pharmazeutische Zusammensetzungen die diese Polypeptide enthalten und ihre Verwendung |
| US4473692A (en) * | 1981-09-04 | 1984-09-25 | Kabushiki Kaisha Yakult Honsha | Camptothecin derivatives and process for preparing same |
| JPS6019790A (ja) * | 1983-07-14 | 1985-01-31 | Yakult Honsha Co Ltd | 新規なカンプトテシン誘導体 |
| PH30995A (en) | 1989-07-07 | 1997-12-23 | Novartis Inc | Sustained release formulations of water soluble peptides. |
| US5786344A (en) | 1994-07-05 | 1998-07-28 | Arch Development Corporation | Camptothecin drug combinations and methods with reduced side effects |
| US5789411A (en) | 1995-09-11 | 1998-08-04 | Lance L. Gooberman P. C. | Improvements to rapid opioid detoxification |
| US5919760A (en) | 1996-04-12 | 1999-07-06 | Intensive Narcotic Detoxification Centers Of America, Llc | Method for treating acute and severe diarrhea |
| BR9807271A (pt) * | 1997-02-27 | 2000-05-23 | Pharmacia & Upjohn Spa | Tamoxifeno como terapia para reduzir diarréia induzida por cloridrato de irinotecano |
-
1999
- 1999-11-29 US US09/450,201 patent/US6159935A/en not_active Expired - Fee Related
-
2000
- 2000-08-25 US US09/648,270 patent/US6395708B1/en not_active Expired - Fee Related
- 2000-11-13 WO PCT/US2000/042136 patent/WO2001037784A2/en not_active Ceased
- 2000-11-13 AU AU34393/01A patent/AU3439301A/en not_active Abandoned
- 2000-11-27 AR ARP000106218A patent/AR026606A1/es unknown
- 2000-11-27 CO CO00090627A patent/CO5271647A1/es not_active Application Discontinuation
-
2001
- 2001-03-27 PE PE2001000284A patent/PE20020903A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US6159935A (en) | 2000-12-12 |
| WO2001037784A2 (en) | 2001-05-31 |
| US6395708B1 (en) | 2002-05-28 |
| AU3439301A (en) | 2001-06-04 |
| AR026606A1 (es) | 2003-02-19 |
| CO5271647A1 (es) | 2003-04-30 |
| WO2001037784A3 (en) | 2002-05-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |