ITTO20060560A1 - INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF ANTIGONISTS OF ANGIOTENSINA II - Google Patents
INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF ANTIGONISTS OF ANGIOTENSINA IIInfo
- Publication number
- ITTO20060560A1 ITTO20060560A1 ITTO20060560A ITTO20060560A1 IT TO20060560 A1 ITTO20060560 A1 IT TO20060560A1 IT TO20060560 A ITTO20060560 A IT TO20060560A IT TO20060560 A1 ITTO20060560 A1 IT TO20060560A1
- Authority
- IT
- Italy
- Prior art keywords
- angiotensina
- antigonists
- preparation
- intermediate compounds
- compounds
- Prior art date
Links
- CZGUSIXMZVURDU-UHFFFAOYSA-N 3-azaniumyl-4-[[1-[[1-[[1-[[1-[[1-[2-[(1-carboxylato-2-phenylethyl)carbamoyl]pyrrolidin-1-yl]-3-(1h-imidazol-5-yl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-(diam Chemical compound C=1N=CNC=1CC(C(=O)N1C(CCC1)C(=O)NC(CC=1C=CC=CC=1)C(O)=O)NC(=O)C(C(C)CC)NC(=O)C(NC(=O)C(NC(=O)C(CCCN=C(N)N)NC(=O)C(N)CC(O)=O)C(C)C)CC1=CC=C(O)C=C1 CZGUSIXMZVURDU-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D257/04—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITTO20060560 ITTO20060560A1 (en) | 2006-07-27 | 2006-07-27 | INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF ANTIGONISTS OF ANGIOTENSINA II |
| PCT/IT2007/000031 WO2008012852A1 (en) | 2006-07-27 | 2007-01-16 | Intermediate compounds for the preparation of angiotensin ii antagonists |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITTO20060560 ITTO20060560A1 (en) | 2006-07-27 | 2006-07-27 | INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF ANTIGONISTS OF ANGIOTENSINA II |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ITTO20060560A1 true ITTO20060560A1 (en) | 2008-01-28 |
Family
ID=37965010
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ITTO20060560 ITTO20060560A1 (en) | 2006-07-27 | 2006-07-27 | INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF ANTIGONISTS OF ANGIOTENSINA II |
Country Status (2)
| Country | Link |
|---|---|
| IT (1) | ITTO20060560A1 (en) |
| WO (1) | WO2008012852A1 (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011084848A2 (en) | 2010-01-07 | 2011-07-14 | Alkermes, Inc. | Prodrugs of heteraromatic compounds |
| CN102351804B (en) * | 2011-09-30 | 2013-07-31 | 浙江新赛科药业有限公司 | Method for recovering valsartan racemate |
| CN102875534B (en) * | 2012-09-10 | 2015-05-27 | 珠海保税区丽珠合成制药有限公司 | Synthetic method of irbesartan |
| WO2019235493A1 (en) * | 2018-06-08 | 2019-12-12 | 株式会社トクヤマ | Method for producing diaminobenzoic acid ester |
| US11655220B2 (en) | 2020-10-22 | 2023-05-23 | Hetero Labs Limited | Process for the preparation of angiotensin II receptor blockers |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE194603T1 (en) * | 1994-01-28 | 2000-07-15 | Takeda Chemical Industries Ltd | A PROCESS FOR PRODUCING TETRAZOLYL COMPOUNDS |
| HU222773B1 (en) * | 2000-04-21 | 2003-10-28 | Richter Gedeon Vegyészeti Gyár Rt. | Process for producing a known tetrazole derivative |
| WO2005116010A1 (en) * | 2004-05-26 | 2005-12-08 | Merck Frosst Canada Ltd. | Ep4 receptor agonist, compositions and methods thereof |
-
2006
- 2006-07-27 IT ITTO20060560 patent/ITTO20060560A1/en unknown
-
2007
- 2007-01-16 WO PCT/IT2007/000031 patent/WO2008012852A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008012852A1 (en) | 2008-01-31 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR19C1035I2 (en) | FUNGICIDAL COMPOSITIONS | |
| LTC2004635I2 (en) | Substituted enaminocarbonyl compounds | |
| FR17C1014I2 (en) | FUNGICIDAL COMPOSITIONS | |
| PL2123158T3 (en) | Herbicidal composition | |
| BRPI0914746A2 (en) | fungicidal compositions | |
| EP1996710A4 (en) | ANTIREAL RIFAXIMINE DYSFUNCTION MANUFACTURE | |
| BRPI0716325A2 (en) | ANTIMICROBIAN COMPOSITION | |
| BRPI0720216A2 (en) | MICROBICIDE COMPOSITIONS | |
| BRPI0922904A2 (en) | "compounds" | |
| EP1985620A4 (en) | 10a-azalide compound | |
| ATE524477T1 (en) | AZIRIDINYLEPOTHILONE COMPOUNDS | |
| ATE485357T1 (en) | DISHWASHING COMPOSITION | |
| EP2043136A4 (en) | FILMOGENE COMPOSITION | |
| FR2899479B1 (en) | CICATRISANTE COMPOSITION | |
| ITMI20052486A1 (en) | INTERMEDIATE SYNTHESIS PROCEDURE FOR THE PREPARATION OF ASTAXANTIN | |
| CY2200166T2 (en) | IMPROVED SLIDE ANCHOR | |
| DK1776090T3 (en) | Stabilized prostaglandin composition | |
| DE602006021644D1 (en) | fungicidal compositions | |
| DE602007012490D1 (en) | herbicidal composition | |
| NO20055643D0 (en) | Preparation of lodixanol | |
| EP1993006A4 (en) | CHRONOGRAPH | |
| BRPI0622061A2 (en) | VIRUCIDAL COMPOSITION | |
| DK1977652T3 (en) | confectionary composition | |
| BRPI0716378A2 (en) | agriculturally useful compositions | |
| ITTO20060560A1 (en) | INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF ANTIGONISTS OF ANGIOTENSINA II |