[go: up one dir, main page]

ITMI942626A0 - Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni - Google Patents

Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni

Info

Publication number
ITMI942626A0
ITMI942626A0 ITMI942626A ITMI942626A ITMI942626A0 IT MI942626 A0 ITMI942626 A0 IT MI942626A0 IT MI942626 A ITMI942626 A IT MI942626A IT MI942626 A ITMI942626 A IT MI942626A IT MI942626 A0 ITMI942626 A0 IT MI942626A0
Authority
IT
Italy
Prior art keywords
azaandrostanes
antiandrogens
thioxo
oxo
compounds derived
Prior art date
Application number
ITMI942626A
Other languages
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Ambrogio Magni
Vincenzo Olgiati
Original Assignee
Poli Ind Chimica Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Poli Ind Chimica Spa filed Critical Poli Ind Chimica Spa
Publication of ITMI942626A0 publication Critical patent/ITMI942626A0/it
Priority to ITMI942626A priority Critical patent/IT1271325B/it
Priority to AU43872/96A priority patent/AU4387296A/en
Priority to DE69523622T priority patent/DE69523622T2/de
Priority to ES95942689T priority patent/ES2163538T3/es
Priority to PCT/EP1995/005008 priority patent/WO1996020210A2/en
Priority to EP95942689A priority patent/EP0799239B1/en
Priority to US08/879,442 priority patent/US6147213A/en
Priority to PT95942689T priority patent/PT799239E/pt
Priority to DK95942689T priority patent/DK0799239T3/da
Priority to AT95942689T priority patent/ATE207929T1/de
Publication of ITMI942626A1 publication Critical patent/ITMI942626A1/it
Application granted granted Critical
Publication of IT1271325B publication Critical patent/IT1271325B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ITMI942626A 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni IT1271325B (it)

Priority Applications (10)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
DE69523622T DE69523622T2 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza-androstanderivate und ihre verwendung als antiandrogene
ES95942689T ES2163538T3 (es) 1994-12-23 1995-12-18 Derivados de 3-oxo y 3-tioxo-4-aza-androstano diastereomericamente puros y su uso como antiandrogenos.
AU43872/96A AU4387296A (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
EP95942689A EP0799239B1 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
US08/879,442 US6147213A (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
PT95942689T PT799239E (pt) 1994-12-23 1995-12-18 Derivados diastereomericamente puros de 3-oxo e 3-tioxo-4-aza-androstano e a sua utilizacao como anti-androgenos
DK95942689T DK0799239T3 (da) 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener
AT95942689T ATE207929T1 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni

Publications (3)

Publication Number Publication Date
ITMI942626A0 true ITMI942626A0 (it) 1994-12-23
ITMI942626A1 ITMI942626A1 (it) 1996-06-23
IT1271325B IT1271325B (it) 1997-05-27

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni

Country Status (10)

Country Link
US (1) US6147213A (it)
EP (1) EP0799239B1 (it)
AT (1) ATE207929T1 (it)
AU (1) AU4387296A (it)
DE (1) DE69523622T2 (it)
DK (1) DK0799239T3 (it)
ES (1) ES2163538T3 (it)
IT (1) IT1271325B (it)
PT (1) PT799239E (it)
WO (1) WO1996020210A2 (it)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
WO2008061212A2 (en) 2006-11-15 2008-05-22 Energ2, Inc. Electric double layer capacitance device
US8552061B2 (en) * 2007-05-03 2013-10-08 Yale University Locally active “soft” antiandrogens
EP4461703A3 (en) 2009-07-01 2025-03-05 BASF Mobile Emissions Catalysts LLC Ultrapure synthetic carbon materials
BR112012014092A2 (pt) * 2009-12-11 2016-07-05 Energ2 Technologies Inc materiais de carvão compreendendo um modificador eletroquímico.
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
US8654507B2 (en) 2010-09-30 2014-02-18 Energ2 Technologies, Inc. Enhanced packing of energy storage particles
WO2012092210A1 (en) 2010-12-28 2012-07-05 Energ2 Technologies, Inc. Carbon materials comprising enhanced electrochemical properties
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
EP2715840B1 (en) 2011-06-03 2015-05-27 Basf Se Carbon-lead blends for use in hybrid energy storage devices
US9409777B2 (en) 2012-02-09 2016-08-09 Basf Se Preparation of polymeric resins and carbon materials
CN105190948B (zh) 2013-03-14 2019-04-26 14族科技公司 包含锂合金化的电化学改性剂的复合碳材料
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
WO2015137980A1 (en) 2014-03-14 2015-09-17 Energ2 Technologies, Inc. Novel methods for sol-gel polymerization in absence of solvent and creation of tunable carbon structure from same
WO2017030995A1 (en) 2015-08-14 2017-02-23 Energ2 Technologies, Inc. Nano-featured porous silicon materials
EP4286355A3 (en) 2015-08-28 2024-05-01 Group14 Technologies, Inc. Novel materials with extremely durable intercalation of lithium and manufacturing methods thereof
US11611071B2 (en) 2017-03-09 2023-03-21 Group14 Technologies, Inc. Decomposition of silicon-containing precursors on porous scaffold materials
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
EP4222109A1 (en) 2020-09-30 2023-08-09 Group14 Technologies, Inc. Methods of passivation to control oxygen content and reactivity of silicon-carbon composite materials

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
EP0799239B1 (en) 2001-10-31
DE69523622D1 (de) 2001-12-06
WO1996020210A3 (en) 1996-09-06
ITMI942626A1 (it) 1996-06-23
DK0799239T3 (da) 2001-12-10
AU4387296A (en) 1996-07-19
ES2163538T3 (es) 2002-02-01
WO1996020210A2 (en) 1996-07-04
IT1271325B (it) 1997-05-27
ATE207929T1 (de) 2001-11-15
PT799239E (pt) 2002-02-28
US6147213A (en) 2000-11-14
DE69523622T2 (de) 2002-05-29
EP0799239A2 (en) 1997-10-08

Similar Documents

Publication Publication Date Title
ITMI942626A0 (it) Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
FI962246L (fi) Apoptoosia inhiboivat koostumukset, koostumusten puhdistusmenetelmät ja niiden käyttö
ITMI950529A0 (it) Composizioni farmaceutiche e procedimento per la loro preparazione
PT101722A (pt) Formulacoes de analogo de insuluna
FI971846A0 (fi) Kaasunilmaisin
DE69723398T2 (de) Polyalkylphenoxyaminoalkane und diese enthaltende freibstoffzusammensetzungen
FI956228L (fi) Sisäänhengitykseen tarkoitettuja koostumuksia
DE69534418D1 (de) Bioarraychip-reaktionsapparatur und ihre herstellung
FI955042A0 (fi) Syklosporiinia sisältävä jauhemainen koostumus
NO941980D0 (no) Gassturbin-luftseparasjonskombinasjonsanlegg
DE69425225D1 (de) Stabilisationssystem für thiol-ene und thiol-nene zusammensetzungen
FI954579L (fi) Uusia pednisolonijohdannaisia
DE69724629D1 (de) Zusammensetzungen und deren verwendungen
BR9508110A (pt) Derivado de triterpeno e composição médica
FI972434L (fi) Lamotrigiiniä sisältävä farmaseuttinen koostumus
GB9420055D0 (en) Anti-inflammatory compositions
FI946106L (fi) Steroidaalisia glykosideja
IL116190A (en) Eleutherobin, analogs thereof and pharmaceutical compositions containing them
BR9710383A (pt) Intensificador de absor-Æo
FI963746A0 (fi) Verikaasun ilmaisin
DE69708418D1 (de) Naphthylverbindungen und Zusammensetzungen
DE69726252D1 (de) Röntgenbildröhre und herstellungsverfahren für dieselbe
ITMI942166A0 (it) Composizioni farmaceutiche miorilassanti
DE69403129D1 (de) Röntgenstrahlen-Analysegerät
ZA956262B (en) Dihydrobenzofuran and related compounds useful as anti-inflammatory agents

Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19971223