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IT1243362B - Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti - Google Patents

Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti

Info

Publication number
IT1243362B
IT1243362B IT02106390A IT2106390A IT1243362B IT 1243362 B IT1243362 B IT 1243362B IT 02106390 A IT02106390 A IT 02106390A IT 2106390 A IT2106390 A IT 2106390A IT 1243362 B IT1243362 B IT 1243362B
Authority
IT
Italy
Prior art keywords
benzimidazole
thiazole
substituted
hiv activity
hiv
Prior art date
Application number
IT02106390A
Other languages
English (en)
Other versions
IT9021063A0 (it
IT9021063A1 (it
Inventor
Alba Chimirri
Silvana Grasso
Anna Maria Monforte
Pietro Monforte
Maria Zappala
Giovanni Romeo
Original Assignee
Pietro Monforte
Anna Maria Monforte
Maria Zappala
Giovanni Romeo
Silvana Grasso
Alba Chimirri
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pietro Monforte, Anna Maria Monforte, Maria Zappala, Giovanni Romeo, Silvana Grasso, Alba Chimirri filed Critical Pietro Monforte
Priority to IT02106390A priority Critical patent/IT1243362B/it
Publication of IT9021063A0 publication Critical patent/IT9021063A0/it
Priority to EP19910112224 priority patent/EP0471991A3/en
Priority to CA002047796A priority patent/CA2047796A1/en
Priority to JP3207158A priority patent/JPH04234395A/ja
Priority to US07/735,914 priority patent/US5217984A/en
Publication of IT9021063A1 publication Critical patent/IT9021063A1/it
Application granted granted Critical
Publication of IT1243362B publication Critical patent/IT1243362B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
IT02106390A 1990-07-25 1990-07-25 Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti IT1243362B (it)

Priority Applications (5)

Application Number Priority Date Filing Date Title
IT02106390A IT1243362B (it) 1990-07-25 1990-07-25 Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti
EP19910112224 EP0471991A3 (en) 1990-07-25 1991-07-22 1-phenyl substituted 1h,3h-thiazolo(3,4-a)benzimidazoles, process for their preparation, and pharmaceutical compositions containing them
CA002047796A CA2047796A1 (en) 1990-07-25 1991-07-24 1-phenyl substituted-1h, 3h-thiazole [3,4-a] benimidazoles, process for their preparation and pharmaceutical compositions containing them
JP3207158A JPH04234395A (ja) 1990-07-25 1991-07-25 新規１−フェニル置換１Ｈ，３Ｈ−チアゾール［３，４−ａ］ベンゾイミダゾール類、それらの調製工程及びそれらを含有する薬剤組成物類
US07/735,914 US5217984A (en) 1990-07-25 1991-07-25 1-phenyl substituted-1H, 3H-thiazole [3,4-a] benzimidazoles and pharmaceutical compositions containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02106390A IT1243362B (it) 1990-07-25 1990-07-25 Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti

Publications (3)

Publication Number Publication Date
IT9021063A0 IT9021063A0 (it) 1990-07-25
IT9021063A1 IT9021063A1 (it) 1992-01-25
IT1243362B true IT1243362B (it) 1994-06-10

Family

ID=11176175

Family Applications (1)

Application Number Title Priority Date Filing Date
IT02106390A IT1243362B (it) 1990-07-25 1990-07-25 Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti

Country Status (5)

Country Link
US (1) US5217984A (it)
EP (1) EP0471991A3 (it)
JP (1) JPH04234395A (it)
CA (1) CA2047796A1 (it)
IT (1) IT1243362B (it)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69814049T2 (de) * 1997-02-25 2004-02-19 The Government of the United States of America, as represented by the Secretary National Institute of Health, Office of Technology Transfer Substituierte benzimidazole als nicht-nucleoside reverse transcriptase inhibitore
US20060040111A1 (en) * 2004-08-20 2006-02-23 Dolechek Kert L Process chamber and system for thinning a semiconductor workpiece
DE102009038123A1 (de) 2009-08-17 2011-02-24 Aicuris Gmbh & Co. Kg Substituierte (Thiazolyl-carbonyl)imidazolidinone und ihre Verwendung

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3665007A (en) * 1970-05-04 1972-05-23 Squibb & Sons Inc Thiazolo (3,4-a) benzimidazoles and derivatives thereof
US3732240A (en) * 1971-01-21 1973-05-08 Squibb & Sons Inc Thiazolo(3,4-a)benzimidazole derivatives and process
FR2463774A1 (fr) * 1979-08-21 1981-02-27 Yamanouchi Pharma Co Ltd Derives du 2-phenylimidazo(2,1-b)benzothiazole
US4464384A (en) * 1981-12-23 1984-08-07 Yamanouchi Pharmaceutical Co., Ltd. 2-Phenylimidazo[2,1-b]benzothiazole compounds, salts thereof, process of producing them, and pharmaceutical compositions containing them
GB8701228D0 (en) * 1987-01-21 1987-02-25 Wyeth John & Brother Ltd Thiazolobenzimidazoles

Also Published As

Publication number Publication date
CA2047796A1 (en) 1992-01-26
US5217984A (en) 1993-06-08
EP0471991A3 (en) 1992-03-11
EP0471991A2 (en) 1992-02-26
IT9021063A0 (it) 1990-07-25
JPH04234395A (ja) 1992-08-24
IT9021063A1 (it) 1992-01-25

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970730