IT1197661B - 1-Phenalkyl-4-imidazo:pyridyl or pyrido:pyrazinyl piperazine derivs.
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1-Phenalkyl-4-imidazo:pyridyl or pyrido:pyrazinyl piperazine derivs.
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Publication number
IT1197661B
IT1197661BIT48453/83AIT4845383AIT1197661BIT 1197661 BIT1197661 BIT 1197661BIT 48453/83 AIT48453/83 AIT 48453/83AIT 4845383 AIT4845383 AIT 4845383AIT 1197661 BIT1197661 BIT 1197661B
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Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Nitrogen Condensed Heterocyclic Rings
(AREA)
Abstract
(A) Piperazine and homopiperazine derivs. of formula (I) and their acid addition salts are new. One of A and B is nitrogen, the other CH. Z is a ring (II) or (III); R1 and R2 are each H, 1-6C alkyl or 7-10C phenalkyl (opt. ring substd. once by halo or 1-4C alkoxy or alkyl. R3 is H or 1-4C alkyl. R'1 and R'2 are H or 1-4C alkyl or together are tri-, tetra- or penta-methylene. m is 1 or 2. R4 and R5 are each H, halo, 1-4C alkyl or alkoxy, 2-4C acyl or trifluoromethyl. X is CH2 and n is 0-3; X is Co and n is 1, 2 or 3, or X is oxygen and n is 2 or 3. Cpds. (I) and (VII) are neuroleptics (e.g. for treatment of schizophrenia); antihypertensives, and bradycardiac agents (e.g. for preventing or treating angina pectoris and tachycardia).
IT48453/83A1982-07-221983-06-081-Phenalkyl-4-imidazo:pyridyl or pyrido:pyrazinyl piperazine derivs.
IT1197661B
(en)
PYRIDO / 3,4-B / PYRROLO / 1,2-E // 1,4,5 / OXADIAZEPINER OCH DAERMED ANALOGER OF NAERBESLAEKTADE, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL.