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IT1161591B - Agenti antiflogistici/antipiretici/analgesici contenenti derivati di teobromina o teofillina come ingrediente attivo - Google Patents

Agenti antiflogistici/antipiretici/analgesici contenenti derivati di teobromina o teofillina come ingrediente attivo

Info

Publication number
IT1161591B
IT1161591B IT19857/83A IT1985783A IT1161591B IT 1161591 B IT1161591 B IT 1161591B IT 19857/83 A IT19857/83 A IT 19857/83A IT 1985783 A IT1985783 A IT 1985783A IT 1161591 B IT1161591 B IT 1161591B
Authority
IT
Italy
Prior art keywords
antiflogistic
antipyretic
active ingredient
agents containing
analgesic agents
Prior art date
Application number
IT19857/83A
Other languages
English (en)
Other versions
IT8319857A0 (it
Inventor
Kaneko Takeru
Ozaki Satoru
Takizawa Kimie
Sugimoto Hachiro
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3168582A external-priority patent/JPS58148819A/ja
Priority claimed from JP3168482A external-priority patent/JPS58148818A/ja
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of IT8319857A0 publication Critical patent/IT8319857A0/it
Application granted granted Critical
Publication of IT1161591B publication Critical patent/IT1161591B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/10Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 3 and 7, e.g. theobromine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT19857/83A 1982-03-02 1983-03-02 Agenti antiflogistici/antipiretici/analgesici contenenti derivati di teobromina o teofillina come ingrediente attivo IT1161591B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP3168582A JPS58148819A (ja) 1982-03-02 1982-03-02 テオブロミン誘導体を有効成分とする消炎・解熱・鎮痛剤
JP3168482A JPS58148818A (ja) 1982-03-02 1982-03-02 テオフイリン誘導体を有効成分とする消炎・解熱・鎮痛剤

Publications (2)

Publication Number Publication Date
IT8319857A0 IT8319857A0 (it) 1983-03-02
IT1161591B true IT1161591B (it) 1987-03-18

Family

ID=26370191

Family Applications (1)

Application Number Title Priority Date Filing Date
IT19857/83A IT1161591B (it) 1982-03-02 1983-03-02 Agenti antiflogistici/antipiretici/analgesici contenenti derivati di teobromina o teofillina come ingrediente attivo

Country Status (4)

Country Link
US (1) US4543254A (it)
EP (1) EP0087810B1 (it)
DE (2) DE3307395A1 (it)
IT (1) IT1161591B (it)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8303412A1 (es) * 1981-10-06 1983-02-01 Invest Tecnica Aplicada Procedimiento de obtencion de nuevas xantinas con actividad farmacologica
HU198052B (en) * 1986-02-14 1989-07-28 Sandoz Ag Process for producing purine derivatives substituted by side chain containing piperazinyl ring and pharmaceutical compositions comprising such compounds
CA1297035C (en) * 1987-12-29 1992-03-10 Warner-Lambert Canada Inc. Chewable, non-gritty calcium citrate tablet
US5164390A (en) * 1988-03-03 1992-11-17 Ortho Pharmaceutical Corporation 6-substituted purinyl piperazine derivatives
US5021574A (en) * 1988-03-03 1991-06-04 Ortho Pharmaceutical Corporation 6-substituted purinyl piperazine derivatives
US4876257A (en) * 1988-03-03 1989-10-24 Ortho Pharmaceutical Corporation 6-Substituted purinyl piperazine derivatives useful as cardiotonic and antiarrhythmic agents
FR2723091B1 (fr) * 1994-07-29 1996-11-08 Esteve Labor Dr Tetrahydropyridine-(6,4-hydroxypiperidine) alkylazoles
AU9002598A (en) 1997-09-16 1999-04-05 Takeda Chemical Industries Ltd. Nitrogenous fused-ring compounds, process for the preparation of the same, and drugs
US6979687B1 (en) * 2002-09-27 2005-12-27 Ing-Jun Chen Theophylline-based soluble guanylyl cyclase activators KMUP-1 analogues enhanced cyclic GMP and K+ channel activities on rabbit corpus cavernosum smooth muscle and intercavernous pressure activities
US20050209243A1 (en) * 2002-09-27 2005-09-22 Ing-Jun Chen Theophylline-based soluble guanylyl cyclase activators KMUP-1 analogues enhanced cyclic GMP and K+ channel activities on rabbit corpus cavernosum smooth muscle and intercavernous pressure activities
EA200600071A1 (ru) * 2003-06-20 2006-08-25 Арена Фармасьютикалз, Инк. Производные n-фенилпиперазина и способы профилактики или лечения заболеваний, связанных с 5ht-рецептором
EP1844792A4 (en) * 2004-12-14 2008-05-21 Shionogi & Co THERAPEUTIC AGENT AGAINST OBSTIPATION
RU2333212C3 (ru) * 2007-03-29 2019-08-26 Общество С Ограниченной Ответственностью "Фармвинг" ПРОИЗВОДНЫЕ 1-И 7-[ω-(БЕНЗГИДРИЛ-4-ПИПЕРАЗИНИЛ-1)АЛКИЛ]-3-АЛКИЛКСАНТИНОВ, ОБЛАДАЮЩИЕ ПРОТИВОГИСТАМИННОЙ И АНТИАЛЛЕРГИЧЕСКОЙ АКТИВНОСТЬЮ
RU2373207C1 (ru) * 2008-03-17 2009-11-20 Общество С Ограниченной Ответственностью "Фармвинг" Способ получения 3-метил-7-[4-(бензгидрил-4-пиперазинил-1) бутил]ксантина и его солей с органическими или неорганическими кислотами
CN101861317B (zh) * 2007-03-29 2013-07-31 A.B.英特尔法玛有限公司 抗组胺类抗过敏剂及其制备方法
WO2009002933A1 (en) * 2007-06-22 2008-12-31 Hydra Biosciences, Inc. Methods and compositions for treating disorders
AU2015202546B8 (en) * 2007-06-22 2017-03-09 Eli Lilly And Company Methods and Compositions for Treating Disorders
WO2009140517A1 (en) 2008-05-14 2009-11-19 Hydra Biosciences, Inc. Compounds and compositions for treating chemical warfare agent-induced injuries
TWI368511B (en) * 2009-04-30 2012-07-21 Univ Kaohsiung Medical Synthesis and pharmacokinetic activities of pulmodil and pulmodil-1, two chlorophenylpiperazine salt derivatives

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1545717A1 (de) * 1965-12-06 1969-07-24 Chugai Pharmaceutical Co Ltd Verfahren zur Herstellung von Theophyllinderivaten
DD143179B1 (de) * 1979-05-16 1983-03-30 Georg Diederich Verfahren zur elektronischen thrombozytenzaehlung
JPS5618983A (en) * 1979-07-25 1981-02-23 Eisai Co Ltd Theophylline derivative and its preapration
CH648559A5 (de) * 1981-07-20 1985-03-29 Siegfried Ag Theophyllinderivate und verfahren zu deren herstellung.
US4374837A (en) * 1981-07-31 1983-02-22 Laroche Navarron, S.A. Piperazine derivatives of theobromine

Also Published As

Publication number Publication date
DE3307395A1 (de) 1983-09-08
EP0087810A1 (en) 1983-09-07
EP0087810B1 (en) 1986-06-25
US4543254A (en) 1985-09-24
DE3364234D1 (en) 1986-07-31
IT8319857A0 (it) 1983-03-02

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