IT1160301B - 1-amino-2-hydroxy-3-phenoxy-3-phenyl-propane derivs. - useful as antidepressants - Google Patents
1-amino-2-hydroxy-3-phenoxy-3-phenyl-propane derivs. - useful as antidepressantsInfo
- Publication number
- IT1160301B IT1160301B IT3053378A IT3053378A IT1160301B IT 1160301 B IT1160301 B IT 1160301B IT 3053378 A IT3053378 A IT 3053378A IT 3053378 A IT3053378 A IT 3053378A IT 1160301 B IT1160301 B IT 1160301B
- Authority
- IT
- Italy
- Prior art keywords
- substd
- opt
- alkyl
- derivs
- aryl
- Prior art date
Links
- SCKQUWRORFAPMX-UHFFFAOYSA-N 3-amino-1-phenoxy-1-phenylpropan-2-ol Chemical compound C=1C=CC=CC=1C(C(O)CN)OC1=CC=CC=C1 SCKQUWRORFAPMX-UHFFFAOYSA-N 0.000 title 1
- 239000000935 antidepressant agent Substances 0.000 title 1
- 229940005513 antidepressants Drugs 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- 125000003118 aryl group Chemical group 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- WUGQZFFCHPXWKQ-UHFFFAOYSA-N Propanolamine Chemical compound NCCCO WUGQZFFCHPXWKQ-UHFFFAOYSA-N 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000000816 ethylene group Chemical group [H]C([H])([*:1])C([H])([H])[*:2] 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002950 monocyclic group Chemical group 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 125000006237 oxymethylenoxy group Chemical group [H]C([H])([*:1])[*:2] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Propanolamine derivs. of formula (I) and their pharmaceutically acceptable salts are new: (n and n1 = 1-3; R and R1 are each same or different H, halo, 1-6C haloalkyl, OH, 1-6C alkoxy or opt. substd. alkyl, aryl(1-6C)-alkyl or aryl(1-6C)alkoxy (both opt. substd.), NO2, NR5R6, or two adjacent gps. are together OCH2O; R2 = H, opt. substd. 1-12C alkyl or aryl(1-6C)alkyl; R3 and R4 = H, 1-6C opt. substd. alkyl, 2-4C alkenyl or alkynyl, aryl(1-4C)alkyl (opt. substd.), 3-7C cycloalkyl (opt. substd.) or R3 + R4 complete a monocyclic 5 or 6 member heterocycle which may be unsatd. or satd. opt. substd. and or contain further O, S or N atoms; R2 and R4 may also together be CH2CH2; R5 and R6 = H or 1-6C alkyl).
Priority Applications (30)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT3053378A IT1160301B (en) | 1978-12-05 | 1978-12-05 | 1-amino-2-hydroxy-3-phenoxy-3-phenyl-propane derivs. - useful as antidepressants |
| IL56369A IL56369A (en) | 1978-01-20 | 1979-01-04 | Alpha-phenoxybenzyl propanolamine derivatives,their preparation and pharmaceutical compositions comprising them |
| US06/001,604 US4229449A (en) | 1978-01-20 | 1979-01-08 | Substituted morpholine derivatives and compositions |
| GB7901130A GB2014981B (en) | 1978-01-20 | 1979-01-11 | Substituted propanolamine and morpholine derivatives |
| CY1172A CY1172A (en) | 1978-01-20 | 1979-01-11 | Substituted propanolamine and morpholine derivatives |
| DE1998175005 DE19875005I2 (en) | 1978-01-20 | 1979-01-12 | Substituted morpholine derivatives and their use |
| DE2901032A DE2901032C2 (en) | 1978-01-20 | 1979-01-12 | Substituted morpholine derivatives and their use |
| AU43327/79A AU525954B2 (en) | 1978-01-20 | 1979-01-12 | Substituted propanolamine and morpholine derivatives |
| NZ189418A NZ189418A (en) | 1978-01-20 | 1979-01-17 | Propanolamine and morpholine derivatives pharmaceutical compositions |
| SI7910096A SI7910096A8 (en) | 1978-01-20 | 1979-01-17 | Process for preparing novel morpholine compounds |
| YU96/79A YU42094B (en) | 1978-01-20 | 1979-01-17 | Process for obtaining new morpnoline compounds |
| NL7900412A NL190327C (en) | 1978-01-20 | 1979-01-18 | SUBSTITUTED 2- (PHENOXYMETHYL) MORPHOLINE DERIVATIVE WITH ANTI-DEPRESSIVE ACTION, METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL PREPARATION CONTAINING SUCH A MORPHOLINE DERIVATIVE. |
| DK022679A DK156565C (en) | 1978-01-20 | 1979-01-18 | ANALOGY PROCEDURE FOR THE PREPARATION OF SUBSTITUTED MORPHOLINE DERIVATIVES |
| AT0040679A AT371813B (en) | 1978-01-20 | 1979-01-19 | METHOD FOR PRODUCING NEW SUBSTITUTED PROPANOLAMINE AND MORPHOLINE DERIVATIVES AND THEIR ISOMERS AND SALTS |
| SE7900498A SE446727B (en) | 1978-01-20 | 1979-01-19 | SUBSTITUTED MORPHOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION THEREOF |
| CA319,931A CA1128942A (en) | 1978-01-20 | 1979-01-19 | Substituted propanolamine and morpholine derivatives and process for their preparation |
| FI790177A FI71135C (en) | 1978-01-20 | 1979-01-19 | FRUIT PROCESSING OF PHARMACOLOGICAL ACTIVE SUBSTITUTES MORPHOLINDERIVAT |
| HUEA000189 HU178214B (en) | 1978-12-05 | 1979-01-19 | Process for producing substituted propanolamine- and morpholine derivatives |
| NO790205A NO146953C (en) | 1978-01-20 | 1979-01-19 | ANALOGY PROCEDURE FOR THE PREPARATION OF SUBSTITUTED PROPANOLAMINE AND MORPHOLINE DERIVATIVES |
| CH582/79A CH650245A5 (en) | 1978-01-20 | 1979-01-19 | SUBSTITUTED PROPANOLAMINE AND MORPHOLINE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF. |
| FR7901413A FR2442839A1 (en) | 1978-01-20 | 1979-01-19 | SUBSTITUTED MORPHOLINE DERIVATIVES USEFUL AS MEDICAMENTS AND PROCESS FOR THEIR PREPARATION |
| JP449479A JPS54148739A (en) | 1978-01-20 | 1979-01-20 | Substituted propanolamine and morpholine derivative |
| IE107/79A IE47727B1 (en) | 1978-01-20 | 1979-01-30 | Substituted propanolamine and morpholine derivatives |
| FR7922678A FR2430412B1 (en) | 1978-01-20 | 1979-09-11 | SUBSTITUTED PROPANOLAMINE DERIVATIVES USEFUL AS MEDICAMENTS AND PROCESS FOR THEIR PREPARATION |
| US06/161,509 US4271160A (en) | 1978-01-20 | 1980-06-20 | Substituted morpholine derivatives and pharmaceutical compositions |
| KE3243A KE3243A (en) | 1978-01-20 | 1982-10-25 | Substituted propanolamine and morpholine derivatives |
| HK57/83A HK5783A (en) | 1978-01-20 | 1983-02-08 | Substituted propanolamine and morpholine derivatives |
| MY8418A MY8400018A (en) | 1978-01-20 | 1984-12-31 | Substituted propanolamine and morpholine derivatives |
| CS914133A CS413391A3 (en) | 1978-01-20 | 1991-12-30 | Substituted propanolamine and morpholine derivatives |
| BG098513A BG61056B2 (en) | 1978-01-20 | 1994-02-22 | Substituted propanolamine and morpholine derivatives |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT3053378A IT1160301B (en) | 1978-12-05 | 1978-12-05 | 1-amino-2-hydroxy-3-phenoxy-3-phenyl-propane derivs. - useful as antidepressants |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT7830533A0 IT7830533A0 (en) | 1978-12-05 |
| IT1160301B true IT1160301B (en) | 1987-03-11 |
Family
ID=11229916
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT3053378A IT1160301B (en) | 1978-01-20 | 1978-12-05 | 1-amino-2-hydroxy-3-phenoxy-3-phenyl-propane derivs. - useful as antidepressants |
Country Status (1)
| Country | Link |
|---|---|
| IT (1) | IT1160301B (en) |
-
1978
- 1978-12-05 IT IT3053378A patent/IT1160301B/en active
Also Published As
| Publication number | Publication date |
|---|---|
| IT7830533A0 (en) | 1978-12-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19961218 |