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IS6844A - Þíasólýl-, oxasólýl-, pýrrólýl- og ímídasólýlsýruamíðafleiður, nytsamlegar sem hindrar PDE4 samsætuensíma - Google Patents

Þíasólýl-, oxasólýl-, pýrrólýl- og ímídasólýlsýruamíðafleiður, nytsamlegar sem hindrar PDE4 samsætuensíma

Info

Publication number
IS6844A
IS6844A IS6844A IS6844A IS6844A IS 6844 A IS6844 A IS 6844A IS 6844 A IS6844 A IS 6844A IS 6844 A IS6844 A IS 6844A IS 6844 A IS6844 A IS 6844A
Authority
IS
Iceland
Prior art keywords
isotopic
oxazolyl
pyrrolyl
thiazolyl
enzymes
Prior art date
Application number
IS6844A
Other languages
English (en)
Inventor
Marfat Anthony
William Mckechney Michael
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of IS6844A publication Critical patent/IS6844A/is

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

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  • Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Molecular Biology (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Transplantation (AREA)
  • Ophthalmology & Optometry (AREA)
  • Biotechnology (AREA)
  • AIDS & HIV (AREA)
IS6844A 2001-01-31 2003-06-16 Þíasólýl-, oxasólýl-, pýrrólýl- og ímídasólýlsýruamíðafleiður, nytsamlegar sem hindrar PDE4 samsætuensíma IS6844A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26548601P 2001-01-31 2001-01-31
PCT/IB2001/002728 WO2002060898A1 (en) 2001-01-31 2001-12-24 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Publications (1)

Publication Number Publication Date
IS6844A true IS6844A (is) 2003-06-16

Family

ID=23010641

Family Applications (1)

Application Number Title Priority Date Filing Date
IS6844A IS6844A (is) 2001-01-31 2003-06-16 Þíasólýl-, oxasólýl-, pýrrólýl- og ímídasólýlsýruamíðafleiður, nytsamlegar sem hindrar PDE4 samsætuensíma

Country Status (24)

Country Link
US (3) US6559168B2 (is)
EP (1) EP1355907A1 (is)
JP (1) JP2004518691A (is)
KR (1) KR20030072614A (is)
CN (1) CN1489588A (is)
BG (1) BG108039A (is)
BR (1) BR0116850A (is)
CA (1) CA2436551A1 (is)
CR (1) CR7038A (is)
CZ (1) CZ20031903A3 (is)
EA (1) EA200300622A1 (is)
EC (1) ECSP034683A (is)
EE (1) EE200300362A (is)
HU (1) HUP0401305A2 (is)
IL (1) IL156412A0 (is)
IS (1) IS6844A (is)
MA (1) MA26985A1 (is)
MX (1) MXPA03006886A (is)
NO (1) NO20033398L (is)
OA (1) OA12542A (is)
PL (1) PL365443A1 (is)
TN (1) TNSN03050A1 (is)
WO (1) WO2002060898A1 (is)
ZA (1) ZA200305769B (is)

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CN1537018A (zh) 2001-05-23 2004-10-13 田边制药株式会社 一种用于软骨疾病再生治疗的组合物
MXPA03010679A (es) * 2001-05-23 2004-03-02 Tanabe Seiyaku Co Una composicion para acelerar la cicatrizacion de fractura osea.
US20040235794A1 (en) * 2001-09-04 2004-11-25 Shinji Nakade Remedies for respiratory diseases comprising sphingosine-1-phosphate receptor controller
US20030171411A1 (en) * 2001-12-21 2003-09-11 Kodra Janos Tibor Amide derivatives as therapeutic agents
US6696473B2 (en) * 2001-12-21 2004-02-24 X-Ceptor Therapeutics, Inc. Heterocyclic modulators of nuclear receptors
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EP1470826B1 (en) 2002-02-01 2009-01-28 AnGes MG, Inc. Decoy-containing pharmaceutical compositions for the treatment of aneurysms
US20050158371A1 (en) * 2002-02-12 2005-07-21 Sumitomo Pharmaceuticals Co., Ltd. Novel external agent
WO2004002481A1 (en) * 2002-06-27 2004-01-08 Novo Nordisk A/S Aryl carbonyl derivatives as therapeutic agents
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FI114917B (fi) * 2002-08-29 2005-01-31 Hormos Nutraceutical Oy Ltd Lignaanikomplekseja
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US7148248B2 (en) * 2002-11-29 2006-12-12 Masako Nozaki Method of treating or inhibiting the development of brain inflammation and sepsis
EP1424101A3 (en) * 2002-11-29 2004-08-18 NOZAKI, Masako Use of a leukotriene C4 and D4 receptor antagonist for the preparation of a medicament for treating or preventing brain inflammation and sepsis
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US7153870B2 (en) 2003-07-25 2006-12-26 Pfizer Inc. Nicotinamide derivatives useful as PDE4 inhibitors
GB0317498D0 (en) * 2003-07-25 2003-08-27 Pfizer Ltd Compounds
US20050020587A1 (en) * 2003-07-25 2005-01-27 Pfizer Inc Nicotinamide derivatives useful as PDE4 inhibitors
US7132435B2 (en) 2003-07-25 2006-11-07 Pfizer Inc. Compounds
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