IL71796A0 - Diphenylazomethines containing an esterified chain,their preparation and pharmaceutical compositions containing them - Google Patents
Diphenylazomethines containing an esterified chain,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL71796A0 IL71796A0 IL71796A IL7179684A IL71796A0 IL 71796 A0 IL71796 A0 IL 71796A0 IL 71796 A IL71796 A IL 71796A IL 7179684 A IL7179684 A IL 7179684A IL 71796 A0 IL71796 A0 IL 71796A0
- Authority
- IL
- Israel
- Prior art keywords
- alkyl radical
- radical
- alkoxy
- chain
- halogen atom
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000005843 halogen group Chemical group 0.000 abstract 5
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 4
- 239000002253 acid Substances 0.000 abstract 3
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical compound Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 229910052783 alkali metal Inorganic materials 0.000 abstract 1
- -1 alkali metal salt Chemical class 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- RWCCWEUUXYIKHB-UHFFFAOYSA-N benzophenone Chemical compound C=1C=CC=CC=1C(=O)C1=CC=CC=C1 RWCCWEUUXYIKHB-UHFFFAOYSA-N 0.000 abstract 1
- 239000012965 benzophenone Substances 0.000 abstract 1
- PFKFTWBEEFSNDU-UHFFFAOYSA-N carbonyldiimidazole Chemical compound C1=CN=CN1C(=O)N1C=CN=C1 PFKFTWBEEFSNDU-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000004170 methylsulfonyl group Chemical group [H]C([H])([H])S(*)(=O)=O 0.000 abstract 1
- 125000002088 tosyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1C([H])([H])[H])S(*)(=O)=O 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/10—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/12—Radicals substituted by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Saccharide Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
1. Claims (for the contracting states : BE, CH, DE, FR, GB, IT, LI, LU, NL, SE) Diphenylazomethines containing an esterified chain and corresponding to the formula (I) see diagramm : EP0125975,P15,F1 in which X1 , X2 and X3 independently of one another each represent a hydrogen or halogen atom or a (C1-6 )alkyl radical, R represents a straight-chain or branched (C1-6 )alkyl radical, n represents an integer from 1 to 10 and R' represents a straight-chain or branched (C1-6 )alkyl radical, a (C3-6 )cycloalkyl(C1-4 )alkyl radical, a (C3-7 )cycloalkyl radical, a (C2-6 )alkenyl radical, a (C3-6 )alkynyl radical, a (C1-4 )alkoxy(C1-4 )alkyl radical, a hydroxy-(C1-4 )alkyl radical, a (C1-4 )alkoxy-[(C1-4 )alkoxy]m -(C1-4 )alkyl radical, in which m is an integer from 1 to 3, a (C1-4 )alkoxycarbonyl(C1-4 )alkyl radical, a tetrahydrofurylmethyl radical, a phenyl-(C1-4 )alkyl radical which can carry a halogen atom, or a (C1-4 )alkoxy radical. 1. Claim (for the contracting state AT) Process for the preparation of diphenylazomethines containing an esterified chain and corresponding to the formula (1) see diagramm : EP0125975,P17,F1 in which X1 , X2 and X3 independently of one another each represent a hydrogen or halogen atom or a (C1-6 )alkyl radical, R represents a straight-chain or branched (C1-6 )alkyl radical, n represents an integer from 1 to 10 and R' represents a straight-chain or branched (C1-6 )alkyl radical, a (C3-6 )cycloalkyl (C1-4 )alkyl radical, a (C3-7 )cycloalkyl radical, a (C2-6 )alkenyl radical, a (C3-6 )alkynyl radical, a (C1-4 )alkoxy-(C1-4 )alkyl radical, a hydroxy-(C1-4 )alkyl radical, a (C1-4 )alkoxy[(C1-4 )alkoxy]m -(C1-4 )alkyl radical, in which m is an integer from 1 to 3, a (C1-4 )alkoxy-carbonyl-(C1-4 )alkyl radical, a tetrahydrofurylmethyl radical, a phenyl-(C1-4 )alkyl radical which can carry a halogen atom, or a (C1-4 )alkoxy radical, process characterised in that either a benzophenone (II) see diagramm : EP0125975,P17,F2 is reacted with the hydrochloride of an ester of an omega-amino-alkanoic acid (III) H2 N-(CH2 )n -COOR', HCl or an acid (IV) see diagramm : EP0125975,P17,F3 is reacted with an alcohol R'OH (V) in the presence of carbonyldiimidazole, or an alkali metal salt of an acid (VI) see diagramm : EP0125975,P18,F1 is reacted with a compound R'Y (VII), in which Y represents a halogen atom or a labil group, such as mesyl or tosyl, the radicals X1 , X2 , X3 , n, R and R' having the meanings given above.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8307863A FR2545822B1 (en) | 1983-05-11 | 1983-05-11 | DIPHENYLAZOMETHINES CARRYING AN ESTERIFIED CHAIN, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL71796A0 true IL71796A0 (en) | 1984-09-30 |
Family
ID=9288787
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL71796A IL71796A0 (en) | 1983-05-11 | 1984-05-10 | Diphenylazomethines containing an esterified chain,their preparation and pharmaceutical compositions containing them |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0125975B1 (en) |
| JP (1) | JPS59212458A (en) |
| AT (1) | ATE18760T1 (en) |
| AU (1) | AU2788584A (en) |
| DE (1) | DE3460059D1 (en) |
| DK (1) | DK232084A (en) |
| ES (1) | ES8502678A1 (en) |
| FI (1) | FI841882A7 (en) |
| FR (1) | FR2545822B1 (en) |
| GR (1) | GR82093B (en) |
| HU (1) | HU191652B (en) |
| IL (1) | IL71796A0 (en) |
| NO (1) | NO841878L (en) |
| NZ (1) | NZ208118A (en) |
| PT (1) | PT78575A (en) |
| ZA (1) | ZA843545B (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007127440A2 (en) * | 2006-04-27 | 2007-11-08 | Intezyne Technologies, Inc. | Heterofunctional poly(ethylene glycol) containing acid-labile amino protecting groups and uses thereof |
| MX2023006325A (en) * | 2021-05-26 | 2023-06-12 | Procter & Gamble | Pro-benefit agent compounds with carbon/nitrogen bonds. |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2319338A1 (en) * | 1975-08-01 | 1977-02-25 | Synthelabo | NEW A-PHENYL BENZYLIDENIC DERIVATIVES OF AMINO ACIDS, THEIR PREPARATION AND THE MEDICINAL PRODUCTS CONTAINING THEM |
-
1983
- 1983-05-11 FR FR8307863A patent/FR2545822B1/en not_active Expired
-
1984
- 1984-05-02 AT AT84400889T patent/ATE18760T1/en not_active IP Right Cessation
- 1984-05-02 DE DE8484400889T patent/DE3460059D1/en not_active Expired
- 1984-05-02 EP EP84400889A patent/EP0125975B1/en not_active Expired
- 1984-05-10 DK DK232084A patent/DK232084A/en not_active Application Discontinuation
- 1984-05-10 ES ES532363A patent/ES8502678A1/en not_active Expired
- 1984-05-10 AU AU27885/84A patent/AU2788584A/en not_active Abandoned
- 1984-05-10 JP JP59094420A patent/JPS59212458A/en active Pending
- 1984-05-10 HU HU841829A patent/HU191652B/en unknown
- 1984-05-10 FI FI841882A patent/FI841882A7/en not_active Application Discontinuation
- 1984-05-10 GR GR74674A patent/GR82093B/el unknown
- 1984-05-10 ZA ZA843545A patent/ZA843545B/en unknown
- 1984-05-10 PT PT78575A patent/PT78575A/en unknown
- 1984-05-10 IL IL71796A patent/IL71796A0/en unknown
- 1984-05-10 NZ NZ208118A patent/NZ208118A/en unknown
- 1984-05-10 NO NO841878A patent/NO841878L/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI841882A7 (en) | 1984-11-12 |
| ES532363A0 (en) | 1985-01-16 |
| ZA843545B (en) | 1984-12-24 |
| HU191652B (en) | 1987-03-30 |
| FI841882A0 (en) | 1984-05-10 |
| NO841878L (en) | 1984-11-12 |
| PT78575A (en) | 1984-06-01 |
| ATE18760T1 (en) | 1986-04-15 |
| EP0125975B1 (en) | 1986-03-26 |
| ES8502678A1 (en) | 1985-01-16 |
| AU2788584A (en) | 1984-11-15 |
| DK232084A (en) | 1984-11-12 |
| JPS59212458A (en) | 1984-12-01 |
| FR2545822B1 (en) | 1985-07-05 |
| NZ208118A (en) | 1987-01-23 |
| EP0125975A1 (en) | 1984-11-21 |
| HUT34436A (en) | 1985-03-28 |
| DK232084D0 (en) | 1984-05-10 |
| DE3460059D1 (en) | 1986-04-30 |
| FR2545822A1 (en) | 1984-11-16 |
| GR82093B (en) | 1984-12-13 |
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