[go: up one dir, main page]

IL160938A0 - Coniosulphides and their derivatives, processes for preparing them, and their use as pharmaceuticals - Google Patents

Coniosulphides and their derivatives, processes for preparing them, and their use as pharmaceuticals

Info

Publication number
IL160938A0
IL160938A0 IL16093802A IL16093802A IL160938A0 IL 160938 A0 IL160938 A0 IL 160938A0 IL 16093802 A IL16093802 A IL 16093802A IL 16093802 A IL16093802 A IL 16093802A IL 160938 A0 IL160938 A0 IL 160938A0
Authority
IL
Israel
Prior art keywords
coniosulphides
pharmaceuticals
derivatives
preparing
processes
Prior art date
Application number
IL16093802A
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of IL160938A0 publication Critical patent/IL160938A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/44Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06017Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0804Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0806Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P11/00Preparation of sulfur-containing organic compounds
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P13/00Preparation of nitrogen-containing organic compounds
    • C12P13/001Amines; Imines
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P13/00Preparation of nitrogen-containing organic compounds
    • C12P13/02Amides, e.g. chloramphenicol or polyamides; Imides or polyimides; Urethanes, i.e. compounds comprising N-C=O structural element or polyurethanes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biomedical Technology (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • General Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
IL16093802A 2001-09-22 2002-09-06 Coniosulphides and their derivatives, processes for preparing them, and their use as pharmaceuticals IL160938A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10146737A DE10146737A1 (en) 2001-09-22 2001-09-22 Coniosulfides and their derivatives, process for their preparation and use as medicines
PCT/EP2002/009977 WO2003029495A2 (en) 2001-09-22 2002-09-06 Coniosulphides and their derivatives, method for their production and use as medicaments

Publications (1)

Publication Number Publication Date
IL160938A0 true IL160938A0 (en) 2004-08-31

Family

ID=7699903

Family Applications (2)

Application Number Title Priority Date Filing Date
IL16093802A IL160938A0 (en) 2001-09-22 2002-09-06 Coniosulphides and their derivatives, processes for preparing them, and their use as pharmaceuticals
IL160938A IL160938A (en) 2001-09-22 2004-03-18 Coniosulphides and their derivatives, processes for preparing them and their use as pharmaceuticals

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL160938A IL160938A (en) 2001-09-22 2004-03-18 Coniosulphides and their derivatives, processes for preparing them and their use as pharmaceuticals

Country Status (12)

Country Link
EP (2) EP1474440B1 (en)
JP (2) JP4287744B2 (en)
AR (1) AR036554A1 (en)
AT (2) ATE407942T1 (en)
AU (1) AU2002339519B2 (en)
CA (1) CA2461033C (en)
DE (3) DE10146737A1 (en)
ES (2) ES2314107T3 (en)
IL (2) IL160938A0 (en)
MX (1) MXPA04001951A (en)
PE (1) PE20030466A1 (en)
WO (1) WO2003029495A2 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2549158T3 (en) * 2008-11-11 2015-10-23 Signum Biosciences, Inc. Isoprenyl compounds and methods thereof
JP7318948B2 (en) * 2018-04-13 2023-08-01 国立大学法人京都大学 Prophylactic, therapeutic or diagnostic agent for Alzheimer's disease using microbial compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9210393D0 (en) * 1992-05-15 1992-07-01 Merck Sharp & Dohme Therapeutic agents
FR2740454B1 (en) * 1995-10-26 1997-11-21 Rhone Poulenc Rorer Sa PEPTIDES CAPABLE OF INHIBITING APP ENDOCYTOSIS AND CORRESPONDING NUCLEOTIDE SEQUENCES
JP2001503988A (en) * 1996-11-08 2001-03-27 ローヌ―プーラン・ロレ・エス・アー Peptides capable of inhibiting APP endocytosis and corresponding nucleotide sequences
NZ520697A (en) * 2000-02-10 2005-11-25 Aventis Pharma Sa Partners of PTB1 domain of FE65, preparation and uses
DE10060810A1 (en) 2000-12-07 2002-06-20 Aventis Pharma Gmbh Coniosetin and derivatives thereof, processes for making and using the same

Also Published As

Publication number Publication date
ATE430131T1 (en) 2009-05-15
MXPA04001951A (en) 2004-06-07
EP1474440B1 (en) 2008-09-10
DE50212774D1 (en) 2008-10-23
JP4287744B2 (en) 2009-07-01
WO2003029495A3 (en) 2004-02-26
CA2461033A1 (en) 2003-04-10
EP1474440A2 (en) 2004-11-10
EP1903033B1 (en) 2009-04-29
ATE407942T1 (en) 2008-09-15
WO2003029495A2 (en) 2003-04-10
EP1903033A1 (en) 2008-03-26
AU2002339519B2 (en) 2007-02-08
AR036554A1 (en) 2004-09-15
DE50213512D1 (en) 2009-06-10
ES2326563T3 (en) 2009-10-14
JP2005504131A (en) 2005-02-10
JP2009149662A (en) 2009-07-09
CA2461033C (en) 2011-12-06
PE20030466A1 (en) 2003-07-08
IL160938A (en) 2010-11-30
ES2314107T3 (en) 2009-03-16
DE10146737A1 (en) 2003-04-10

Similar Documents

Publication Publication Date Title
TWI347201B (en) Pharmaceutical products,uses thereof and methods for preparing the same
IL160440A (en) Dihydropteridinones, method for producing the same and the use thereof as medicaments
AU2002365516A1 (en) Benzamide derivatives, processes for their preparation, and their pharmaceutical use
HUP0401648A3 (en) 6-hydroxy isoflavon compounds, their derivatives and medicaments involving the same
HUP0402264A3 (en) Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines process for preparing them, pharmaceutical compositions containing them and use thereof
IL157471A (en) Xanthine derivatives, production thereof and their use as medicaments
HUP0303729A3 (en) Novel heteroaryl derivatives and the use thereof as pharmaceuticals and process for their preparation
TWI319764B (en) Mercaptoacetylamide derivatives, a process for their preparation and their use
MXPA03006538A (en) Novel urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use.
MXPA03008630A (en) Arylisoxazoline derivatives, method for production and use thereof as pesticides.
PL350190A1 (en) Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
IL162316A0 (en) Substituted 4-phenyltetrahydroisoquinolines, method for the production thereof, the use thereof as medicaments, in addition t
IL159570A0 (en) Phenylacetamido-thiazole derivatives, process for their preparation and their use as antitumor agents
MXPA03006478A (en) Chromane derivatives, process for their preparation and their use as antitumor agents.
IL164248A0 (en) Acyl-3-carboxyphenylurea derivatives, processes for preparing them and their use
MXPA03006249A (en) 2-arylimino-2,3-dihydrothiazole derivatives, methods for preparing them and therapeutic use thereof.
AU2002233407A1 (en) 2-arylimino-2,3-dihydrothiazole derivatives, methods for preparing them and therapeutic use thereof
IL164815A0 (en) Halosulfonylbenzoyl halides, processes for their preparation and their use for preparing substitutedphenylsulfonylureas
IL160606A0 (en) C2-substituted indan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals
IL160938A (en) Coniosulphides and their derivatives, processes for preparing them and their use as pharmaceuticals
IL160608A0 (en) C2-substituted indan-1-ones and their derivatives, processes for their preparation and their use as pharmaceuticals
IL159561A0 (en) Eurotinones and derivatives thereof, processes for preparing them, and their use
IL157793A0 (en) Caloporoside derivatives, methods for the production thereof and their use
AU2003264894A8 (en) Novel method for preparing alpha-glycosylceramides, novel alpha-glycosylceramide derivatives and their uses
AU2002333449A1 (en) C2-substituted indane-1-ols and their derivatives, method for their production and their use as medicaments