IL160084A0 - Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity - Google Patents

Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity

Info

Publication number: IL160084A0
Authority: IL; Israel
Prior art keywords: thieno; pyrimidines; combined; agonistic activity; fsh agonistic
Prior art date: 2001-09-04

Application number

IL16008402A

Other languages

English (en)

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-09-04

Filing date

2002-08-29

Publication date

2004-06-20

2002-08-29 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2004-06-20 Publication of IL160084A0 publication Critical patent/IL160084A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
- A61P5/08—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

IL16008402A 2001-09-04 2002-08-29 Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity IL160084A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP01203327		2001-09-04
PCT/EP2002/009647 WO2003020726A1 (en)	2001-09-04	2002-08-29	Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity

Publications (1)

Publication Number	Publication Date
IL160084A0 true IL160084A0 (en)	2004-06-20

Family

ID=8180876

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL16008402A IL160084A0 (en)	2001-09-04	2002-08-29	Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity

Country Status (28)

Country	Link
US (1)	US7317006B2 (xx)
EP (1)	EP1427733B1 (xx)
JP (1)	JP4262092B2 (xx)
KR (1)	KR100900018B1 (xx)
CN (1)	CN1246324C (xx)
AR (1)	AR036407A1 (xx)
AT (1)	ATE345345T1 (xx)
AU (1)	AU2002337035B2 (xx)
BR (1)	BR0211938A (xx)
CA (1)	CA2456901C (xx)
CY (1)	CY1106012T1 (xx)
DE (1)	DE60216128T2 (xx)
DK (1)	DK1427733T3 (xx)
ES (1)	ES2275005T3 (xx)
HR (1)	HRP20040202A2 (xx)
HU (1)	HUP0401444A3 (xx)
IL (1)	IL160084A0 (xx)
IS (1)	IS2424B (xx)
MX (1)	MXPA04002045A (xx)
NO (1)	NO20040927L (xx)
NZ (1)	NZ531340A (xx)
PE (1)	PE20030439A1 (xx)
PL (1)	PL368502A1 (xx)
PT (1)	PT1427733E (xx)
RU (1)	RU2298011C2 (xx)
TW (1)	TWI228508B (xx)
WO (1)	WO2003020726A1 (xx)
ZA (1)	ZA200401455B (xx)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6890923B2 (en) *	2002-12-16	2005-05-10	Astrazeneca Ab	Compounds
GB0315950D0 (en) *	2003-06-11	2003-08-13	Xention Discovery Ltd	Compounds
GB0525164D0 (en) *	2005-12-09	2006-01-18	Xention Discovery Ltd	Compounds
CN100430403C (zh) *	2006-10-13	2008-11-05	中国科学院上海有机化学研究所	3-芳基-5,6-取代噻吩并嘧啶-4-羰基-2-巯基乙腈、合成方法和用途
US20090118276A1 (en) *	2007-11-02	2009-05-07	Wyeth	Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors
TWI389913B (zh) *	2008-09-08	2013-03-21	Lg Life Sciences Ltd	并合雜環化合物
EP2358684B8 (en)	2008-10-20	2014-10-22	The Government of the United States of America as represented by the Secretary of the Department of Health and Human Services	Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
GB0905525D0 (en)	2009-03-31	2009-05-13	Univ Leiden	Compounds and uses
EP2525658B1 (de)	2010-01-22	2017-03-01	Bayer Intellectual Property GmbH	Akarizide und/oder insektizide wirkstoffkombinationen
WO2011127388A2 (en)	2010-04-08	2011-10-13	The United States Of America, As Represented By The Secretary, Department Of Health And Human Services	Inverse agonists and neutral antagonists for the tsh receptor
WO2016029372A1 (en)	2014-08-27	2016-03-03	The Procter & Gamble Company	Wearable article having elastic belt
WO2016029375A1 (en)	2014-08-27	2016-03-03	The Procter & Gamble Company	Wearable article having elastic belt
RU2619091C2 (ru) *	2015-10-13	2017-05-11	Министерство Промышленности И Торговли Рф	Цилиндрический термоэмиссионный катод
CN108883011B (zh)	2016-04-08	2021-05-07	宝洁公司	具有艺术作品的可穿着制品
CA3258277A1 (en) *	2022-06-08	2023-12-14	Icahn School Of Medicine At Mount Sinai	METHOD FOR OBESITY TREATMENT WITH A LUTEINIZING HORMONE RECEPTOR AGONIST

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0303306B1 (en)	1987-08-08	1993-03-10	Akzo N.V.	Contraceptive implant
TW564247B (en) *	1999-04-08	2003-12-01	Akzo Nobel Nv	Bicyclic heteraromatic compound

2002
- 2002-07-22 TW TW091116284A patent/TWI228508B/zh not_active IP Right Cessation
- 2002-08-29 CA CA2456901A patent/CA2456901C/en not_active Expired - Fee Related
- 2002-08-29 MX MXPA04002045A patent/MXPA04002045A/es active IP Right Grant
- 2002-08-29 IL IL16008402A patent/IL160084A0/xx not_active IP Right Cessation
- 2002-08-29 ES ES02772230T patent/ES2275005T3/es not_active Expired - Lifetime
- 2002-08-29 HU HU0401444A patent/HUP0401444A3/hu unknown
- 2002-08-29 DK DK02772230T patent/DK1427733T3/da active
- 2002-08-29 BR BR0211938-2A patent/BR0211938A/pt not_active IP Right Cessation
- 2002-08-29 EP EP02772230A patent/EP1427733B1/en not_active Expired - Lifetime
- 2002-08-29 PT PT02772230T patent/PT1427733E/pt unknown
- 2002-08-29 NZ NZ531340A patent/NZ531340A/en unknown
- 2002-08-29 HR HR20040202A patent/HRP20040202A2/hr not_active Application Discontinuation
- 2002-08-29 JP JP2003524996A patent/JP4262092B2/ja not_active Expired - Fee Related
- 2002-08-29 AT AT02772230T patent/ATE345345T1/de not_active IP Right Cessation
- 2002-08-29 AU AU2002337035A patent/AU2002337035B2/en not_active Ceased
- 2002-08-29 PL PL02368502A patent/PL368502A1/xx not_active Application Discontinuation
- 2002-08-29 DE DE60216128T patent/DE60216128T2/de not_active Expired - Lifetime
- 2002-08-29 CN CNB028172604A patent/CN1246324C/zh not_active Expired - Fee Related
- 2002-08-29 WO PCT/EP2002/009647 patent/WO2003020726A1/en not_active Ceased
- 2002-08-29 KR KR1020047003095A patent/KR100900018B1/ko not_active Expired - Fee Related
- 2002-08-29 US US10/488,482 patent/US7317006B2/en not_active Expired - Lifetime
- 2002-08-29 RU RU2004110042/04A patent/RU2298011C2/ru not_active IP Right Cessation
- 2002-09-02 AR ARP020103309A patent/AR036407A1/es unknown
- 2002-09-03 PE PE2002000840A patent/PE20030439A1/es not_active Application Discontinuation
2004
- 2004-01-29 IS IS7130A patent/IS2424B/is unknown
- 2004-02-23 ZA ZA200401455A patent/ZA200401455B/en unknown
- 2004-03-03 NO NO20040927A patent/NO20040927L/no not_active Application Discontinuation
2007
- 2007-02-13 CY CY20071100189T patent/CY1106012T1/el unknown

Also Published As

Publication number	Publication date
CY1106012T1 (el)	2011-04-06
CA2456901A1 (en)	2003-03-13
PE20030439A1 (es)	2003-05-17
RU2004110042A (ru)	2005-08-20
NO20040927L (no)	2004-03-03
ES2275005T3 (es)	2007-06-01
KR20040029134A (ko)	2004-04-03
HUP0401444A3 (en)	2008-05-28
MXPA04002045A (es)	2004-07-08
EP1427733B1 (en)	2006-11-15
HRP20040202A2 (en)	2004-08-31
JP2005505555A (ja)	2005-02-24
IS2424B (is)	2008-10-15
DK1427733T3 (da)	2007-03-19
CN1551884A (zh)	2004-12-01
NZ531340A (en)	2005-08-26
HUP0401444A2 (hu)	2004-11-29
PL368502A1 (en)	2005-04-04
US20040180873A1 (en)	2004-09-16
CN1246324C (zh)	2006-03-22
PT1427733E (pt)	2007-02-28
DE60216128D1 (de)	2006-12-28
WO2003020726A1 (en)	2003-03-13
JP4262092B2 (ja)	2009-05-13
AU2002337035B2 (en)	2008-04-24
TWI228508B (en)	2005-03-01
US7317006B2 (en)	2008-01-08
AR036407A1 (es)	2004-09-08
EP1427733A1 (en)	2004-06-16
ATE345345T1 (de)	2006-12-15
IS7130A (is)	2004-01-29
CA2456901C (en)	2011-01-04
DE60216128T2 (de)	2007-09-27
BR0211938A (pt)	2004-09-21
ZA200401455B (en)	2004-11-19
RU2298011C2 (ru)	2007-04-27
KR100900018B1 (ko)	2009-06-01

Publication	Publication Date	Title
IL159832A0 (en)	2004-06-20	4-amino-6-phenyl-pyrrolo[2,3-d] pyrimidine derivatives
TWI371450B (en)	2012-09-01	Novel substituted dihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use
PL363866A1 (en)	2004-11-29	4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives
IL160084A0 (en)	2004-06-20	Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity
PL353366A1 (en)	2003-11-17	Pyrazolo[4,3-d]pyrimidines
PL358551A1 (en)	2004-08-09	5-aminoalkyl-pyrazolo[4,3-d]pyrimidines
IL135982A0 (en)	2001-05-20	Fungicidal combinations comprising thieno[2,3-d]pyrimidin-4-one
MXPA03006802A (es)	2003-11-13	Formulaciones farmaceuticas que contienen pirazolo (4,3-d) pirimidinas y antagonistas del receptor de endotelina o tienopirimidinas y antagonistas del receptor de endotelina.
IL160194A0 (en)	2004-07-25	GLYCINE-SUBSTITUTED THIENO [2,3-d] PYRIMIDINE WITH COMBINED LH AND FSH AGONISTIC ACTIVITY
HUP0104350A3 (en)	2002-12-28	Synergetic fungicidal composition comprising thieno[2,3-d]pyrimidin-4-one and its use
MXPA03004498A (es)	2003-09-05	Uso de pirazolo (4,3-d)pirimidinas.
MXPA03004907A (es)	2003-09-05	Uso de pirazolo (4,3-d) pirimidinas.
GB2363377B (en)	2004-06-09	Novel thieno[2,3-d]pyrimidinediones and therapeutic uses thereof
AU8578501A (en)	2002-01-08	2-aminoalkyl-thieno(2,3-d)pyrimidines
HK1064387A (en)	2005-01-28	Thieno [2,3-d] pyrimidines with combined lh and fsh agonistic activity
HK1064386A (en)	2005-01-28	Glycine-substituted thieno [2,3-d] pyrimidines with combined lh and fsh agonistic activity
IL155380A0 (en)	2003-11-23	SUBSTITUTED 3,4-DIHYDRO-PYRIDO[1,2-a] PYRIMIDINES
GB0130695D0 (en)	2002-02-06	Pyrazola[4,3]pyrimidine
AU2002226519A1 (en)	2002-07-24	Pyrrolo(2,3-d)pyrimidine and their use as purinergic receptor antagonists
SI1210349T1 (en)	2003-06-30	PYRAZOLO 4,3-d)PYRIMIDINES
AU2002217336A1 (en)	2002-07-24	Thieno(3,2-d)pyrimidines and furano(3,2-d)pyrimidines and their use as purinergic receptor antagonists
HK1065035A (en)	2005-02-08	4-thioxo-4, 7-dihydro-thieno[2,3-b]pyridine-5-carboxamides as antiviral agents
AU2002305292A1 (en)	2002-11-11	Novel 4-amino-5,6-substituted thiopheno(2,3-d)pyrimidines
ZA200110327B (en)	2003-05-28	Hexahydropyrrolo(1,2-C)pyrimidines as antiviral, antifungal and/or antitumor agents.
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Legal Events

Date	Code	Title	Description
2010-11-30	FF	Patent granted
2011-07-31	MM9K	Patent not in force due to non-payment of renewal fees