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IL166821A0 - Novel 1,4-diazabicycloalkane derivatives their preparation and use - Google Patents

Novel 1,4-diazabicycloalkane derivatives their preparation and use

Info

Publication number
IL166821A0
IL166821A0 IL16682105A IL16682105A IL166821A0 IL 166821 A0 IL166821 A0 IL 166821A0 IL 16682105 A IL16682105 A IL 16682105A IL 16682105 A IL16682105 A IL 16682105A IL 166821 A0 IL166821 A0 IL 166821A0
Authority
IL
Israel
Prior art keywords
novel
preparation
diazabicycloalkane derivatives
diazabicycloalkane
derivatives
Prior art date
Application number
IL16682105A
Other versions
IL166821A (en
Original Assignee
Neurosearch As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/DK2003/000639 external-priority patent/WO2004029053A1/en
Application filed by Neurosearch As filed Critical Neurosearch As
Publication of IL166821A0 publication Critical patent/IL166821A0/en
Publication of IL166821A publication Critical patent/IL166821A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL166821A 2002-09-30 2005-02-10 1,4-diazabicyloalkane derivatives, their preparation and use IL166821A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200201456 2002-09-30
DKPA200201738 2002-11-11
PCT/DK2003/000639 WO2004029053A1 (en) 2002-09-30 2003-09-29 Novel 1,4-diazabicycloalkane derivatives, their preparation and use

Publications (2)

Publication Number Publication Date
IL166821A0 true IL166821A0 (en) 2006-01-15
IL166821A IL166821A (en) 2009-06-15

Family

ID=34828377

Family Applications (1)

Application Number Title Priority Date Filing Date
IL166821A IL166821A (en) 2002-09-30 2005-02-10 1,4-diazabicyloalkane derivatives, their preparation and use

Country Status (11)

Country Link
JP (1) JP4711391B2 (en)
KR (1) KR20050062575A (en)
CN (1) CN1326857C (en)
BR (1) BR0314183A (en)
IL (1) IL166821A (en)
IS (1) IS7829A (en)
MX (1) MXPA05003344A (en)
NO (1) NO20052124L (en)
PT (1) PT1551835E (en)
RU (1) RU2323218C2 (en)
SI (1) SI1551835T1 (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2368614C2 (en) * 2004-02-04 2009-09-27 НьюроСёрч А/С Diazabicyclic aryl derivatives used as modulators of cholinergic receptors
JO3019B1 (en) * 2006-04-19 2016-09-05 Janssen Pharmaceutica Nv Trisubstituted 1,2,4-Triazoles
AU2007267175A1 (en) * 2006-05-30 2007-12-06 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl derivatives and their medical use
WO2008016123A1 (en) * 2006-08-03 2008-02-07 Takeda Pharmaceutical Company Limited GSK-3β INHIBITOR
AR065344A1 (en) * 2007-02-15 2009-06-03 Argenta Discovery Ltd DERIVATIVES OF AZONIA OCTANO BICYCLE AS ACTIVATORS OF THE M3 RECEIVER
BR112014012056B1 (en) 2011-11-18 2021-12-14 Heptares Therapeutics Limited MUSCARINE M1 RECEPTOR AGONIST COMPOUNDS, A PHARMACEUTICAL COMPOSITION COMPRISING SUCH COMPOUNDS AND USE THEREOF TO TREAT A COGNITIVE OR PSYCHOTIC DISORDER OR TO TREAT OR REDUCE THE SEVERITY OF ACUTE, CHRONIC, NEUROPATHIC OR INFLAMMATORY PAIN
GB201404922D0 (en) 2014-03-19 2014-04-30 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201513743D0 (en) 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonists
GB201519352D0 (en) 2015-11-02 2015-12-16 Heptares Therapeutics Ltd Pharmaceutical compounds
EA201800367A1 (en) * 2015-12-10 2019-02-28 ПиТиСи ТЕРАПЬЮТИКС, ИНК. METHODS OF TREATMENT OF HUNTINGTON'S DISEASE
CN106432126B (en) * 2016-09-18 2018-12-28 广西师范大学 1-Oxygen-2,8-diazacyclononane derivative and its synthesis method
GB201617454D0 (en) 2016-10-14 2016-11-30 Heptares Therapeutics Limited Pharmaceutical compounds
GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ226000A (en) * 1987-09-10 1991-06-25 Merck Sharp & Dohme Oxadiazolyl-azabicycloheptanes and pharmaceutical compositions
US5854239A (en) * 1993-12-29 1998-12-29 Pfizer Inc. Diazabicyclic neuokinin antagonists
US5478939A (en) * 1994-07-20 1995-12-26 American Cyanamid Company (R,R) and (S,S) 2,5-diazabicyclo [2,2,1]heptane derivatives
FR2786770B1 (en) * 1998-12-04 2001-01-19 Synthelabo NONANE 1,4-DIAZABICYCLO [3.2.2.] DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
AU781235B2 (en) * 1999-07-09 2005-05-12 Ortho-Mcneil Pharmaceutical, Inc. Neurotrophic pyrrolidines and piperidines, and related compositions and methods
FR2804430B1 (en) * 2000-01-28 2002-03-22 Sanofi Synthelabo 4-HETEROARYL-1,4-DIAZABICYCLO [3.2.2] NONANE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2809732B1 (en) * 2000-05-31 2002-07-19 Sanofi Synthelabo DERIVATIVES OF 4 (-2-PHENYLTHIAZOL-5-yl) -1,4-DIAZABICYCLO- [3.2.2] NONANE, THEIR PREPARATION AND THEIR THERAPY APPLICATION
FR2809731B1 (en) * 2000-05-31 2002-07-19 Sanofi Synthelabo 1,4-DIAZABICYCLO- [3.2.2] NONANE-PHEYLISOXAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
US20020086871A1 (en) * 2000-12-29 2002-07-04 O'neill Brian Thomas Pharmaceutical composition for the treatment of CNS and other disorders
FR2832713B1 (en) * 2001-11-23 2004-02-13 Sanofi Synthelabo DERIVATIVES OF 4- (1,3,4-THIADIAZOL-2-YL) -1,4-DIAZABICYCLO [3.2.2] NONANE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Also Published As

Publication number Publication date
MXPA05003344A (en) 2005-11-23
RU2323218C2 (en) 2008-04-27
CN1684965A (en) 2005-10-19
RU2005105048A (en) 2005-11-20
HK1081954A1 (en) 2006-05-26
NO20052124L (en) 2005-06-29
NO20052124D0 (en) 2005-04-29
CN1326857C (en) 2007-07-18
PT1551835E (en) 2007-03-30
KR20050062575A (en) 2005-06-23
SI1551835T1 (en) 2007-06-30
JP4711391B2 (en) 2011-06-29
IS7829A (en) 2005-04-28
IL166821A (en) 2009-06-15
JP2006503062A (en) 2006-01-26
BR0314183A (en) 2005-08-09

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees