IL155520A0 - Benzoxazinone derivatives, their preparation and use - Google Patents

Benzoxazinone derivatives, their preparation and use

Info

Publication number: IL155520A0
Authority: IL; Israel
Prior art keywords: preparation; benzoxazinone derivatives; benzoxazinone; derivatives
Prior art date: 2000-10-26

Application number

IL15552001A

Other languages

English (en)

Original Assignee

Smithkline Beecham Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-26

Filing date

2001-10-22

Publication date

2003-11-23

2000-10-26 Priority claimed from GB0026224A external-priority patent/GB0026224D0/en

2001-05-15 Priority claimed from GB0111858A external-priority patent/GB0111858D0/en

2001-10-22 Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc

2003-11-23 Publication of IL155520A0 publication Critical patent/IL155520A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

IL15552001A 2000-10-26 2001-10-22 Benzoxazinone derivatives, their preparation and use IL155520A0 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB0026224A GB0026224D0 (en)	2000-10-26	2000-10-26	Novel compounds
GB0111858A GB0111858D0 (en)	2001-05-15	2001-05-15	Novel compounds
PCT/EP2001/012344 WO2002034754A2 (en)	2000-10-26	2001-10-22	Benzoxazinone derivatives, their preparation and use

Publications (1)

Publication Number	Publication Date
IL155520A0 true IL155520A0 (en)	2003-11-23

Family

ID=26245199

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL15552001A IL155520A0 (en)	2000-10-26	2001-10-22	Benzoxazinone derivatives, their preparation and use

Country Status (20)

Country	Link
US (1)	US6939871B2 (es)
EP (1)	EP1330460B1 (es)
JP (1)	JP4242643B2 (es)
KR (1)	KR20030051747A (es)
CN (1)	CN1478092A (es)
AR (1)	AR034174A1 (es)
AT (1)	ATE357448T1 (es)
AU (1)	AU2002224791A1 (es)
BR (1)	BR0114881A (es)
CA (1)	CA2426706A1 (es)
CZ (1)	CZ20031163A3 (es)
DE (1)	DE60127434T2 (es)
ES (1)	ES2280417T3 (es)
HU (1)	HUP0301458A2 (es)
IL (1)	IL155520A0 (es)
MX (1)	MXPA03003820A (es)
NO (1)	NO20031838L (es)
PL (1)	PL366378A1 (es)
TW (1)	TWI237023B (es)
WO (1)	WO2002034754A2 (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0203804D0 (en)	2002-02-18	2002-04-03	Glaxo Group Ltd	Compounds
GB0203811D0 (en)	2002-02-18	2002-04-03	Glaxo Group Ltd	Compounds
GB0203778D0 (en) *	2002-02-18	2002-04-03	Glaxo Group Ltd	Compounds
GB0209244D0 (en) *	2002-04-23	2002-06-05	Glaxo Group Ltd	Compounds
MXPA05002003A (es) *	2002-09-26	2005-08-03	Warner Lambert Co	Piperazinas sustituidas heterociclicas para el tratamiento de la esquizofrenia.
BR0315221A (pt)	2002-10-10	2005-08-23	Morphochem Ag Komb Chemie	Compostos com atividade antibacteriana
KR100683361B1 (ko)	2002-11-08	2007-02-15	에프. 호프만-라 로슈 아게	치환된 벤즈옥사진온 및 그의 용도
GB0227240D0 (en) *	2002-11-21	2002-12-31	Glaxo Group Ltd	Compounds
EP1600067B1 (en)	2003-01-10	2012-12-12	Zuiko Corporation	Wearing article and method of manufacturing the same
CA2523085A1 (en) *	2003-04-30	2004-11-18	Fmc Corporation	Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives
GB0310849D0 (en) *	2003-05-12	2003-06-18	Glaxo Group Ltd	Compounds
GB0310851D0 (en) *	2003-05-12	2003-06-18	Glaxo Group Ltd	Compounds
GB0316915D0 (en)	2003-07-18	2003-08-20	Glaxo Group Ltd	Compounds
CN101365696A (zh) *	2004-07-28	2009-02-11	Irm责任有限公司	作为类固醇激素核受体调节剂的化合物和组合物
JP2009511530A (ja) *	2005-10-13	2009-03-19	モルフォケムアクチェンゲゼルシャフトフュアコンビナトリシェヘミー	抗菌活性を有する５−キノリン誘導体
CA2750047A1 (en)	2009-01-21	2010-07-29	Basilea Pharmaceutica Ag	Novel bicyclic antibiotics
PT2513115E (pt)	2009-12-18	2013-12-19	Basilea Pharmaceutica Ag	Antibióticos tricíclicos
US9321788B2 (en)	2011-06-17	2016-04-26	Basilea Pharmaceutica Ag	Tricyclic antibiotics
SMT201900517T1 (it)	2017-03-20	2019-11-13	Forma Therapeutics Inc	Composizioni di pirrolopirrolo come attivatori di piruvato chinasi (pkr)
US20200129485A1 (en)	2018-09-19	2020-04-30	Forma Therapeutics, Inc.	Treating sickle cell disease with a pyruvate kinase r activating compound
CN113226356B (zh)	2018-09-19	2025-03-04	诺沃挪第克健康护理股份公司	活化丙酮酸激酶r
CN114615977B (zh)	2019-09-19	2025-01-14	诺沃挪第克健康护理股份公司	丙酮酸激酶r(pkr)活化组合物
US12128035B2 (en)	2021-03-19	2024-10-29	Novo Nordisk Health Care Ag	Activating pyruvate kinase R

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2191180T3 (es) *	1996-05-29	2003-09-01	Warner Lambert Co	Antagonistas de los receptores de la dopamina benzoxazinona d4.
EP0900792B1 (en)	1997-09-02	2003-10-29	Duphar International Research B.V	Piperazine and piperidine derivatives as 5-HT1A and dopamine D2-receptor (ant)agonists
AU2494300A (en) *	1999-01-07	2000-07-24	American Home Products Corporation	3,4-dihydro-2h-benzo(1,4)oxazine derivatives
TW546299B (en) *	1999-01-07	2003-08-11	Wyeth Corp	3,4-dihydro-2H-benzo[1,4]oxazinyl-methyl-[3-(1H-indol-3-yl)-alkyl]-amines

2001
- 2001-10-22 CA CA002426706A patent/CA2426706A1/en not_active Abandoned
- 2001-10-22 DE DE60127434T patent/DE60127434T2/de not_active Expired - Fee Related
- 2001-10-22 WO PCT/EP2001/012344 patent/WO2002034754A2/en not_active Ceased
- 2001-10-22 MX MXPA03003820A patent/MXPA03003820A/es unknown
- 2001-10-22 KR KR10-2003-7005789A patent/KR20030051747A/ko not_active Withdrawn
- 2001-10-22 IL IL15552001A patent/IL155520A0/xx unknown
- 2001-10-22 US US10/415,119 patent/US6939871B2/en not_active Expired - Fee Related
- 2001-10-22 HU HU0301458A patent/HUP0301458A2/hu unknown
- 2001-10-22 CZ CZ20031163A patent/CZ20031163A3/cs unknown
- 2001-10-22 ES ES01988720T patent/ES2280417T3/es not_active Expired - Lifetime
- 2001-10-22 BR BR0114881-8A patent/BR0114881A/pt not_active IP Right Cessation
- 2001-10-22 PL PL01366378A patent/PL366378A1/xx not_active Application Discontinuation
- 2001-10-22 EP EP01988720A patent/EP1330460B1/en not_active Expired - Lifetime
- 2001-10-22 AU AU2002224791A patent/AU2002224791A1/en not_active Abandoned
- 2001-10-22 CN CNA018197663A patent/CN1478092A/zh active Pending
- 2001-10-22 JP JP2002537744A patent/JP4242643B2/ja not_active Expired - Fee Related
- 2001-10-22 AT AT01988720T patent/ATE357448T1/de not_active IP Right Cessation
- 2001-10-24 TW TW090126222A patent/TWI237023B/zh not_active IP Right Cessation
- 2001-10-24 AR ARP010104975A patent/AR034174A1/es not_active Application Discontinuation
2003
- 2003-04-24 NO NO20031838A patent/NO20031838L/no unknown

Also Published As

Publication number	Publication date
MXPA03003820A (es)	2003-07-28
EP1330460B1 (en)	2007-03-21
US6939871B2 (en)	2005-09-06
KR20030051747A (ko)	2003-06-25
HUP0301458A2 (hu)	2003-10-28
US20040063704A1 (en)	2004-04-01
WO2002034754A3 (en)	2002-07-11
ES2280417T3 (es)	2007-09-16
NO20031838L (no)	2003-06-24
JP4242643B2 (ja)	2009-03-25
CZ20031163A3 (cs)	2004-04-14
PL366378A1 (en)	2005-01-24
NO20031838D0 (no)	2003-04-24
WO2002034754A2 (en)	2002-05-02
TWI237023B (en)	2005-08-01
CN1478092A (zh)	2004-02-25
BR0114881A (pt)	2003-09-30
ATE357448T1 (de)	2007-04-15
JP2004516250A (ja)	2004-06-03
AR034174A1 (es)	2004-02-04
AU2002224791A1 (en)	2002-05-06
EP1330460A2 (en)	2003-07-30
CA2426706A1 (en)	2002-05-02
DE60127434T2 (de)	2007-11-29
DE60127434D1 (de)	2007-05-03

Publication	Publication Date	Title
IL155520A0 (en)	2003-11-23	Benzoxazinone derivatives, their preparation and use
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ZA200107983B (en)	2002-05-29	New compounds, their preparation and use.
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IL159275A0 (en)	2004-06-01	Phenylsulfonyl-1, 3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use
AU2001248279A1 (en)	2001-10-30	New compounds, their preparation and use
AU2002359126A8 (en)	2003-06-30	Benzodiazepine derivatives, preparation thereof and use thereof
HUP0303291A3 (en)	2005-11-28	Herbicidal composition, preparation and use thereof
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