ID26804A - Metode untuk menghambat mrp1 - Google Patents
Metode untuk menghambat mrp1Info
- Publication number
- ID26804A ID26804A IDW20002006A ID20002006A ID26804A ID 26804 A ID26804 A ID 26804A ID W20002006 A IDW20002006 A ID W20002006A ID 20002006 A ID20002006 A ID 20002006A ID 26804 A ID26804 A ID 26804A
- Authority
- ID
- Indonesia
- Prior art keywords
- inhibiting mrp1
- mrp1
- inhibiting
- Prior art date
Links
- 102100021339 Multidrug resistance-associated protein 1 Human genes 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 108010066052 multidrug resistance-associated protein 1 Proteins 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8108898P | 1998-04-08 | 1998-04-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ID26804A true ID26804A (id) | 2001-02-08 |
Family
ID=22162031
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IDW20002006A ID26804A (id) | 1998-04-08 | 1999-04-07 | Metode untuk menghambat mrp1 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US6221876B1 (id) |
| EP (1) | EP1067932A4 (id) |
| JP (1) | JP2002510632A (id) |
| KR (1) | KR20010042481A (id) |
| CN (1) | CN1296410A (id) |
| AU (1) | AU3550299A (id) |
| BR (1) | BR9909446A (id) |
| CA (1) | CA2327452A1 (id) |
| EA (1) | EA200001035A1 (id) |
| HU (1) | HUP0102548A2 (id) |
| ID (1) | ID26804A (id) |
| IL (1) | IL138393A0 (id) |
| NO (1) | NO20005041L (id) |
| PL (1) | PL343320A1 (id) |
| SK (1) | SK14992000A3 (id) |
| TR (1) | TR200002804T2 (id) |
| WO (1) | WO1999051236A1 (id) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE315033T1 (de) | 1998-08-07 | 2006-02-15 | Chiron Corp | Subtituierte isoxazole derivate als estrogen rezeptor modulatore |
| WO2001046199A1 (en) * | 1999-12-22 | 2001-06-28 | Eli Lilly And Company | Methods and compounds for inhibiting mrp1 |
| US6743794B2 (en) | 1999-12-22 | 2004-06-01 | Eli Lilly And Company | Methods and compounds for inhibiting MRP1 |
| CA2411813A1 (en) * | 2000-06-14 | 2001-12-20 | Eli Lilly And Company | Tricyclic compounds as mrp1-inhibitors |
| WO2002081481A1 (en) * | 2001-04-09 | 2002-10-17 | Eli Lilly And Company | Compounds and methods for inhibiting mrp1 |
| CN1281210C (zh) * | 2003-11-29 | 2006-10-25 | 胡汛 | 五味子乙素在制备治疗肿瘤药物中的应用 |
| WO2005113004A2 (en) * | 2004-05-14 | 2005-12-01 | The Cleveland Clinic Founfation | Small molecule inhibitors for mrp1 and other multidrug transporters |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5182290A (en) * | 1991-08-27 | 1993-01-26 | Neurogen Corporation | Certain oxazoloquinolinones; a new class of GABA brain receptor ligands |
-
1999
- 1999-04-07 TR TR2000/02804T patent/TR200002804T2/xx unknown
- 1999-04-07 US US09/646,063 patent/US6221876B1/en not_active Expired - Fee Related
- 1999-04-07 CN CN99804797A patent/CN1296410A/zh active Pending
- 1999-04-07 WO PCT/US1999/007615 patent/WO1999051236A1/en not_active Ceased
- 1999-04-07 PL PL99343320A patent/PL343320A1/xx not_active Application Discontinuation
- 1999-04-07 BR BR9909446-0A patent/BR9909446A/pt not_active IP Right Cessation
- 1999-04-07 HU HU0102548A patent/HUP0102548A2/hu unknown
- 1999-04-07 ID IDW20002006A patent/ID26804A/id unknown
- 1999-04-07 AU AU35502/99A patent/AU3550299A/en not_active Abandoned
- 1999-04-07 EA EA200001035A patent/EA200001035A1/ru unknown
- 1999-04-07 CA CA002327452A patent/CA2327452A1/en not_active Abandoned
- 1999-04-07 EP EP99917359A patent/EP1067932A4/en not_active Withdrawn
- 1999-04-07 KR KR1020007011101A patent/KR20010042481A/ko not_active Withdrawn
- 1999-04-07 IL IL13839399A patent/IL138393A0/xx unknown
- 1999-04-07 SK SK1499-2000A patent/SK14992000A3/sk unknown
- 1999-04-07 JP JP2000542007A patent/JP2002510632A/ja not_active Withdrawn
-
2000
- 2000-10-06 NO NO20005041A patent/NO20005041L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IL138393A0 (en) | 2001-10-31 |
| NO20005041D0 (no) | 2000-10-06 |
| CN1296410A (zh) | 2001-05-23 |
| PL343320A1 (en) | 2001-08-13 |
| EP1067932A1 (en) | 2001-01-17 |
| WO1999051236A1 (en) | 1999-10-14 |
| KR20010042481A (ko) | 2001-05-25 |
| CA2327452A1 (en) | 1999-10-14 |
| TR200002804T2 (tr) | 2001-02-21 |
| EP1067932A4 (en) | 2001-11-14 |
| BR9909446A (pt) | 2000-12-12 |
| JP2002510632A (ja) | 2002-04-09 |
| SK14992000A3 (sk) | 2001-06-11 |
| AU3550299A (en) | 1999-10-25 |
| NO20005041L (no) | 2000-10-06 |
| EA200001035A1 (ru) | 2001-04-23 |
| US6221876B1 (en) | 2001-04-24 |
| HUP0102548A2 (hu) | 2001-11-28 |
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