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HUP9700806A2 - Tianeptin-nátriumsó nyújtott felszabadulását biztosító, szájon át beadható mátrix tabletta és eljárás előállítására - Google Patents

Tianeptin-nátriumsó nyújtott felszabadulását biztosító, szájon át beadható mátrix tabletta és eljárás előállítására

Info

Publication number
HUP9700806A2
HUP9700806A2 HU9700806A HUP9700806A HUP9700806A2 HU P9700806 A2 HUP9700806 A2 HU P9700806A2 HU 9700806 A HU9700806 A HU 9700806A HU P9700806 A HUP9700806 A HU P9700806A HU P9700806 A2 HUP9700806 A2 HU P9700806A2
Authority
HU
Hungary
Prior art keywords
matrix tablet
sodium salt
tianeptine
preparation
prolonged release
Prior art date
Application number
HU9700806A
Other languages
English (en)
Inventor
Bruno Huet De Barochez
Patrick Wüthrich
Original Assignee
Adir Et Compagnie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adir Et Compagnie filed Critical Adir Et Compagnie
Publication of HU9700806D0 publication Critical patent/HU9700806D0/hu
Publication of HUP9700806A2 publication Critical patent/HUP9700806A2/hu
Publication of HUP9700806A3 publication Critical patent/HUP9700806A3/hu
Publication of HU224192B1 publication Critical patent/HU224192B1/hu

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Engineering & Computer Science (AREA)
  • Inorganic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Cephalosporin Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

A találmány tárgya tianeptin-nátriűmsó nyújtőtt felszabadűlásátbiztősító mátrixtabletta, mely galenikűs főrmában őrális útőn adhatóbe, és felszívódás űtán a vérben állandó és egyenletes kőncentrációtbiztősít. A találmány tárgya tővábbá eljárás a mátrixtabletta előállítására. Atianeptin elsősőrban szőrőngás és depresszió kezelésére alkalmas. ŕ
HU9700806A 1996-04-24 1997-04-24 Tianeptin-nátriumsó nyújtott felszabadulását biztosító, szájon át beadható mátrix tabletta és eljárás előállítására HU224192B1 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9605174A FR2747921B1 (fr) 1996-04-24 1996-04-24 Comprime matriciel permettant la liberation prolongee du sel de sodium de tianeptine apres administration par voie orale

Publications (4)

Publication Number Publication Date
HU9700806D0 HU9700806D0 (en) 1997-06-30
HUP9700806A2 true HUP9700806A2 (hu) 1998-10-28
HUP9700806A3 HUP9700806A3 (en) 2000-01-28
HU224192B1 HU224192B1 (hu) 2005-06-28

Family

ID=9491549

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9700806A HU224192B1 (hu) 1996-04-24 1997-04-24 Tianeptin-nátriumsó nyújtott felszabadulását biztosító, szájon át beadható mátrix tabletta és eljárás előállítására

Country Status (18)

Country Link
US (1) US5888542A (hu)
EP (1) EP0803253B1 (hu)
JP (1) JPH1036268A (hu)
CN (1) CN1116029C (hu)
AT (1) ATE205715T1 (hu)
AU (1) AU719822B2 (hu)
CA (1) CA2203310C (hu)
DE (1) DE69706748T2 (hu)
DK (1) DK0803253T3 (hu)
ES (1) ES2164310T3 (hu)
FR (1) FR2747921B1 (hu)
GR (1) GR3037043T3 (hu)
HU (1) HU224192B1 (hu)
NO (1) NO315407B1 (hu)
NZ (1) NZ314662A (hu)
PL (1) PL188135B1 (hu)
PT (1) PT803253E (hu)
ZA (1) ZA973495B (hu)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2791891A1 (fr) * 1999-04-07 2000-10-13 Adir Utilisation de la tianeptine pour l'obtention de medicaments destines au traitement des pathologies de la neurodegenerescence
US6683072B1 (en) 2003-02-04 2004-01-27 Vela Pharmaceuticals, Inc. Compositions and methods for treatment of irritable bowel syndrome and nonulcer dyspepsia
EP1575565B1 (en) * 2003-08-08 2010-01-06 Biovail Laboratories International Srl Modified-release tablet of bupropion hydrochloride
US20050227961A1 (en) * 2004-04-08 2005-10-13 Vela Pharmaceuticals, Inc. Compositions and methods for treatment of neuropathic pain, fibromyalgia and chronic fatigue syndrome
US9314469B2 (en) 2008-05-05 2016-04-19 Tonix Pharma Holdings Limited Method for treating neurocognitive dysfunction
US8198268B2 (en) 2008-10-31 2012-06-12 Janssen Biotech, Inc. Tianeptine sulfate salt forms and methods of making and using the same
US8355927B2 (en) 2010-11-05 2013-01-15 Genomind, Llc Neuropsychiatric test reports
US20110237537A1 (en) * 2009-05-29 2011-09-29 Lombard Jay L Methods for assessment and treatment of mood disorders via single nucleotide polymorphisms analysis
WO2010138796A2 (en) * 2009-05-29 2010-12-02 Genomind, Llc Methods for assessment and treatment of depression via utilization of single nucleotide polymorphisms analysis
KR20120092993A (ko) * 2011-02-14 2012-08-22 지엘팜텍 주식회사 티아넵틴 또는 이의 약제학적으로 허용되는 염을 포함하는 경구투여용 서방성 정제
PL2561864T3 (pl) * 2011-08-25 2015-05-29 Zakl Farmaceutyczne Polpharma Sa Tabletka powlekana zawierająca tianeptynę i sposób jej otrzymywania
KR101136976B1 (ko) * 2011-09-06 2012-05-30 건일제약 주식회사 티아넵틴 또는 그의 염을 포함하는 탈모증의 예방 또는 치료용 약학 조성물
GB201208315D0 (en) 2012-05-11 2012-06-27 Numedicus Ltd Pharmaceutical methods and compositions
CN104031005B (zh) * 2014-05-30 2016-04-27 济南诚汇双达化工有限公司 一种噻萘普汀钠中间体的制备方法
KR20180101307A (ko) 2018-09-04 2018-09-12 지엘팜텍주식회사 티아넵틴 또는 이의 약제학적으로 허용되는 염을 포함하는 경구투여용 서방성 정제
KR20200104265A (ko) 2020-08-21 2020-09-03 지엘팜텍주식회사 티아넵틴 또는 이의 약제학적으로 허용되는 염을 포함하는 경구투여용 서방성 정제
WO2024206520A1 (en) 2023-03-27 2024-10-03 Tonix Pharmaceuticals Holding Corp. (s)-tianeptine and use in treating disorders and conditions associated with peroxisome proliferator-activated receptor

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5446070A (en) * 1991-02-27 1995-08-29 Nover Pharmaceuticals, Inc. Compositions and methods for topical administration of pharmaceutically active agents
FR2635461B1 (fr) * 1988-08-18 1992-01-17 Adir Utilisation de derives tricycliques pour l'obtention de medicaments destines au traitement du stress
FR2716623B1 (fr) * 1994-02-25 1996-08-23 Adir Utilisation d'un dérivé tricyclique pour l'obtention de médicaments destinés au traitement des troubles mnémo-cognitifs.

Also Published As

Publication number Publication date
NO971860L (no) 1997-10-27
CA2203310A1 (fr) 1997-10-24
PT803253E (pt) 2001-12-28
AU1904197A (en) 1997-10-30
CN1116029C (zh) 2003-07-30
ATE205715T1 (de) 2001-10-15
NZ314662A (en) 1998-12-23
US5888542A (en) 1999-03-30
DE69706748D1 (de) 2001-10-25
JPH1036268A (ja) 1998-02-10
PL188135B1 (pl) 2004-12-31
NO971860D0 (no) 1997-04-23
FR2747921A1 (fr) 1997-10-31
GR3037043T3 (en) 2002-01-31
HU224192B1 (hu) 2005-06-28
HUP9700806A3 (en) 2000-01-28
CA2203310C (fr) 2001-10-23
CN1168792A (zh) 1997-12-31
DK0803253T3 (da) 2001-11-19
ES2164310T3 (es) 2002-02-16
EP0803253A1 (fr) 1997-10-29
FR2747921B1 (fr) 1998-10-30
HU9700806D0 (en) 1997-06-30
AU719822B2 (en) 2000-05-18
NO315407B1 (no) 2003-09-01
EP0803253B1 (fr) 2001-09-19
DE69706748T2 (de) 2002-07-04
ZA973495B (en) 1997-11-18
PL319627A1 (en) 1997-10-27

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Legal Events

Date Code Title Description
HFG4 Patent granted, date of granting

Effective date: 20050420

MM4A Lapse of definitive patent protection due to non-payment of fees