HRP20060008A2 - 7-substituted 3-nitro-pyrazolo[1,5-a] pyrimidines - Google Patents

7-substituted 3-nitro-pyrazolo[1,5-a] pyrimidines

Info

Publication number: HRP20060008A2
Authority: HR; Croatia
Prior art keywords: pyrazolo; pyrimidines; nitro; substituted; compounds
Prior art date: 2003-07-24

Application number

HR20060008A

Other languages

English (en)

Croatian (hr)

Inventor

Anglada Luis

Palomer Albert

Princep Marta

Guglietta Antonio

Original Assignee

Ferrer Internacional

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-07-24

Filing date

2004-07-22

Publication date

2006-07-31

2003-07-24 Priority claimed from ES200301747A external-priority patent/ES2222814B1/es

2004-07-22 Application filed by Ferrer Internacional filed Critical Ferrer Internacional

2006-07-31 Publication of HRP20060008A2 publication Critical patent/HRP20060008A2/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Anesthesiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

HR20060008A 2003-07-24 2004-07-22 7-substituted 3-nitro-pyrazolo[1,5-a] pyrimidines HRP20060008A2 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
ES200301747A ES2222814B1 (es)	2003-07-24	2003-07-24	3-nitro-pirazolo(1,5-a)pirimidinas 7-sustituidas y composiciones y metodos relacionados.
ES200401696A ES2245893B1 (es)	2003-07-24	2004-07-12	Mejoras en el objeto de la patente de invencion n.p200301747 que se refiere a "3-nitro-pirazolo(1,5-a)pirimidinas 7-sustituidas y composiciones y metodos relacionados".
PCT/EP2004/008207 WO2005014596A1 (en)	2003-07-24	2004-07-22	7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines

Publications (1)

Publication Number	Publication Date
HRP20060008A2 true HRP20060008A2 (en)	2006-07-31

Family

ID=34137683

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HR20060008A HRP20060008A2 (en)	2003-07-24	2004-07-22	7-substituted 3-nitro-pyrazolo[1,5-a] pyrimidines

Country Status (15)

Country	Link
US (1)	US20070043064A1 (es)
EP (1)	EP1648896B1 (es)
JP (1)	JP2006528607A (es)
KR (1)	KR20060030907A (es)
AT (1)	ATE386040T1 (es)
AU (1)	AU2004263277A1 (es)
BR (1)	BRPI0412837A (es)
CA (1)	CA2532431A1 (es)
DE (1)	DE602004011780D1 (es)
HR (1)	HRP20060008A2 (es)
MX (1)	MXPA06000774A (es)
NO (1)	NO20060586L (es)
TW (1)	TWI252851B (es)
UY (1)	UY28439A1 (es)
WO (1)	WO2005014596A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20050245517A1 (en) *	2004-04-29	2005-11-03	Phil Skolnick	2-pyridinyl[7-(substituted-pyridin-4-yl) pyrazolo[1,5-a]pyrimidin-3-yl]methanones
EP1884516A1 (en) *	2006-08-04	2008-02-06	Ferrer Internacional, S.A.	Pyrazolo[1,5-a]pyrimidines, processes, uses and compositions
GB201223308D0 (en)	2012-12-21	2013-02-06	Univ Sunderland	Enzyme inhibitors

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE792533A (fr) *	1971-12-09	1973-06-08	Int Chem & Nuclear Corp	Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US4626538A (en) *	1983-06-23	1986-12-02	American Cyanamid Company	[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines
EP0264773A1 (en) *	1986-10-16	1988-04-27	American Cyanamid Company	4,5-dihydro and 4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidines
DE4333705C2 (de) *	1993-10-02	2003-10-30	Guenter Ege	Arylmethylsubstituierte Pyrazolo-azine, insbesondere 3-Arylmethylpyrazolo[1,5-a]pyrimidine und Verfahren zur Herstellung von 8-Arylmethyl-pyrazolo[5,1-c][1,2,4]triazinen
US5538977A (en) *	1995-03-17	1996-07-23	American Cyanamid Company	3-Substituted-7-[3-(imidazol-1-yl)phenyl]-pyrazolo[1,5-a]pyrimidines
WO2000059908A2 (en) *	1999-04-06	2000-10-12	Du Pont Pharmaceuticals Company	Pyrazolopyrimidines as crf antagonists
US6399621B1 (en) *	1999-08-10	2002-06-04	American Cyanamid Company	N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1, 5-α]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto
DE10153344A1 (de) *	2001-10-29	2003-05-15	Gruenenthal Gmbh	Verwendung von substituierten Pyrazolopyrimidinen als Liganden von Nucleosid-Transport-Proteinen und/oder von Purinorezeptoren

2004
- 2004-07-15 TW TW093121112A patent/TWI252851B/zh not_active IP Right Cessation
- 2004-07-22 KR KR1020067001168A patent/KR20060030907A/ko not_active Ceased
- 2004-07-22 US US10/563,104 patent/US20070043064A1/en not_active Abandoned
- 2004-07-22 JP JP2006520795A patent/JP2006528607A/ja not_active Abandoned
- 2004-07-22 EP EP04741222A patent/EP1648896B1/en not_active Expired - Lifetime
- 2004-07-22 AT AT04741222T patent/ATE386040T1/de not_active IP Right Cessation
- 2004-07-22 DE DE602004011780T patent/DE602004011780D1/de not_active Expired - Lifetime
- 2004-07-22 WO PCT/EP2004/008207 patent/WO2005014596A1/en not_active Ceased
- 2004-07-22 CA CA002532431A patent/CA2532431A1/en not_active Abandoned
- 2004-07-22 HR HR20060008A patent/HRP20060008A2/xx not_active Application Discontinuation
- 2004-07-22 BR BRPI0412837-0A patent/BRPI0412837A/pt not_active IP Right Cessation
- 2004-07-22 AU AU2004263277A patent/AU2004263277A1/en not_active Abandoned
- 2004-07-22 MX MXPA06000774A patent/MXPA06000774A/es not_active Application Discontinuation
- 2004-07-26 UY UY28439A patent/UY28439A1/es unknown
2006
- 2006-02-06 NO NO20060586A patent/NO20060586L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO2005014596A1 (en)	2005-02-17
TW200504074A (en)	2005-02-01
DE602004011780D1 (de)	2008-03-27
MXPA06000774A (es)	2006-04-18
BRPI0412837A (pt)	2006-09-26
AU2004263277A1 (en)	2005-02-17
US20070043064A1 (en)	2007-02-22
TWI252851B (en)	2006-04-11
CA2532431A1 (en)	2005-02-17
UY28439A1 (es)	2004-11-08
EP1648896A1 (en)	2006-04-26
KR20060030907A (ko)	2006-04-11
EP1648896B1 (en)	2008-02-13
JP2006528607A (ja)	2006-12-21
NO20060586L (no)	2006-02-06
ATE386040T1 (de)	2008-03-15

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Legal Events

Date	Code	Title	Description
2006-07-31	A1OB	Publication of a patent application
2007-05-31	AKOB	Publication of a request for the grant of a patent not including a substantive examination of a patent application (a consensual patent)
2007-07-20	ODRP	Renewal fee for the maintenance of a patent	Payment date: 20070720 Year of fee payment: 4
2009-02-06	ODBI	Application refused