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HN2010000295A - NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORS - Google Patents

NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORS

Info

Publication number
HN2010000295A
HN2010000295A HN2010000295A HN2010000295A HN2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A
Authority
HN
Honduras
Prior art keywords
new
triazolopiridacina
bencimidazol
benzotiazol
sulfanil
Prior art date
Application number
HN2010000295A
Other languages
Spanish (es)
Inventor
Albert Eva
Bacque Eric
Nemeneck Conception
Ugolini Antonio
Wentzler Sylvie
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of HN2010000295A publication Critical patent/HN2010000295A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A LSO PRODUCTOS NUEVOS DE LA FORMULA (I): EN LA QUE REPRESENTA UN ENLACE SENCILLO O DOBLE RA PRESENTADA H,Hal, ALCOXI, O- CICLOALQUILO HETEROARILO, FENILO, NHCOalk, NHCOcicloalk O NR1R2; X REPRESENTA S, SO, O SO3 ; A REPRESENTA NH O S; W REPRESENTA H, ALQUILO O COR CON R QUE REPRESENTA CICLOALQUILO; ALQUILO SUSTITUIDO OPCIONALEMNETE CON NR3R4 ALCOXI, HIDROXI, FELINO, HETEROARILO O HETEROCICLOALQUILO... VER EXPEDIENTETHE PRESENT INVENTION REFERS TO THE NEW PRODUCTS OF THE FORMULA (I): IN WHICH IT REPRESENTS A SINGLE OR DOUBLE RA LINK PRESENTED H, Hal, ALCOXI, O- CYCLALKYL HETEROARILE, PHENYL, NHCOalk, NHCOcicloalk OR NR1R2; X REPRESENTS S, SO, OR SO3; A REPRESENTATIVE NH O S; W REPRESENTS H, RENT OR COR WITH R THAT REPRESENTS CYCLALKYL; OPTIONAL SUBSTITUTE RENT WITH NR3R4 ALCOXI, HYDROXI, FELINE, HETEROARILO or HETEROCICLOALQUILO ... SEE RECORD

HN2010000295A 2007-08-09 2010-02-08 NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORS HN2010000295A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0705789A FR2919870B1 (en) 2007-08-09 2007-08-09 NOVEL 6-TRIAZOLOPYRIDAZINE-SULFANYL BENZOTHIAZOLE AND BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, PROCESS, PHARMACEUTICAL COMPOSITIONS, AND NOVEL USE AS CMET INHIBITORS

Publications (1)

Publication Number Publication Date
HN2010000295A true HN2010000295A (en) 2013-04-22

Family

ID=39304792

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2010000295A HN2010000295A (en) 2007-08-09 2010-02-08 NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORS

Country Status (3)

Country Link
FR (1) FR2919870B1 (en)
HN (1) HN2010000295A (en)
PH (1) PH12014501625A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010092371A1 (en) 2009-02-10 2010-08-19 Astrazeneca Ab Triazolo [4,3-b] pyridazine derivatives and their uses for prostate cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20080080584A (en) * 2005-11-30 2008-09-04 버텍스 파마슈티칼스 인코포레이티드 Inhibitors of c-methet and uses thereof
MY159523A (en) * 2005-12-21 2017-01-13 Janssen Pharmaceutica Nv Triazolopyridazines as tyrosine kinase modulators
CA2651979A1 (en) * 2006-05-30 2007-12-06 Pfizer Products Inc. Triazolopyridazine derivatives
PE20121506A1 (en) * 2006-07-14 2012-11-26 Amgen Inc TRIAZOLOPYRIDINE COMPOUNDS AS C-MET INHIBITORS

Also Published As

Publication number Publication date
FR2919870A1 (en) 2009-02-13
PH12014501625A1 (en) 2016-01-18
FR2919870B1 (en) 2014-05-16

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