HN2010000295A - NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORS - Google Patents
NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORSInfo
- Publication number
- HN2010000295A HN2010000295A HN2010000295A HN2010000295A HN2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A HN 2010000295 A HN2010000295 A HN 2010000295A
- Authority
- HN
- Honduras
- Prior art keywords
- new
- triazolopiridacina
- bencimidazol
- benzotiazol
- sulfanil
- Prior art date
Links
- 229940079593 drug Drugs 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 241000282324 Felis Species 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical class [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A LSO PRODUCTOS NUEVOS DE LA FORMULA (I): EN LA QUE REPRESENTA UN ENLACE SENCILLO O DOBLE RA PRESENTADA H,Hal, ALCOXI, O- CICLOALQUILO HETEROARILO, FENILO, NHCOalk, NHCOcicloalk O NR1R2; X REPRESENTA S, SO, O SO3 ; A REPRESENTA NH O S; W REPRESENTA H, ALQUILO O COR CON R QUE REPRESENTA CICLOALQUILO; ALQUILO SUSTITUIDO OPCIONALEMNETE CON NR3R4 ALCOXI, HIDROXI, FELINO, HETEROARILO O HETEROCICLOALQUILO... VER EXPEDIENTETHE PRESENT INVENTION REFERS TO THE NEW PRODUCTS OF THE FORMULA (I): IN WHICH IT REPRESENTS A SINGLE OR DOUBLE RA LINK PRESENTED H, Hal, ALCOXI, O- CYCLALKYL HETEROARILE, PHENYL, NHCOalk, NHCOcicloalk OR NR1R2; X REPRESENTS S, SO, OR SO3; A REPRESENTATIVE NH O S; W REPRESENTS H, RENT OR COR WITH R THAT REPRESENTS CYCLALKYL; OPTIONAL SUBSTITUTE RENT WITH NR3R4 ALCOXI, HYDROXI, FELINE, HETEROARILO or HETEROCICLOALQUILO ... SEE RECORD
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0705789A FR2919870B1 (en) | 2007-08-09 | 2007-08-09 | NOVEL 6-TRIAZOLOPYRIDAZINE-SULFANYL BENZOTHIAZOLE AND BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, PROCESS, PHARMACEUTICAL COMPOSITIONS, AND NOVEL USE AS CMET INHIBITORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HN2010000295A true HN2010000295A (en) | 2013-04-22 |
Family
ID=39304792
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HN2010000295A HN2010000295A (en) | 2007-08-09 | 2010-02-08 | NEW DERIVATIVES OF 6- TRIAZOLOPIRIDACINA-SULFANIL BENZOTIAZOL AND BENCIMIDAZOL ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICATIONS, PHARMACEUTICAL COMPOSITIONS AND NEW MAIN USE AS MET INHIBITORS |
Country Status (3)
| Country | Link |
|---|---|
| FR (1) | FR2919870B1 (en) |
| HN (1) | HN2010000295A (en) |
| PH (1) | PH12014501625A1 (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010092371A1 (en) | 2009-02-10 | 2010-08-19 | Astrazeneca Ab | Triazolo [4,3-b] pyridazine derivatives and their uses for prostate cancer |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20080080584A (en) * | 2005-11-30 | 2008-09-04 | 버텍스 파마슈티칼스 인코포레이티드 | Inhibitors of c-methet and uses thereof |
| MY159523A (en) * | 2005-12-21 | 2017-01-13 | Janssen Pharmaceutica Nv | Triazolopyridazines as tyrosine kinase modulators |
| CA2651979A1 (en) * | 2006-05-30 | 2007-12-06 | Pfizer Products Inc. | Triazolopyridazine derivatives |
| PE20121506A1 (en) * | 2006-07-14 | 2012-11-26 | Amgen Inc | TRIAZOLOPYRIDINE COMPOUNDS AS C-MET INHIBITORS |
-
2007
- 2007-08-09 FR FR0705789A patent/FR2919870B1/en not_active Expired - Fee Related
-
2010
- 2010-02-08 HN HN2010000295A patent/HN2010000295A/en unknown
-
2014
- 2014-07-15 PH PH12014501625A patent/PH12014501625A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2919870A1 (en) | 2009-02-13 |
| PH12014501625A1 (en) | 2016-01-18 |
| FR2919870B1 (en) | 2014-05-16 |
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