HN2001000019A - Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4. - Google Patents
Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4.Info
- Publication number
- HN2001000019A HN2001000019A HN2001000019A HN2001000019A HN2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A
- Authority
- HN
- Honduras
- Prior art keywords
- pde4
- isozimas
- benzocondensada
- heterociclico
- nicotinamide
- Prior art date
Links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract
LA PRESENTE INVENCION SE REFIERE TAMBIEN AL USO DE INHIBIDORES SELECTIVOS DE LAS PDE4 PARA UN MEJOR TRATAMIENTO TERAPEUTICO DE UNA SERIE DE ENFERMEDADES Y CONDICIONES INFLAMATORIAS, RESPIRATORIAS Y ALERGICAS, PERO ESPECIALMENTE PARA EL TRATAMIENTO DEL ASMA
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17928400P | 2000-01-31 | 2000-01-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HN2001000019A true HN2001000019A (es) | 2001-09-06 |
Family
ID=22655931
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HN2001000019A HN2001000019A (es) | 2000-01-31 | 2001-06-30 | Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4. |
Country Status (40)
| Country | Link |
|---|---|
| US (1) | US7354941B2 (es) |
| EP (1) | EP1252158B1 (es) |
| JP (1) | JP3917863B2 (es) |
| KR (1) | KR20020072299A (es) |
| CN (1) | CN1404481A (es) |
| AP (1) | AP2002002589A0 (es) |
| AR (1) | AR027337A1 (es) |
| AT (1) | ATE293624T1 (es) |
| AU (1) | AU2700201A (es) |
| BG (1) | BG106852A (es) |
| BR (1) | BR0107964A (es) |
| CA (1) | CA2398182C (es) |
| CO (1) | CO5261634A1 (es) |
| CZ (1) | CZ20022410A3 (es) |
| DE (1) | DE60110205T2 (es) |
| EA (1) | EA004885B1 (es) |
| EE (1) | EE200200425A (es) |
| ES (1) | ES2238415T3 (es) |
| GE (1) | GEP20043302B (es) |
| GT (1) | GT200100022A (es) |
| HN (1) | HN2001000019A (es) |
| HU (1) | HUP0204262A2 (es) |
| IL (1) | IL150641A0 (es) |
| IS (1) | IS6421A (es) |
| MA (1) | MA26870A1 (es) |
| MX (1) | MXPA02007419A (es) |
| NO (1) | NO20023613L (es) |
| NZ (1) | NZ519547A (es) |
| OA (1) | OA12169A (es) |
| PA (1) | PA8511201A1 (es) |
| PE (1) | PE20011058A1 (es) |
| PL (1) | PL357995A1 (es) |
| PT (1) | PT1252158E (es) |
| SK (1) | SK10142002A3 (es) |
| SV (1) | SV2002000299A (es) |
| TN (1) | TNSN01020A1 (es) |
| TR (1) | TR200201880T2 (es) |
| UY (1) | UY26569A1 (es) |
| WO (1) | WO2001057036A1 (es) |
| ZA (1) | ZA200206033B (es) |
Families Citing this family (43)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1121111T3 (da) * | 1998-10-15 | 2010-05-31 | Imp Innovations Ltd | Forbindelser til behandling af vægttab |
| US20010033861A1 (en) * | 2000-01-28 | 2001-10-25 | Lasic Danilo D. | Liposomes containing an entrapped compound in supersaturated solution |
| WO2002022583A2 (en) * | 2000-09-18 | 2002-03-21 | E. I. Du Pont De Nemours And Company | Pyridinyl amides and imides for use as fungicides |
| PL364135A1 (en) | 2001-01-31 | 2004-12-13 | Pfizer Products Inc. | Nicotinamide biaryl derivatives useful as inhibitors of pde4 isozymes |
| BR0116850A (pt) | 2001-01-31 | 2004-02-25 | Pfizer Prod Inc | Derivados de amida de ácido tiazolil-, oxazolil-, pirrolil- e imidazolil- úteis como inibidores de isoenzimas de pde4 |
| US7250518B2 (en) | 2001-01-31 | 2007-07-31 | Pfizer Inc. | Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4861891A (en) * | 1988-08-31 | 1989-08-29 | Pfizer Inc. | Antidepressant N-substituted nicotinamide compounds |
| TW429148B (en) | 1995-10-27 | 2001-04-11 | Pfizer | Pharmaceutical agents for the treatment of acute and chronic inflammatory diseases |
| EA003528B1 (ru) | 1997-04-04 | 2003-06-26 | Пфайзер Продактс Инк. | Производные никотинамида, их применение, фармацевтическая композиция, способ лечения и способ ингибирования изоферментов фдэ4 d |
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- 2001-01-30 MX MXPA02007419A patent/MXPA02007419A/es active IP Right Grant
- 2001-01-30 AU AU27002/01A patent/AU2700201A/en not_active Abandoned
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