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HK1209748B - 用於製備整合酶抑制劑的方法和中間產物 - Google Patents

用於製備整合酶抑制劑的方法和中間產物 Download PDF

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Publication number
HK1209748B
HK1209748B HK15110645.1A HK15110645A HK1209748B HK 1209748 B HK1209748 B HK 1209748B HK 15110645 A HK15110645 A HK 15110645A HK 1209748 B HK1209748 B HK 1209748B
Authority
HK
Hong Kong
Prior art keywords
compound
formula
salt
mixture
converting
Prior art date
Application number
HK15110645.1A
Other languages
German (de)
English (en)
French (fr)
Other versions
HK1209748A1 (zh
Inventor
Pcion Dominika
Tomasi Carrie
Charles Whitcomb Mark
D. Dowdy Eric
Fu Wenyi
Macleod Patricia
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Priority claimed from PCT/US2013/053295 external-priority patent/WO2014022707A1/en
Publication of HK1209748A1 publication Critical patent/HK1209748A1/zh
Publication of HK1209748B publication Critical patent/HK1209748B/zh

Links

HK15110645.1A 2012-08-03 2013-08-01 用於製備整合酶抑制劑的方法和中間產物 HK1209748B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261679475P 2012-08-03 2012-08-03
US61/679,475 2012-08-03
PCT/US2013/053295 WO2014022707A1 (en) 2012-08-03 2013-08-01 Process and intermediates for preparing integrase inhibitors

Publications (2)

Publication Number Publication Date
HK1209748A1 HK1209748A1 (zh) 2016-04-08
HK1209748B true HK1209748B (zh) 2017-12-08

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