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HK1240916A1 - Fused pentacyclic imidazole derivatives - Google Patents

Fused pentacyclic imidazole derivatives Download PDF

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Publication number
HK1240916A1
HK1240916A1 HK18100075.8A HK18100075A HK1240916A1 HK 1240916 A1 HK1240916 A1 HK 1240916A1 HK 18100075 A HK18100075 A HK 18100075A HK 1240916 A1 HK1240916 A1 HK 1240916A1
Authority
HK
Hong Kong
Prior art keywords
disorders
imidazole derivatives
fused pentacyclic
pentacyclic imidazole
derivatives
Prior art date
Application number
HK18100075.8A
Other languages
Chinese (zh)
Other versions
HK1240916B (en
Inventor
Teresa DE HARO GARCIA
Michael Deligny
Jag Paul Heer
Joanna Rachel Quincey
Mengyang XUAN
Zhaoning Zhu
Daniel Christopher Brookings
Mark Daniel Calmiano
Yves EVRARD
Martin Clive Hutchings
James Andrew Johnson
Sophie JADOT
Jean KEYAERTS
Malcolm Mac Coss
Matthew Duncan Selby
Michael Alan SHAW
Dominique Louis Léon SWINNEN
Laurent Schio
Yann Foricher
Bruno Filoche-Romme
Original Assignee
Ucb Biopharma Sprl
Sanofi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Biopharma Sprl, Sanofi filed Critical Ucb Biopharma Sprl
Publication of HK1240916A1 publication Critical patent/HK1240916A1/en
Publication of HK1240916B publication Critical patent/HK1240916B/en

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Abstract

A series of fused pentacyclic imidazole derivatives, being potent modulators of human TNFa activity, are accordingly of benefit in the treatment and/or prevention of various human ailments, including autoimmune and inflammatory disorders; neurological and neurodegenerative disorders; pain and nociceptive disorders; cardiovascular disorders; metabolic disorders; ocular disorders; and oncological disorders. In particular, the present invention is concerned with 6,7-dihydro-7,14-methanobenzimidazo[1,2-b][2,5]benzodiazocin-5(14H)-one derivatives and analogs thereof.
HK18100075.8A 2014-10-03 2015-10-02 Fused pentacyclic imidazole derivatives HK1240916B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14290299.8 2014-10-03
EP15162641.3 2015-04-07
EP15171036.5 2015-06-08

Publications (2)

Publication Number Publication Date
HK1240916A1 true HK1240916A1 (en) 2018-06-01
HK1240916B HK1240916B (en) 2022-02-11

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