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HK1114080B - 同素環和雜環化合物適合作為膽固醇酯轉運蛋白(cetp)抑制劑 - Google Patents

同素環和雜環化合物適合作為膽固醇酯轉運蛋白(cetp)抑制劑 Download PDF

Info

Publication number
HK1114080B
HK1114080B HK08109606.9A HK08109606A HK1114080B HK 1114080 B HK1114080 B HK 1114080B HK 08109606 A HK08109606 A HK 08109606A HK 1114080 B HK1114080 B HK 1114080B
Authority
HK
Hong Kong
Prior art keywords
fluoro
phenyl
trifluoromethyl
phenylethyl
tetrafluoroethoxy
Prior art date
Application number
HK08109606.9A
Other languages
German (de)
English (en)
French (fr)
Other versions
HK1114080A1 (zh
Inventor
Mark E. Salvati
Heather Finlay
Bang-Chi Chen
Lalgudi S. Harikrishnan
Ji Jiang
James A. Johnson
Muthoni G. Kamau
Michael R. Lawrence
Jianqing Li
John Lloyd
Michael Matthew Miller
Zulan Pi
Jennifer X. Qiao
Richard Rampulla
Tammy C. Wang
Yufeng Wang
Wu Yang
Jacques Y. Roberge
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/558,979 external-priority patent/US7790770B2/en
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of HK1114080A1 publication Critical patent/HK1114080A1/zh
Publication of HK1114080B publication Critical patent/HK1114080B/zh

Links

HK08109606.9A 2005-11-23 2006-11-16 同素環和雜環化合物適合作為膽固醇酯轉運蛋白(cetp)抑制劑 HK1114080B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US73937405P 2005-11-23 2005-11-23
US60/739,374 2005-11-23
US11/558,979 US7790770B2 (en) 2005-11-23 2006-11-13 Heterocyclic CETP inhibitors
US11/558,979 2006-11-13
PCT/US2006/060958 WO2007062308A2 (en) 2005-11-23 2006-11-16 Homo- and heterocyclic compounds suitable as cetp inhibitors

Publications (2)

Publication Number Publication Date
HK1114080A1 HK1114080A1 (zh) 2008-10-24
HK1114080B true HK1114080B (zh) 2011-12-09

Family

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HK1114080B (zh) 同素環和雜環化合物適合作為膽固醇酯轉運蛋白(cetp)抑制劑